CASELLI, Emilia
Dettaglio
CASELLI, Emilia
Dipartimento di Scienze della Vita
Pubblicazioni
Risultati 1 - 20 di 52 (tempo di esecuzione: 0.0 secondi).
Titolo | Data di pubblicazione | Autore(i) | |
---|---|---|---|
1 | 1,2,3-Triazolylmethaneboronate: A Structure Activity Relationship Study of a Class of β-Lactamase Inhibitors against Acinetobacter baumannii Cephalosporinase | 2020 | Caselli, E.; Fini, F.; Introvigne, M. L.; Stucchi, M.; Taracila, M. A.; Fish, E. R.; Smolen, K. A.; Rather, P. N.; Powers, R. A.; Wallar, B. J.; Bonomo, R. A.; Prati, F. |
2 | Acetamidomethaneboronic acids bearing the R1 side chains of beta-lactams as inhibitors of beta-lactamase enzymes | - | L. C., Blaszczak; Caselli, Emilia; Prati, Fabio; B. K., Shoichet |
3 | Acido alfa-Acetammido-alfa-Fenilmetanboronico come Agente Derivatizzante Chirale per la Determinazione dell’Eccesso Enantiomerico di 1,2-Dioli | 2003 | B., Bonfiglio; Caselli, Emilia; Forni, Arrigo; Danieli, Chiara; Prati, Fabio |
4 | Biocatalytic asymmetric synthesis of (S)- and (R)-Timolol | 2004 | Tosi, Giovanni; F., Zironi; Caselli, Emilia; Forni, Arrigo; Prati, Fabio |
5 | Biochemical and structural analysis of inhibitors targeting the ADC-7 cephalosporinase of Acinetobacter baumannii | 2014 | R. A., Powers; H. C., Swanson; M. A., Taracila; N. W., Florek; Romagnoli, Chiara; Caselli, Emilia; Prati, Fabio; R. A., Bonomo; B. J., Wallar |
6 | Boronic acid inhibitors of beta-lactamases as therapeutic agents in treatment of antibiotic-resistant infection diseases | - | Prati, Fabio; Caselli, Emilia |
7 | Boronic acid transition state inhibitors active against KPC and other class a β-lactamases: Structure-activity relationships as a guide to inhibitor design | 2016 | Rojas, Laura J.; Taracila, Magdalena A.; Papp Wallace, Krisztina M.; Bethel, Christopher R.; Caselli, Emilia; Romagnoli, Chiara; Winkler, Marisa L.; Spellberg, Brad; Prati, Fabio; Bonomo, Robert A. |
8 | Chemo-enzymatic synthesis of levodropropizine | 2003 | Caselli, Emilia; Tosi, Giovanni; Forni, Arrigo; Bucciarelli, Maria; Prati, Fabio |
9 | Click Chemistry in Lead Optimization of Boronic Acids as β-Lactamase Inhibitors | 2015 | Caselli, Emilia; Romagnoli, Chiara; Vahabi, Roza; Taracila, Magdalena A; Bonomo, Robert A; Prati, Fabio |
10 | A Common Mechanism Underlying Promiscuous Inhibitors from Virtual and High-Throughput Screening | 2002 | Susan L., Mcgovern; Caselli, Emilia; Nikolaus, Grigorieff; Brian K., Shoichet |
11 | A comprehensive and contemporary “snapshot” of β-lactamases in carbapenem resistant Acinetobacter baumannii | 2021 | Hujer, A. M.; Hujer, K. M.; Leonard, D. A.; Powers, R. A.; Wallar, B. J.; Mack, A. R.; Taracila, M. A.; Rather, P. N.; Higgins, P. G.; Prati, F.; Caselli, E.; Marshall, S. H.; Clarke, T.; Greco, C.; Venepally, P.; Brinkac, L.; Kreiswirth, B. N.; Fouts, D. E.; Bonomo, R. A. |
12 | Crystal structures of KPC-2 and SHV-1 β-lactamases in complex with the boronic acid transition state analog S02030 | 2016 | Nguyen, Nhu Q.; Krishnan, Nikhil P.; Rojas, Laura J.; Prati, Fabio; Caselli, Emilia; Romagnoli, Chiara; Bonomo, Robert A.; Van Den Akker, Focco |
13 | Deciphering the evolution of cephalosporin resistance to ceftolozane-tazobactam in pseudomonas aeruginosa | 2018 | Barnes, Melissa D.; Taracila, Magdalena A.; Rutter, Joseph D.; Bethel, Christopher R.; Galdadas, Ioannis; Hujer, Andrea M.; Caselli, Emilia; Prati, Fabio; Dekker, John P.; Papp-Wallace, Krisztina M.; Haider, Shozeb; Bonomo, Robert A. |
14 | Design and exploration of novel boronic acid Inhibitors reveals important Interactions with a clavulanic acid-resistant sulfhydryl- variable (SHV) β‑ lactamase | 2013 | Marisa L., Winkler; Elizabeth A., Rodkey; Magdalena A., Taracila; Sarah M., Drawz; Christopher R., Bethel; Krisztina M., Papp Wallace; Kerri M., Smith; Yan, Xu; Jeffrey R., Dwulit Smith; Romagnoli, Chiara; Caselli, Emilia; Prati, Fabio; Focco van den, Akker; Robert A., Bonomo |
15 | Design, synthesis, crystal structures and antimicrobial activity of sulfonamide boronic acids as beta-lactamase inhibitors | 2010 | Oliv, Eidam; Romagnoli, Chiara; Caselli, Emilia; Joel, Karpiak; Kerim, Babaoglu; Denise Teotico, Pohlhaus; Richard, Bonnet; Brian K., Shoichet; Prati, Fabio |
16 | Enantiomeric excess of 1,2-diols by formation of cyclic boronates: an improved method | 2005 | Morandi, Stefania; Caselli, Emilia; Forni, Arrigo; Bucciarelli, Maria; Torre, Giovanni; Prati, Fabio |
17 | Energetic, structural, and antimicrobial analyses of beta-lactam side chain recognition by beta-lactamases | 2001 | Caselli, Emilia; Powers, Ra; Blasczcak, Lc; Wu, Cye; Prati, Fabio; Shoichet, Bk |
18 | Exploring novel inhibitors of FOX-4 Class C β-lactamase | 2010 | S., Mallo; C., Bethel; F., Perez llarena; Prati, Fabio; Caselli, Emilia; M., Page; G., Bou; R., Bonomo |
19 | Exploring sequence requirements for C3/C4 carboxylate recognition in the Pseudomonas aeruginosa cephalosporinase: Insights into plasticity of the AmpC β-lactamase | 2011 | Sarah M., Drawz; Magdalena, Taracila; Caselli, Emilia; Prati, Fabio; Robert A., Bonomo |
20 | Fragment-guided Design of Subnanomolar β-Lactamase Inhibitors Active in vivo | 2012 | O., Eidam; Romagnoli, Chiara; G., Dalmasso; S., Barelier; Caselli, Emilia; R., Bonnet; B. K., Shoichet; Prati, Fabio |