PINZI, LUCA

PINZI, LUCA  

Dipartimento di Scienze della Vita  

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Titolo Data di pubblicazione Autore(i) File
2-Phenyloxazole-4-carboxamide as a Scaffold for Selective Inhibition of Human Monoamine Oxidase B 1-gen-2019 Di Paolo, M. L.; Christodoulou, M. S.; Calogero, A. M.; Pinzi, L.; Rastelli, G.; Passarella, D.; Cappelletti, G.; Dalla Via, L.
An unexpected reversal in the pharmacological stereoselectivity of benzothiadiazine AMPA positive allosteric modulators 1-gen-2016 Battisti, UMBERTO MARIA; Citti, Cinzia; Rastelli, Giulio; Pinzi, Luca; Puja, Giulia; Ravazzini, Federica; Ciccarella, Giuseppe; Braghiroli, Daniela; Cannazza, Giuseppe
Antifungal Activity and DNA Topoisomerase Inhibition of Hydrolysable Tannins from Punica granatum L 1-gen-2021 Brighenti, V.; Iseppi, R.; Pinzi, L.; Mincuzzi, A.; Ippolito, A.; Messi, P.; Sanzani, S. M.; Rastelli, G.; Pellati, F.
Chemoinformatics Analyses of Tau Ligands Reveal Key Molecular Requirements for the Identification of Potential Drug Candidates against Tauopathies 1-gen-2021 Pinzi, Luca; Tinivella, Annachiara; Rastelli, Giulio
Computational polypharmacology comes of age 1-gen-2015 Rastelli, Giulio; Pinzi, Luca
Design and Synthesis of Hsp90 Inhibitors with B-Raf and PDHK1 Multi-Target Activity 1-gen-2021 Pinzi, L.; Foschi, F.; Christodoulou, M. S.; Passarella, D.; Rastelli, G.
Design of dual inhibitors of histone deacetylase 6 and heat shock protein 90 1-gen-2020 Pinzi, L.; Benedetti, R.; Altucci, L.; Rastelli, G.
Development and application of LigAdvisor, a user-friendly web-platform for polypharmacology and drug repurposing 1-gen-2021 Pinzi, Luca; Tinivella, Annachiara; Rastelli, Giulio
Drug Repurposing and Polypharmacology to Fight SARS-CoV-2 Through Inhibition of the Main Protease 1-gen-2021 Pinzi, Luca; Tinivella, Annachiara; Caporuscio, Fabiana; Rastelli, Giulio
Dual Targeting Strategies On Histone Deacetylase 6 (HDAC6) And Heat Shock Protein 90 (Hsp90) 1-gen-2021 Bonanni, Davide; Citarella, Andrea; Moi, Davide; Pinzi, Luca; Bergamini, Elisa; Rastelli, Giulio
Evaluation of Amides, Carbamates, Sulfonamides, and Ureas of 4-Prop-2-ynylidenecycloalkylamine as Potent, Selective, and Bioavailable Negative Allosteric Modulators of Metabotropic Glutamate Receptor 5 1-gen-2019 Graziani, Davide; Caligari, Silvia; Callegari, Elisa; De Toma, Carlo; Longhi, Matteo; Frigerio, Fabio; Dilernia, Roberto; Menegon, Sergio; Pinzi, Luca; Pirona, Lorenza; Tazzari, Valerio; Valsecchi, Anna Elisa; Vistoli, Giulio; Rastelli, Giulio; Ruga Riva, Carlo
Heat shock protein 90 and serine/threonine kinase B-Raf inhibitors have overlapping chemical space 1-gen-2017 Anighoro, A.; Pinzi, Luca; Marverti, Gaetano; Bajorath, J; Rastelli, Giulio
Hydroxamic Acid Derivatives: From Synthetic Strategies to Medicinal Chemistry Applications 1-gen-2021 Citarella, A.; Moi, D.; Pinzi, L.; Bonanni, D.; Rastelli, G.
Identification of 4-aryl-1H-pyrrole[2,3-b]pyridine derivatives for the development of new B-Raf inhibitors 1-gen-2018 Pinzi, Luca; Anighoro, Andrew; Bajorath, Jürgen; Rastelli, Giulio
Identification of potential biological targets of oxindole scaffolds via in silico repositioning strategies 1-gen-2022 Tinivella, Annachiara; Pinzi, Luca; Gambacorta, Guido; Baxendale, Ian; Rastelli, Giulio
Identification of small-molecule EGFR allosteric inhibitors by high-Throughput docking 1-gen-2018 Caporuscio, Fabiana; Tinivella, Annachiara; Restelli, Valentina; Semrau, Marta S; Pinzi, Luca; Storici, Paola; Broggini, Massimo; Rastelli, Giulio
Identification of Target Associations for Polypharmacology from Analysis of Crystallographic Ligands of the Protein Data Bank 1-gen-2020 Pinzi, L.; Rastelli, G.
In silico repositioning of cannabigerol as a novel inhibitor of the enoyl acyl carrier protein (ACP) reductase (INHA) 1-gen-2019 Pinzi, L.; Lherbet, C.; Baltas, M.; Pellati, F.; Rastelli, G.
Inhibitors of histone deacetylase 6 based on a novel 3-hydroxy-isoxazole zinc binding group 1-gen-2021 Linciano, P.; Pinzi, L.; Belluti, S.; Chianese, U.; Benedetti, R.; Moi, D.; Altucci, L.; Franchini, S.; Imbriano, C.; Sorbi, C.; Rastelli, G.
Investigation of the effect of different linker chemotypes on the inhibition of histone deacetylases (HDACs) 1-gen-2021 Linciano, P.; Benedetti, R.; Pinzi, L.; Russo, F.; Chianese, U.; Sorbi, C.; Altucci, L.; Rastelli, G.; Brasili, L.; Franchini, S.