Sfoglia per Autore
Quinoxaline chemistry. Part 11. 3-phenyl-2[phenoxy- and phenoxymethyl]-6(7) or 6,8-substituted quinoxalines and N-[4-(6(7)-substituted or 6,8-disubstituted-3-phenylquinoxalin-2-yl)hydroxy or hydroxymethyl]benzoylglutamates. Synthesis and evaluation of in
1998 Corona, P; Vitale, G; Loriga, M; Paglietti, G; Costi, Maria Paola
3-Aminophenylboronic acid derivative inhibitors of beta-lactamases, their preparation, and their therapeutic use.
1998 SHOICHET BRIAN, K.; Costi, Maria Paola; Tondi, Donatella
Thymidylate Synthase as a potential new target in drug resistance antimicrobial therapy.
1999 Costi, Maria Paola; A., Gelain; I., Cardilicchio; Soragni, Fabrizia; Rinaldi, Marcella; Pecorari, Piergiorgio; Tondi, Donatella; D. V., Santi
Structure-based discovery and in-parallel optimization of novel competitive inhibitors of thymidylate synthase
1999 Tondi, Donatella; U., Slomczynska; Costi, Maria Paola; Dm, Watterson; Ghelli, Stefano; Bk, Shoichet
Separation, structural determination and biological evaluation of the thymidylate synthase inhibitor 3,3-di(4'-hydroxyphenyl)-6(7)-chloro-1-oxo-1H,3H-naphtho[1,8-cd]pyran
1999 Costi, Maria Paola; Tondi, Donatella; Pecorari, Piergiorgio; Rinaldi, M; Celentano, G; Ghelli, Stefano; Antolini, L; Barlocco, Daniela
Phthalein derivatives as a new tool for selectivity in thymidylate synthase inhibition
1999 Costi, Maria Paola; Rinaldi, Marcella; Tondi, Donatella; Pecorari, Piergiorgio; Barlocco, Daniela; Ghelli, Stefano; Rm, Stroud; Dv, Santi; Tj, Stout; C., Musiu; Em, Marangiu; A., Pani; D., Congiu; Ga, Loi; P., La Colla
Structure-based design of inhibitors specific for bacterial thymidylate synthase
1999 Tj, Stout; Tondi, Donatella; Rinaldi, Marcella; Barlocco, Daniela; Pecorari, Piergiorgio; Dv, Santi; I., Kuntz; Rm, Stroud; Costi, Maria Paola; Bk, Shoichet
Structure based design and combinatorial optimization of novel Thymidylate synthase inhibitors. Meeting Abstract : 217th ACS National Meeting, Chicago March 1999
1999 Tondi, Donatella; Slomcynska, U.; Ghelli, Stefano; Watterson, D. M.; Costi, Maria Paola; Shoichet, B. K.
Sulfonamide Boronic Acid Inhibitors of AmpC b-lactamase to Reverse Bacterial Resistance to b-lactam Antibiotics.
1999 Shoichet, B. K.; Tondi, Donatella; Costi, Maria Paola; M., P.
Amide Boronic Acid Inhibitors of AmpC b-lactamase to Reverse Bacterial Resistance to b-lactam Antibiotics.
1999 Shoichet, B. K.; Tondi, Donatella; Costi, Maria Paola; M., P.
Phenylboronic acid derivative inhibitors of β-lactamases, their preparation, pharmaceutical compositions, and therapeutic use
1999 Shoichet, B K; Costi, Maria Paola; Tondi, Donatella
Structure-Based Design and In Parallel Synthesis of Boronic Acid Inhibitors of AmpC 61538;-Lactamase
2000 Tondi, Donatella; Powers, R.; Caselli, Emilia; Costi, Maria Paola; Shoichet, B. K.
Studi termodinamici e strutturali dell’interazione tra derivati densilici e Timidilato Sintasi Batteriche
2000 Tondi, Donatella; Venturelli, Alberto; Skinner, M. A.; Brown, K.; Costi, Maria Paola
Phenylboronic acid derivative inhibitors of ?-lactamases, their preparation, pharmaceutical compositions, and therapeutic use.
2000 Shoichet, B. K.; Costi, Maria Paola; Tondi, Donatella
Structures and reactivities of 1-oxo-cycloalkan-2-ylidenacetic acids. A 1H-NMR, modeling and photochemical study
2000 S., Ghelli; L., Toma; D., Barlocco; Costi, Maria Paola; Ponterini, Glauco
3-Aminophenylboronic acid derivative inhibitors of β-lactamases, their preparation, and their therapeutic use
2000 Shoichet, B. K.; Costi, Maria Paola; Tondi, Donatella
Probing Molecular Recognition of Dansyl Derivatives vs Bacterial Thymidylate Synthase (TS)
2001 Tondi, Donatella; Calò, S.; Fritz, T.; Stroud, R.; Costi, Maria Paola
Structural and thermodynamic combined studies for inhibitors binding to Thymidylate Synthase
2001 Venturelli, Alberto; Tondi, Donatella; Skinner, M. A.; Brown, K. A.; Ponterini, Glauco; Costi, Maria Paola
Structure-based design and solid phase synthesis of novel AmpC b-lactamase inhibitors
2001 Tondi, Donatella; Powers, R.; Caselli, E.; Costi, M. P.; Shoichet, B. K.
Enhancement of the drug discovery process by integration of Structure-based drug design and combinatorial chemistry
2001 Tondi, Donatella; Costi, Maria Paola
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