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Titolo Data di pubblicazione Autore(i) File
Probing Molecular Recognition of Dansyl Derivatives vs Bacterial Thymidylate Synthase (TS) 1-gen-2001 Tondi, Donatella; Calò, S.; Fritz, T.; Stroud, R.; Costi, Maria Paola
Structural and thermodynamic combined studies for inhibitors binding to Thymidylate Synthase 1-gen-2001 Venturelli, Alberto; Tondi, Donatella; Skinner, M. A.; Brown, K. A.; Ponterini, Glauco; Costi, Maria Paola
Structure-based design and solid phase synthesis of novel AmpC b-lactamase inhibitors 1-gen-2001 Tondi, Donatella; Powers, R.; Caselli, E.; Costi, M. P.; Shoichet, B. K.
Enhancement of the drug discovery process by integration of Structure-based drug design and combinatorial chemistry 1-gen-2001 Tondi, Donatella; Costi, Maria Paola
Predicting and harnessing protein flexibility in the design of species-specific inhibitors of thymidylate synthase 1-gen-2001 Ta, Fritz; Tondi, Donatella; J., FINER MOORE; Costi, Maria Paola; Rm, Stroud
Structure-based design and in-parallel synthesis of inhibitors of AmpC β-lactamase 1-gen-2001 Tondi, Donatella; Ra, Powers; Caselli, Emilia; Mc, Negri; J., Blazquez; Costi, Maria Paola; Bk, Shoichet
Structure-based design and in parallel synthesis of boronic acid inhibitors of AmpC beta-lactamase 1-gen-2002 Tondi, Donatella; Costi, Maria Paola; B. K., Shoichet
Dal Ligand based design di inibitori della Timidilato Sintasi all'Analisi Comparativa dei Complessi Enzima-Inibitore 1-gen-2002 Costi, Maria Paola; Ferrari, Stefania; Pecorari, Piergiorgio; Rinaldi, Marcella; Tondi, Donatella; Venturelli, Alberto; Wade, R. C.
Structure-based studies on species-specific inhibition of thymidylate synthase 1-gen-2002 Costi, Maria Paola; Tondi, Donatella; Rinaldi, Marcella; Barlocco, Daniela; Pecorari, Piergiorgio; Soragni, Fabrizia; Venturelli, Alberto; Stroud, Rm
From ligand-based design to Hit validation of new thymidylate synthase inhibitors 1-gen-2003 Costi, Maria Paola; Ferrari, Stefania; Rinaldi, Marcella; Tondi, Donatella; Wade, R. C.
Ortho-halogen naphthaleins as specific inhibitors of Lactobacillus casei thymidylate synthase. Conformational properties and biological activity 1-gen-2003 S., Ghelli; M., Rinaldi; D., Barlocco; A., Gelain; P., Pecorari; Tondi, Donatella; Rastelli, Giulio; Costi, Maria Paola
Rapid-Throughput Technologies Applied to the Discovery of New Hits against Thymidylate synthase Enzymes 1-gen-2004 Ferrari, Stefania; Malaguti, E; Calò, S; Tondi, Donatella; Venturelli, Alberto; Costi, Maria Paola
“A step further in the discovery of phthalein derivatives as Thymidylate Synthase inhibitors” 1-gen-2004 Calo', Samuele; Tondi, Donatella; Venturelli, A.; Ferrari, Stefania; Pecorari, Piergiorgio; Rinaldi, Marcella; Ghelli, S.; Costi, Maria Paola
Structure-Based Optimization of a Non-β-lactam Lead Results in Inhibitors That Do Not Up-Regulate β-Lactamase Expression in Cell Culture 1-gen-2005 Tondi, Donatella; Federica, Morandi; Richard, Bonnet; Costi, Maria Paola; Brian K., Shoichet
AmpC beta-lactamase in complex with 3-(3-nitro-phenylsulfamoyl)-thiophene-2-carboxylic acid 1-gen-2005 Tondi, Donatella
Structure-based inhibitor design vs. beta-lactamase 1-gen-2005 Shoichet, B; Tondi, Donatella; Morandi, F; Babaoglu, K.
Structure-based optimization of a non-beta-lactam lead results in inhibitors that do not up-regulate beta-lactamase expression in cell culture 1-gen-2005 Tondi, Donatella; Morandi, Federica; R., Bonnet; Costi, Maria Paola; Bk, Shoichet
Second Joint Italian-Swiss Meeting on Medicinal Chemistry , Italy, Modena 19-20 February 2005. 1-gen-2005 Brasili, Livio; Benvenuti, Stefania; Costantino, Luca; Costi, Maria Paola; Philipp, Floersheim; Franchini, Silvia; Gamberini, Gianfranco; Parenti, Carlo; Rastelli, Giulio; Rustichelli, Cecilia; Tait, Annalisa; Tondi, Donatella
Crystallographic studies of novel inhibitors of [beta]-lactamases 1-gen-2005 Tondi, Donatella; Venturelli, Alberto; Morandi, Federica; Bonnet, Richard; Shoichet, Brian K.; Costi, Maria Paola
Thymidylate synthase structure, function and implication in drug discovery 1-gen-2005 Costi, Maria Paola; Ferrari, Stefania; Venturelli, A; Calo, S; Tondi, Donatella; Barlocco, D.
Mostrati risultati da 21 a 40 di 110
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