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Update on antifolate drugs targets 1-gen-2001 Costi, Maria Paola; Ferrari, Stefania
Predicting and harnessing protein flexibility in the design of species-specific inhibitors of thymidylate synthase 1-gen-2001 Ta, Fritz; Tondi, Donatella; J., FINER MOORE; Costi, Maria Paola; Rm, Stroud
Structure-based design and in-parallel synthesis of inhibitors of AmpC β-lactamase 1-gen-2001 Tondi, Donatella; Ra, Powers; Caselli, Emilia; Mc, Negri; J., Blazquez; Costi, Maria Paola; Bk, Shoichet
Dal Ligand based design di inibitori della Timidilato Sintasi all'Analisi Comparativa dei Complessi Enzima-Inibitore 1-gen-2002 Costi, Maria Paola; Ferrari, Stefania; Pecorari, Piergiorgio; Rinaldi, Marcella; Tondi, Donatella; Venturelli, Alberto; Wade, R. C.
Structure-based studies on species-specific inhibition of thymidylate synthase 1-gen-2002 Costi, Maria Paola; Tondi, Donatella; Rinaldi, Marcella; Barlocco, Daniela; Pecorari, Piergiorgio; Soragni, Fabrizia; Venturelli, Alberto; Stroud, Rm
Drug resistance - Developing targets and strategies in drug resistance - Preface 1-gen-2002 Costi, Maria Paola
Structure-based design and in parallel synthesis of boronic acid inhibitors of AmpC beta-lactamase 1-gen-2002 Tondi, Donatella; Costi, Maria Paola; B. K., Shoichet
Inhibitor Specificity via Protein Dynamics. Insights from the Design of Antibacterial Agents Targeted Against Thymidylate Synthase 1-gen-2003 Ferrari, Stefania; Costi, Maria Paola; Wade, R. C.
Ortho-halogen naphthaleins as specific inhibitors of Lactobacillus casei thymidylate synthase. Conformational properties and biological activity 1-gen-2003 S., Ghelli; M., Rinaldi; D., Barlocco; A., Gelain; P., Pecorari; Tondi, Donatella; Rastelli, Giulio; Costi, Maria Paola
Developing New beta-Lactamase Inhibitors Through Structure-Based Design and Pharmacokinetic Improvement 1-gen-2003 Venturelli, Alberto; B., Shoichet; Prati, Fabio; Cannazza, Giuseppe; Costi, Maria Paola
From ligand-based design to Hit validation of new thymidylate synthase inhibitors 1-gen-2003 Costi, Maria Paola; Ferrari, Stefania; Rinaldi, Marcella; Tondi, Donatella; Wade, R. C.
Quinoxaline chemistry. Part 15. 4-[2-Quinoxalylmethylenimino]- benzoylglutamates and -benzoates, 4-[2-quinoxalylmethyl-N-methylamino]- benzoylglutamates as analogues of classical antifolate agents. Synthesis, elucidation of structures and in vitro evaluation of antifolate and anticancer activities 1-gen-2003 Loriga, M.; Piras, S.; Paglietti, G.; Costi, Maria Paola; Venturelli, Alberto
Saturation site-directed mutagenesis of Lactobacillus casei Thymidylate synthase. Mutagenesis strategy and replacement sets of Pro-196 and Pro-197 1-gen-2003 Paconowska, D. G; Carreras, M. A.; Costi, Maria Paola; Santi, D. V.
Aza-boronic acids as non-beta-lactam inhibitors of AmpC-beta-lactamase 1-gen-2004 Buzzoni, V.; Blazquez, J.; Ferrari, Stefania; Calo, S.; Venturelli, A.; Costi, Maria Paola
Medicinal chemistry in parasitology 1-gen-2004 Costi, Maria Paola; Ferrari, Stefania; Rastelli, Giulio
“A step further in the discovery of phthalein derivatives as Thymidylate Synthase inhibitors” 1-gen-2004 Calo', Samuele; Tondi, Donatella; Venturelli, A.; Ferrari, Stefania; Pecorari, Piergiorgio; Rinaldi, Marcella; Ghelli, S.; Costi, Maria Paola
Rapid-Throughput Technologies Applied to the Discovery of New Hits against Thymidylate synthase Enzymes 1-gen-2004 Ferrari, Stefania; Malaguti, E; Calò, S; Tondi, Donatella; Venturelli, Alberto; Costi, Maria Paola
Structure-Based Optimization of a Non-β-lactam Lead Results in Inhibitors That Do Not Up-Regulate β-Lactamase Expression in Cell Culture 1-gen-2005 Tondi, Donatella; Federica, Morandi; Richard, Bonnet; Costi, Maria Paola; Brian K., Shoichet
Second Joint Italian-Swiss Meeting on Medicinal Chemistry , Italy, Modena 19-20 February 2005. 1-gen-2005 Brasili, Livio; Benvenuti, Stefania; Costantino, Luca; Costi, Maria Paola; Philipp, Floersheim; Franchini, Silvia; Gamberini, Gianfranco; Parenti, Carlo; Rastelli, Giulio; Rustichelli, Cecilia; Tait, Annalisa; Tondi, Donatella
Crystallographic studies of novel inhibitors of [beta]-lactamases 1-gen-2005 Tondi, Donatella; Venturelli, Alberto; Morandi, Federica; Bonnet, Richard; Shoichet, Brian K.; Costi, Maria Paola
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