BATTISTI, UMBERTO MARIA
BATTISTI, UMBERTO MARIA
Dipartimento di Scienze della Vita
7-Chloro-5-(furan-3-yl)-3-methyl-4H-benzo[e][1,2,4]thiadiazine 1,1-Dioxide as Positive Allosteric Modulator of α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor. The End of the Unsaturated-Inactive Paradigm?
2016-01-01 Citti, Cinzia; Battisti, UMBERTO MARIA; Cannazza, Giuseppe; Jozwiak, Krzysztof; Stasiak, Natalia; Puja, Giulia; Ravazzini, Federica; Ciccarella, Giuseppe; Braghiroli, Daniela; Parenti, Carlo; Troisi, Luigino; Zoli, Michele
BENZOTHIADIAZINES DERIVATIVES AS NOVEL ALLOSTERIC MODULATORS OF KAINIC ACID RECEPTORS
2022-01-01 Puja, G.; Ravazzini, F.; Losi, G.; Bardoni, R.; Battisti, U. M.; Citti, C.; Cannazza, G.
Design, stereoselective synthesis, configurational stability and biological activity of 7-chloro-9-(furan-3-yl)-2,3,3a,4-tetrahydro-1H-benzo[e]pyrrolo[2,1-c][1,2,4]thiadiazine 5,5-dioxide
2014-01-01 Carrozzo, Marina Maria; Battisti, UMBERTO MARIA; Cannazza, Giuseppe; Puja, Giulia; Ravazzini, Federica; Falchicchio, Aurelia; Perrone, Serena; Citti, Cinzia; Jozwiak, Krzysztof; Braghiroli, Daniela; Parenti, Carlo; Troisi, Luigino
Determination of kinetic parameters of enantiomerization of benzothiadiazines by DCXplorer
2010-01-01 CANNAZZA, Giuseppe; CARROZZO, Marina Maria; BATTISTI, UMBERTO MARIA; BRAGHIROLI, Daniela; PARENTI, Carlo; Troisi, Alessandro; Troisi, Luigino
Efficient synthesis of 5,6-dihydro-8H-[1,2,4]thiadiazino[6,5,4-de] phenanthridine 4,4-dioxide and 5,6-dihydro-8H-[1,2,4]-thiadiazino[6,5,4-ij] thieno[2,3-c]quinoline 4,4-dioxide
2012-01-01 Battisti, UMBERTO MARIA; Carrozzo, Marina Maria; Cannazza, Giuseppe; Braghiroli, Daniela; Parenti, Carlo; Brasili, Livio; Cinzia, Citti; Luigino, Troisi
Enantiomeric resolution of [(2,2-diphenyl-1,3-dioxolan-4-yl)methyl](2-phenoxyethyl)amine, a potent α1and 5-HT1Areceptor ligand: an in vitro and computational study
2015-01-01 Franchini, Silvia; Baraldi, Anna Maria; Sorbi, Claudia; Pellati, Federica; Cichero, Elena; Battisti, UMBERTO MARIA; Angeli, Piero; Cilia, Antonio; Brasili, Livio
Epimerization and hydrolysis of 3,6-dimethyl-2,3,5,6-tetrahydro[1,2,4]thiadiazino[6,5,4-hi]indole 1,1-dioxide
2010-01-01 Carrozzo, Marina Maria; Cannazza, Giuseppe; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Troisi, Luigino; Parenti, Carlo
Evaluation of stereo and chemical stability of chiral compounds
2011-01-01 Cannazza, Giuseppe; Battisti, UMBERTO MARIA; Carrozzo, Marina Maria; Brasili, Livio; Braghiroli, Daniela; Parenti, Carlo
A Metabolomic Approach Applied to a LiquidChromatography Coupled to High-ResolutionTandem Mass Spectrometry Method (HPLC-ESI-HRMS/MS): Towards the ComprehensiveEvaluation of the Chemical Composition ofCannabis Medicinal Extracts
2018-01-01 Citti, Cinzia; Battisti, Umberto Maria; Braghiroli, Daniela; Ciccarella, Giuseppe; Schmid, Martin; Vandelli, Maria Angela; Cannazza, Giuseppe
Molecular modeling studies, synthesis, configurational stability and biological activity of 8-chloro-2,3,5,6-tetrahydro-3,6-dimethyl-pyrrolo[1,2,3-de]-1,2,4-benzothiadiazine 1,1-dioxide
2011-01-01 Battisti, UMBERTO MARIA; Carrozzo, Marina Maria; Cannazza, Giuseppe; Puja, Giulia; Giulia, ; L., Troisi; Braghiroli, Daniela; Parenti, Carlo; K., Jozwiak
A New and Versatile Synthesis of 1,3-Dioxan-5-yl-pyrimidine and Purine Nucleoside Analogues
2015-01-01 Sorbi, Claudia; Prandi, Adolfo; Battisti, UMBERTO MARIA; Franchini, Silvia; Cornia, Andrea; Balzarini, Jan; Jeong, Lak Shin; Lee, Sang Kook; Song, Jayoung; Brasili, Livio
On-line racemization by high-performance liquid chromatography
2009-01-01 Cannazza, Giuseppe; Carrozzo, Marina Maria; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Parenti, Carlo
Quantitative analysis of acetylcholine in rat brain microdialysates by liquid chromatography coupled with electrospray ionization tandem mass spectrometry
2010-01-01 Carrozzo, Marina Maria; Cannazza, Giuseppe; Pinetti, Diego; DI VIESTI, Vittoria; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Parenti, Carlo; Baraldi, Mario
Regioselective cyclization of chloroacylaminobenzenesulfonamide derivatives
2012-01-01 Carrozzo, Marina Maria; Battisti, UMBERTO MARIA; Cannazza, Giuseppe; C., Citti; Parenti, Carlo; L., Troisi
Regioselective reduction of 3-substituted 2,3-dihydrobenzothiadiazines with borohydrides
2010-01-01 Battisti, UMBERTO MARIA; Cannazza, Giuseppe; M. M., Carrozzo; Braghiroli, Daniela; Parenti, Carlo; F., Rosato; L., Troisi
Scouting new sigma receptor ligands: Synthesis, pharmacological evaluation and molecular modeling of 1,3-dioxolane-based structures and derivatives
2016-01-01 Franchini, Silvia; Battisti, Umberto Maria; Prandi, Adolfo; Tait, Annalisa; Borsari, Chiara; Cichero, Elena; Fossa, Paola; Cilia, Antonio; Prezzavento, Orazio; Ronsisvalle, Simone; Aricò, Giuseppina; Parenti, Carmela; Brasili, Livio
Simultaneous Determination of Enantiomerizationand Hydrolysis Kinetic Parameters of ChiralN-Alkylbenzothiadiazine Derivatives
2010-01-01 Carrozzo, Marina Maria; Cannazza, Giuseppe; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Parenti, Carlo
Spiroxatrine derivatives towards 5-HT1A receptor selectivity
2020-01-01 Sorbi, C.; Tait, A.; Battisti, U. M.; Brasili, L.
Structure-Activity Relationship within a new series of σ1 and σ2 receptor ligands: identification of a novel σ2R agonist (BS148) with selective toxicity against metastatic melanoma
2017-01-01 Franchini, Silvia; Sorbi, Claudia; Battisti, Umberto Maria; Tait, Annalisa; Bencheva, Leda Ivanova; Cichero, Elena; Fossa, Paola; Cilia, Antonio; Prezzavento, Orazio; Ronsisvalle, Simone; Aricò, Giuseppina; Benassi, Luisa; Vaschieri, Cristina; Azzoni, Paola; Magnoni, Cristina; Brasili, Livio
Structure-affinity/activity relationships of 1,4-dioxa-spiro[4.5]decane based ligands at α1 and 5-HT1A receptors
2014-01-01 Franchini, Silvia; Battisti, UMBERTO MARIA; Baraldi, Anna Maria; Prandi, Adolfo; Fossa, Paola; Cichero, Elena; Tait, Annalisa; Sorbi, Claudia; Marucci, Gabriella; Cilia, Antonio; Pirona, Lorenza; Brasili, Livio
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 7-Chloro-5-(furan-3-yl)-3-methyl-4H-benzo[e][1,2,4]thiadiazine 1,1-Dioxide as Positive Allosteric Modulator of α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor. The End of the Unsaturated-Inactive Paradigm? | 1-gen-2016 | Citti, Cinzia; Battisti, UMBERTO MARIA; Cannazza, Giuseppe; Jozwiak, Krzysztof; Stasiak, Natalia; Puja, Giulia; Ravazzini, Federica; Ciccarella, Giuseppe; Braghiroli, Daniela; Parenti, Carlo; Troisi, Luigino; Zoli, Michele | |
| BENZOTHIADIAZINES DERIVATIVES AS NOVEL ALLOSTERIC MODULATORS OF KAINIC ACID RECEPTORS | 1-gen-2022 | Puja, G.; Ravazzini, F.; Losi, G.; Bardoni, R.; Battisti, U. M.; Citti, C.; Cannazza, G. | |
| Design, stereoselective synthesis, configurational stability and biological activity of 7-chloro-9-(furan-3-yl)-2,3,3a,4-tetrahydro-1H-benzo[e]pyrrolo[2,1-c][1,2,4]thiadiazine 5,5-dioxide | 1-gen-2014 | Carrozzo, Marina Maria; Battisti, UMBERTO MARIA; Cannazza, Giuseppe; Puja, Giulia; Ravazzini, Federica; Falchicchio, Aurelia; Perrone, Serena; Citti, Cinzia; Jozwiak, Krzysztof; Braghiroli, Daniela; Parenti, Carlo; Troisi, Luigino | |
| Determination of kinetic parameters of enantiomerization of benzothiadiazines by DCXplorer | 1-gen-2010 | CANNAZZA, Giuseppe; CARROZZO, Marina Maria; BATTISTI, UMBERTO MARIA; BRAGHIROLI, Daniela; PARENTI, Carlo; Troisi, Alessandro; Troisi, Luigino | |
| Efficient synthesis of 5,6-dihydro-8H-[1,2,4]thiadiazino[6,5,4-de] phenanthridine 4,4-dioxide and 5,6-dihydro-8H-[1,2,4]-thiadiazino[6,5,4-ij] thieno[2,3-c]quinoline 4,4-dioxide | 1-gen-2012 | Battisti, UMBERTO MARIA; Carrozzo, Marina Maria; Cannazza, Giuseppe; Braghiroli, Daniela; Parenti, Carlo; Brasili, Livio; Cinzia, Citti; Luigino, Troisi | |
| Enantiomeric resolution of [(2,2-diphenyl-1,3-dioxolan-4-yl)methyl](2-phenoxyethyl)amine, a potent α1and 5-HT1Areceptor ligand: an in vitro and computational study | 1-gen-2015 | Franchini, Silvia; Baraldi, Anna Maria; Sorbi, Claudia; Pellati, Federica; Cichero, Elena; Battisti, UMBERTO MARIA; Angeli, Piero; Cilia, Antonio; Brasili, Livio | |
| Epimerization and hydrolysis of 3,6-dimethyl-2,3,5,6-tetrahydro[1,2,4]thiadiazino[6,5,4-hi]indole 1,1-dioxide | 1-gen-2010 | Carrozzo, Marina Maria; Cannazza, Giuseppe; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Troisi, Luigino; Parenti, Carlo | |
| Evaluation of stereo and chemical stability of chiral compounds | 1-gen-2011 | Cannazza, Giuseppe; Battisti, UMBERTO MARIA; Carrozzo, Marina Maria; Brasili, Livio; Braghiroli, Daniela; Parenti, Carlo | |
| A Metabolomic Approach Applied to a LiquidChromatography Coupled to High-ResolutionTandem Mass Spectrometry Method (HPLC-ESI-HRMS/MS): Towards the ComprehensiveEvaluation of the Chemical Composition ofCannabis Medicinal Extracts | 1-gen-2018 | Citti, Cinzia; Battisti, Umberto Maria; Braghiroli, Daniela; Ciccarella, Giuseppe; Schmid, Martin; Vandelli, Maria Angela; Cannazza, Giuseppe | |
| Molecular modeling studies, synthesis, configurational stability and biological activity of 8-chloro-2,3,5,6-tetrahydro-3,6-dimethyl-pyrrolo[1,2,3-de]-1,2,4-benzothiadiazine 1,1-dioxide | 1-gen-2011 | Battisti, UMBERTO MARIA; Carrozzo, Marina Maria; Cannazza, Giuseppe; Puja, Giulia; Giulia, ; L., Troisi; Braghiroli, Daniela; Parenti, Carlo; K., Jozwiak | |
| A New and Versatile Synthesis of 1,3-Dioxan-5-yl-pyrimidine and Purine Nucleoside Analogues | 1-gen-2015 | Sorbi, Claudia; Prandi, Adolfo; Battisti, UMBERTO MARIA; Franchini, Silvia; Cornia, Andrea; Balzarini, Jan; Jeong, Lak Shin; Lee, Sang Kook; Song, Jayoung; Brasili, Livio | |
| On-line racemization by high-performance liquid chromatography | 1-gen-2009 | Cannazza, Giuseppe; Carrozzo, Marina Maria; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Parenti, Carlo | |
| Quantitative analysis of acetylcholine in rat brain microdialysates by liquid chromatography coupled with electrospray ionization tandem mass spectrometry | 1-gen-2010 | Carrozzo, Marina Maria; Cannazza, Giuseppe; Pinetti, Diego; DI VIESTI, Vittoria; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Parenti, Carlo; Baraldi, Mario | |
| Regioselective cyclization of chloroacylaminobenzenesulfonamide derivatives | 1-gen-2012 | Carrozzo, Marina Maria; Battisti, UMBERTO MARIA; Cannazza, Giuseppe; C., Citti; Parenti, Carlo; L., Troisi | |
| Regioselective reduction of 3-substituted 2,3-dihydrobenzothiadiazines with borohydrides | 1-gen-2010 | Battisti, UMBERTO MARIA; Cannazza, Giuseppe; M. M., Carrozzo; Braghiroli, Daniela; Parenti, Carlo; F., Rosato; L., Troisi | |
| Scouting new sigma receptor ligands: Synthesis, pharmacological evaluation and molecular modeling of 1,3-dioxolane-based structures and derivatives | 1-gen-2016 | Franchini, Silvia; Battisti, Umberto Maria; Prandi, Adolfo; Tait, Annalisa; Borsari, Chiara; Cichero, Elena; Fossa, Paola; Cilia, Antonio; Prezzavento, Orazio; Ronsisvalle, Simone; Aricò, Giuseppina; Parenti, Carmela; Brasili, Livio | |
| Simultaneous Determination of Enantiomerizationand Hydrolysis Kinetic Parameters of ChiralN-Alkylbenzothiadiazine Derivatives | 1-gen-2010 | Carrozzo, Marina Maria; Cannazza, Giuseppe; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Parenti, Carlo | |
| Spiroxatrine derivatives towards 5-HT1A receptor selectivity | 1-gen-2020 | Sorbi, C.; Tait, A.; Battisti, U. M.; Brasili, L. | |
| Structure-Activity Relationship within a new series of σ1 and σ2 receptor ligands: identification of a novel σ2R agonist (BS148) with selective toxicity against metastatic melanoma | 1-gen-2017 | Franchini, Silvia; Sorbi, Claudia; Battisti, Umberto Maria; Tait, Annalisa; Bencheva, Leda Ivanova; Cichero, Elena; Fossa, Paola; Cilia, Antonio; Prezzavento, Orazio; Ronsisvalle, Simone; Aricò, Giuseppina; Benassi, Luisa; Vaschieri, Cristina; Azzoni, Paola; Magnoni, Cristina; Brasili, Livio | |
| Structure-affinity/activity relationships of 1,4-dioxa-spiro[4.5]decane based ligands at α<alpha>1 and 5-HT1A receptors | 1-gen-2014 | Franchini, Silvia; Battisti, UMBERTO MARIA; Baraldi, Anna Maria; Prandi, Adolfo; Fossa, Paola; Cichero, Elena; Tait, Annalisa; Sorbi, Claudia; Marucci, Gabriella; Cilia, Antonio; Pirona, Lorenza; Brasili, Livio |