Sfoglia per Autore
Conformational analysis of phthalein derivatives acting as thymidylate synthase inhibitors by means of 1H NMR and quantum chemical calculations
1996 S., Ghelli; Rastelli, Giulio; D., Barlocco; M., Rinaldi; Tondi, Donatella; P., Pecorari; Costi, Maria Paola
Naphthalimido Derivatives as Antifolate Thymidylate Synthase Inhibitors
1996 Costi, Mp; Tondi, Donatella; Rinaldi, M; Barlocco, D; Cignarella, G; Santi, Dv; Musiu, C; Pudu, I; Vacca, G; Lacolla, P.
"Structure-Based Discovery & In parallel Optimization of Novel Inhibitors of Thymidylate Synthase"
1997 Tondi, D.; Slomczynska, U.; Ghelli, S.; Wattweson, D. M.; Costi, M. P.; Shoichet, B. K.
1H-NMR conformational studies of some phtalein derivatives acting as thymidylate synthase inhibitors
1997 S., Ghelli; Costi, Maria Paola; D., Barlocco; M., Rinaldi; Tondi, Donatella; P., Pecorari; Rastelli, Giulio
Mono- and Disubstituted-3,8-diazabicyclo[3.2.1]octane Derivatives as Analgesics Structurally Related to Epibatidine: Synthesis, Activity, and Modeling.
1998 Barlocco, Daniela; Cignarella, Giorgio; Tondi, Donatella; Vianello, Paola; Villa, Stefania; Bartolini, Alessandro; Ghelardini, Carla; Galeotti, Nicoletta; ANDERSON DAVID, J. KUNTZWEILER THERESA A.; Colombo, Diego; Toma, Lucio
3-Aminophenylboronic acid derivative inhibitors of beta-lactamases, their preparation, and their therapeutic use.
1998 SHOICHET BRIAN, K.; Costi, Maria Paola; Tondi, Donatella
Thymidylate Synthase as a potential new target in drug resistance antimicrobial therapy.
1999 Costi, Maria Paola; A., Gelain; I., Cardilicchio; Soragni, Fabrizia; Rinaldi, Marcella; Pecorari, Piergiorgio; Tondi, Donatella; D. V., Santi
Structure based design and combinatorial optimization of novel Thymidylate synthase inhibitors. Meeting Abstract : 217th ACS National Meeting, Chicago March 1999
1999 Tondi, Donatella; Slomcynska, U.; Ghelli, Stefano; Watterson, D. M.; Costi, Maria Paola; Shoichet, B. K.
Structure-based design of inhibitors specific for bacterial thymidylate synthase
1999 Tj, Stout; Tondi, Donatella; Rinaldi, Marcella; Barlocco, Daniela; Pecorari, Piergiorgio; Dv, Santi; I., Kuntz; Rm, Stroud; Costi, Maria Paola; Bk, Shoichet
Separation, structural determination and biological evaluation of the thymidylate synthase inhibitor 3,3-di(4'-hydroxyphenyl)-6(7)-chloro-1-oxo-1H,3H-naphtho[1,8-cd]pyran
1999 Costi, Maria Paola; Tondi, Donatella; Pecorari, Piergiorgio; Rinaldi, M; Celentano, G; Ghelli, Stefano; Antolini, L; Barlocco, Daniela
Structure-based discovery and combinatorial optimization of novel competitive inhibitors of thymidylate synthase
1999 Sholchet, Bk; Tondi, Donatella; Slomczynska, U.
Phthalein derivatives as a new tool for selectivity in thymidylate synthase inhibition
1999 Costi, Maria Paola; Rinaldi, Marcella; Tondi, Donatella; Pecorari, Piergiorgio; Barlocco, Daniela; Ghelli, Stefano; Rm, Stroud; Dv, Santi; Tj, Stout; C., Musiu; Em, Marangiu; A., Pani; D., Congiu; Ga, Loi; P., La Colla
Structure-based discovery and in-parallel optimization of novel competitive inhibitors of thymidylate synthase
1999 Tondi, Donatella; U., Slomczynska; Costi, Maria Paola; Dm, Watterson; Ghelli, Stefano; Bk, Shoichet
Sulfonamide Boronic Acid Inhibitors of AmpC b-lactamase to Reverse Bacterial Resistance to b-lactam Antibiotics.
1999 Shoichet, B. K.; Tondi, Donatella; Costi, Maria Paola; M., P.
Phenylboronic acid derivative inhibitors of β-lactamases, their preparation, pharmaceutical compositions, and therapeutic use
1999 Shoichet, B K; Costi, Maria Paola; Tondi, Donatella
Amide Boronic Acid Inhibitors of AmpC b-lactamase to Reverse Bacterial Resistance to b-lactam Antibiotics.
1999 Shoichet, B. K.; Tondi, Donatella; Costi, Maria Paola; M., P.
Phenylboronic acid derivative inhibitors of ?-lactamases, their preparation, pharmaceutical compositions, and therapeutic use.
2000 Shoichet, B. K.; Costi, Maria Paola; Tondi, Donatella
Studi termodinamici e strutturali dell’interazione tra derivati densilici e Timidilato Sintasi Batteriche
2000 Tondi, Donatella; Venturelli, Alberto; Skinner, M. A.; Brown, K.; Costi, Maria Paola
Structure-Based Design and In Parallel Synthesis of Boronic Acid Inhibitors of AmpC 61538;-Lactamase
2000 Tondi, Donatella; Powers, R.; Caselli, Emilia; Costi, Maria Paola; Shoichet, B. K.
3-Aminophenylboronic acid derivative inhibitors of β-lactamases, their preparation, and their therapeutic use
2000 Shoichet, B. K.; Costi, Maria Paola; Tondi, Donatella
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Conformational analysis of phthalein derivatives acting as thymidylate synthase inhibitors by means of 1H NMR and quantum chemical calculations | 1-gen-1996 | S., Ghelli; Rastelli, Giulio; D., Barlocco; M., Rinaldi; Tondi, Donatella; P., Pecorari; Costi, Maria Paola | |
Naphthalimido Derivatives as Antifolate Thymidylate Synthase Inhibitors | 1-gen-1996 | Costi, Mp; Tondi, Donatella; Rinaldi, M; Barlocco, D; Cignarella, G; Santi, Dv; Musiu, C; Pudu, I; Vacca, G; Lacolla, P. | |
"Structure-Based Discovery & In parallel Optimization of Novel Inhibitors of Thymidylate Synthase" | 1-gen-1997 | Tondi, D.; Slomczynska, U.; Ghelli, S.; Wattweson, D. M.; Costi, M. P.; Shoichet, B. K. | |
1H-NMR conformational studies of some phtalein derivatives acting as thymidylate synthase inhibitors | 1-gen-1997 | S., Ghelli; Costi, Maria Paola; D., Barlocco; M., Rinaldi; Tondi, Donatella; P., Pecorari; Rastelli, Giulio | |
Mono- and Disubstituted-3,8-diazabicyclo[3.2.1]octane Derivatives as Analgesics Structurally Related to Epibatidine: Synthesis, Activity, and Modeling. | 1-gen-1998 | Barlocco, Daniela; Cignarella, Giorgio; Tondi, Donatella; Vianello, Paola; Villa, Stefania; Bartolini, Alessandro; Ghelardini, Carla; Galeotti, Nicoletta; ANDERSON DAVID, J. KUNTZWEILER THERESA A.; Colombo, Diego; Toma, Lucio | |
3-Aminophenylboronic acid derivative inhibitors of beta-lactamases, their preparation, and their therapeutic use. | 16-dic-1998 | SHOICHET BRIAN, K.; Costi, Maria Paola; Tondi, Donatella | |
Thymidylate Synthase as a potential new target in drug resistance antimicrobial therapy. | 1-gen-1999 | Costi, Maria Paola; A., Gelain; I., Cardilicchio; Soragni, Fabrizia; Rinaldi, Marcella; Pecorari, Piergiorgio; Tondi, Donatella; D. V., Santi | |
Structure based design and combinatorial optimization of novel Thymidylate synthase inhibitors. Meeting Abstract : 217th ACS National Meeting, Chicago March 1999 | 1-gen-1999 | Tondi, Donatella; Slomcynska, U.; Ghelli, Stefano; Watterson, D. M.; Costi, Maria Paola; Shoichet, B. K. | |
Structure-based design of inhibitors specific for bacterial thymidylate synthase | 1-gen-1999 | Tj, Stout; Tondi, Donatella; Rinaldi, Marcella; Barlocco, Daniela; Pecorari, Piergiorgio; Dv, Santi; I., Kuntz; Rm, Stroud; Costi, Maria Paola; Bk, Shoichet | |
Separation, structural determination and biological evaluation of the thymidylate synthase inhibitor 3,3-di(4'-hydroxyphenyl)-6(7)-chloro-1-oxo-1H,3H-naphtho[1,8-cd]pyran | 1-gen-1999 | Costi, Maria Paola; Tondi, Donatella; Pecorari, Piergiorgio; Rinaldi, M; Celentano, G; Ghelli, Stefano; Antolini, L; Barlocco, Daniela | |
Structure-based discovery and combinatorial optimization of novel competitive inhibitors of thymidylate synthase | 1-gen-1999 | Sholchet, Bk; Tondi, Donatella; Slomczynska, U. | |
Phthalein derivatives as a new tool for selectivity in thymidylate synthase inhibition | 1-gen-1999 | Costi, Maria Paola; Rinaldi, Marcella; Tondi, Donatella; Pecorari, Piergiorgio; Barlocco, Daniela; Ghelli, Stefano; Rm, Stroud; Dv, Santi; Tj, Stout; C., Musiu; Em, Marangiu; A., Pani; D., Congiu; Ga, Loi; P., La Colla | |
Structure-based discovery and in-parallel optimization of novel competitive inhibitors of thymidylate synthase | 1-gen-1999 | Tondi, Donatella; U., Slomczynska; Costi, Maria Paola; Dm, Watterson; Ghelli, Stefano; Bk, Shoichet | |
Sulfonamide Boronic Acid Inhibitors of AmpC b-lactamase to Reverse Bacterial Resistance to b-lactam Antibiotics. | 16-dic-1999 | Shoichet, B. K.; Tondi, Donatella; Costi, Maria Paola; M., P. | |
Phenylboronic acid derivative inhibitors of β-lactamases, their preparation, pharmaceutical compositions, and therapeutic use | 16-dic-1999 | Shoichet, B K; Costi, Maria Paola; Tondi, Donatella | |
Amide Boronic Acid Inhibitors of AmpC b-lactamase to Reverse Bacterial Resistance to b-lactam Antibiotics. | 16-dic-1999 | Shoichet, B. K.; Tondi, Donatella; Costi, Maria Paola; M., P. | |
Phenylboronic acid derivative inhibitors of ?-lactamases, their preparation, pharmaceutical compositions, and therapeutic use. | 1-gen-2000 | Shoichet, B. K.; Costi, Maria Paola; Tondi, Donatella | |
Studi termodinamici e strutturali dell’interazione tra derivati densilici e Timidilato Sintasi Batteriche | 1-gen-2000 | Tondi, Donatella; Venturelli, Alberto; Skinner, M. A.; Brown, K.; Costi, Maria Paola | |
Structure-Based Design and In Parallel Synthesis of Boronic Acid Inhibitors of AmpC 61538;-Lactamase | 1-gen-2000 | Tondi, Donatella; Powers, R.; Caselli, Emilia; Costi, Maria Paola; Shoichet, B. K. | |
3-Aminophenylboronic acid derivative inhibitors of β-lactamases, their preparation, and their therapeutic use | 22-giu-2000 | Shoichet, B. K.; Costi, Maria Paola; Tondi, Donatella |
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