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EVALUATION OF LR STABILITY BY LC CHIP Q-TOF AND QUANTITATIVE DETERMINATION OF LR PEPTIDE CELL PENETRATION BY LC-MS/MS 1-gen-2014 Cazzato, ADDOLORATA STEFANIA; Cannazza, Giuseppe; Ponterini, Glauco; Marraccini, Chiara; Pirondi, Silvia; Genovese, Filippo; Costi, Maria Paola
Development of an in vitro liquid chromatography-mass spectrometry method to evaluate stereo and chemical stability of new drug candidates employing immobilized artificial membrane column 1-gen-2014 Cannazza, Giuseppe; Battisti, Umberto M.; Carrozzo, Marina M.; Cazzato, Addolorata S.; Braghiroli, Daniela; Parenti, Carlo; Troisi, Luigino
Development of lipid nanocarriers as delivery systems for a small peptide with anti-ovarian activity 1-gen-2014 Sacchetti, Francesca; Cazzato, ADDOLORATA STEFANIA; Marraccini, Chiara; Cannazza, Giuseppe; Iannuccelli, Valentina; Maretti, Eleonora; Costi, Maria Paola; Leo, Eliana Grazia
Design, stereoselective synthesis, configurational stability and biological activity of 7-chloro-9-(furan-3-yl)-2,3,3a,4-tetrahydro-1H-benzo[e]pyrrolo[2,1-c][1,2,4]thiadiazine 5,5-dioxide 1-gen-2014 Carrozzo, Marina Maria; Battisti, UMBERTO MARIA; Cannazza, Giuseppe; Puja, Giulia; Ravazzini, Federica; Falchicchio, Aurelia; Perrone, Serena; Citti, Cinzia; Jozwiak, Krzysztof; Braghiroli, Daniela; Parenti, Carlo; Troisi, Luigino
Internalization and stability of a thymidylate synthase peptide inhibitor in ovarian cancer cells 1-gen-2014 Cannazza, Giuseppe; Cazzato, ADDOLORATA STEFANIA; Marraccini, Chiara; Pavesi, Giorgia; Pirondi, Silvia; R., Guerrini; M., Pelà; Frassineti, Chiara; Ferrari, Stefania; Marverti, Gaetano; Ponterini, Glauco; Costi, Maria Paola
Stereoselective synthesis of α-alkylidene β-oxo amides by palladium-catalyzed carbonylation 1-gen-2014 Perrone, Serena; Salomone, Antonio; Caroli, Antonio; Falcicchio, Aurelia; Citti, Cinzia; Cannazza, Giuseppe; Troisi, Luigino
One-pot synthesis of azobenzene derivatives by oxidation of 2,3-dihydrobenzothiadiazines 1-gen-2014 Cannazza, Giuseppe; Perrone, Serena; Rosato, Francesca; D'Accolti, Lucia; Parenti, Carlo; Troisi, Luigino
The cytisine derivatives, CC4 and CC26, reduce nicotine-induced conditioned place preference in zebrafish by acting on heteromeric neuronal nicotinic acetylcholine receptors 1-gen-2014 Ponzoni, Luisa; Braida, Daniela; Pucci, Luca; Andrea, Donzelli; Fasoli, Francesca; Manfredi, Irene; Papke, Roger L.; Stokes, Clare; Cannazza, Giuseppe; Clementi, Francesco; Gotti, Cecilia; Sala, Mariaelvina
Ring opening of heterocycles containing a C–N double bond: a simple synthesis of imides promoted by acyl palladium species 1-gen-2014 Perrone, Serena; Cannazza, Giuseppe; Caroli, Antonio; Salomone, Antonio; Troisi, Luigino
Different physiological and behavioural effects of e-cigarette vapour and cigarette smoke in mice 1-gen-2015 Ponzoni, L; Moretti, M; Sala, M; Fasoli, F; Mucchietto, V; Lucini, V; Cannazza, Giuseppe; Gallesi, G; Castellana, Carmela Nives; Clementi, F; Zoli, Michele; Gotti, C; Braida, D.
A direct synthesis of 3-acyl-4-hydroxy-2-pyranone derivatives via palladium-catalyzed carbonylation of α-chloroketones. A cascade reaction involving acylketenes 1-gen-2015 Perrone, Serena; Caroli, Antonio; Cannazza, Giuseppe; Granito, Catia; Salomone, Antonio; Troisi, Luigino
Nanoencapsulation of an hTS inhibitor octapeptide against ovarian cancer in solid lipid matrix 1-gen-2015 Sacchetti, Francesca; Marraccini, Chiara; Cannazza, Giuseppe; Iannuccelli, Valentina; Hanuskova, Miriam; Maretti, Eleonora; Costi, Maria Paola; Leo, Eliana Grazia
Calcium-Carbonate Nanocapsules Improve the Efficacy of BEZ235 in Lymphoma a Cell Line: A Promising New Technology of Drug Delivery 1-gen-2015 Civallero, Monica; Vergaro, Viviana; Citti, Cinzia; Cosenza, Maria; Cannazza, Giuseppe; Parenti, Carlo; Bari, Alessia; Ciccarella, Giuseppe; Sacchi, Stefano; Pozzi, Samantha
Interaction between human serum albumin and different anatase TiO2 nanoparticles: A nano-bio interface study 1-gen-2015 Vergaro, Viviana; Carlucci, Claudia; Cascione, Mariafrancesca; Lorusso, Caterina; Conciauro, Francesca; Scremin, Barbara Federica; Congedo, Paolo Maria; Cannazza, Giuseppe; Citti, Cinzia; Ciccarella, Giuseppe
7-Chloro-5-(furan-3-yl)-3-methyl-4H-benzo[e][1,2,4]thiadiazine 1,1-Dioxide as Positive Allosteric Modulator of α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor. The End of the Unsaturated-Inactive Paradigm? 1-gen-2016 Citti, Cinzia; Battisti, UMBERTO MARIA; Cannazza, Giuseppe; Jozwiak, Krzysztof; Stasiak, Natalia; Puja, Giulia; Ravazzini, Federica; Ciccarella, Giuseppe; Braghiroli, Daniela; Parenti, Carlo; Troisi, Luigino; Zoli, Michele
"Heart-cut" bidimensional achiral-chiral liquid chromatography applied to the evaluation of stereoselective metabolism, in vivo biological activity and brain response to chiral drug candidates targeting the central nervous system 1-gen-2016 Battisti, Umberto M.; Citti, Cinzia; Larini, Martina; Ciccarella, Giuseppe; Stasiak, Natalia; Troisi, Luigino; Braghiroli, Daniela; Parenti, Carlo; Zoli, Michele; Cannazza, Giuseppe
Analytical and preparative enantioseparation and main chiroptical properties of Iridium(III) bis(4,6-difluorophenylpyridinato)picolinato 1-gen-2016 Citti, Cinzia; Battisti, Umberto M.; Ciccarella, Giuseppe; Maiorano, Vincenzo; Gigli, Giuseppe; Abbate, Sergio; Mazzeo, Giuseppe; Castiglioni, Ettore; Longhi, Giovanna; Cannazza, Giuseppe
Synthesis of β-enamino acid and heteroaryl acetic acid derivatives by Pd-catalyzed carbonylation of α-chloroimines and 2-chloromethyl aza-heterocycles 1-gen-2016 Perrone, Serena; Capua, Martina; Cannazza, Giuseppe; Salomone, Antonio; Troisi, Luigino
Medicinal cannabis: Principal cannabinoids concentration and their stability evaluated by a high performance liquid chromatography coupled to diode array and quadrupole time of flight mass spectrometry method 1-gen-2016 Citti, Cinzia; Ciccarella, Giuseppe; Braghiroli, Daniela; Parenti, Carlo; Vandelli, Maria Angela; Cannazza, Giuseppe
An unexpected reversal in the pharmacological stereoselectivity of benzothiadiazine AMPA positive allosteric modulators 1-gen-2016 Battisti, UMBERTO MARIA; Citti, Cinzia; Rastelli, Giulio; Pinzi, Luca; Puja, Giulia; Ravazzini, Federica; Ciccarella, Giuseppe; Braghiroli, Daniela; Cannazza, Giuseppe
Mostrati risultati da 41 a 60 di 119
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