Sfoglia per Autore
Stereoselective synthesis of erythro beta-substituted aspartates
1997 Antolini, Luciano; Bucciarelli, Maria; Caselli, Emilia; Davoli, Paolo; Forni, Arrigo; Moretti, Irene; Prati, Fabio; Torre, Giovanni
Structure-Based Design and In Parallel Synthesis of Boronic Acid Inhibitors of AmpC 61538;-Lactamase
2000 Tondi, Donatella; Powers, R.; Caselli, Emilia; Costi, Maria Paola; Shoichet, B. K.
Structure-based design and solid phase synthesis of novel AmpC b-lactamase inhibitors
2001 Tondi, Donatella; Powers, R.; Caselli, E.; Costi, M. P.; Shoichet, B. K.
Progettazione, Sintesi ed Attività di Acidi 1-Acilamminoalcanboronici Inibitori di beta-Lattamasi
2001 Caselli, Emilia; Forni, Arrigo; SHOICHET B., K; Prati, Fabio
Energetic, structural, and antimicrobial analyses of beta-lactam side chain recognition by beta-lactamases
2001 Caselli, Emilia; Powers, Ra; Blasczcak, Lc; Wu, Cye; Prati, Fabio; Shoichet, Bk
Structure-based design and in-parallel synthesis of inhibitors of AmpC β-lactamase
2001 Tondi, Donatella; Ra, Powers; Caselli, Emilia; Mc, Negri; J., Blazquez; Costi, Maria Paola; Bk, Shoichet
The structures of Ceftazidime and Its Transition State Analog in Complex with AmpC-beta-lactamase: Implication for Resistance Mutation and Inhibitor Design
2001 R. A., Powers; Caselli, Emilia; P. J., Focia; Prati, Fabio; B. K., Shoichet
Highly enantioselective reduction of ethyl 4-chloro-3-oxobutanoate to L-and D-3-hydroxyesters with baker`s yeast
2002 Forni, Arrigo; Caselli, Emilia; Prati, Fabio; Bucciarelli, Maria; Torre, Giovanni
Lipase-Catalyzed Resolution and Desymmetrization of 2-Hydroxymethylaziridines
2002 Davoli, Paolo; Caselli, Emilia; Bucciarelli, Maria; Forni, Arrigo; Torre, Giovanni; Prati, Fabio
A Common Mechanism Underlying Promiscuous Inhibitors from Virtual and High-Throughput Screening
2002 Susan L., Mcgovern; Caselli, Emilia; Nikolaus, Grigorieff; Brian K., Shoichet
Acido alfa-Acetammido-alfa-Fenilmetanboronico come Agente Derivatizzante Chirale per la Determinazione dell’Eccesso Enantiomerico di 1,2-Dioli
2003 B., Bonfiglio; Caselli, Emilia; Forni, Arrigo; Danieli, Chiara; Prati, Fabio
Sintesi Stereoselettiva di Acidi Boronici Inibitori di beta-Lattamasi
2003 Morandi, Stefania; Caselli, Emilia; S., Baldini; Prati, Fabio
Recognition and resistance in TEM beta-lactamase
2003 Xj, Wang; G., Minasov; J., Blazquez; Caselli, Emilia; Prati, Fabio; Bk, Shoichet
Nanomolar inhibitors of AmpC beta-lactamase
2003 Morandi, Federica; Caselli, Emilia; Morandi, Stefania; P. J., Focia; J., Blazquez; B. K., Shoichet; Prati, Fabio
(S)-(+)-N-acetylphenylglycineboronic acid: A chiral derivatizing agent for Ee determination of 1,2-diols
2003 Caselli, Emilia; Danieli, Chiara; Morandi, Stefania; B., Bonfiglio; Forni, Arrigo; Prati, Fabio
Chemo-enzymatic synthesis of levodropropizine
2003 Caselli, Emilia; Tosi, Giovanni; Forni, Arrigo; Bucciarelli, Maria; Prati, Fabio
Biocatalytic asymmetric synthesis of (S)- and (R)-Timolol
2004 Tosi, Giovanni; F., Zironi; Caselli, Emilia; Forni, Arrigo; Prati, Fabio
Enantiomeric excess of 1,2-diols by formation of cyclic boronates: an improved method
2005 Morandi, Stefania; Caselli, Emilia; Forni, Arrigo; Bucciarelli, Maria; Torre, Giovanni; Prati, Fabio
Using Boronic Acid Transition State Inhibitors to understand the extended spectrum (ES) and carbapenemase phenotypes of class A beta-lactamases in Klebsiella pneumoniae
2007 BETHEL C., R; Prati, Fabio; Caselli, Emilia; Bonomo, R. A.
Structure-based optimization of cephalotin analogue boronic acids as beta-lactamase inhibitors
2008 Morandi, Stefania; Morandi, Federica; Caselli, Emilia; B. K., Shoichet; Prati, Fabio
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Stereoselective synthesis of erythro beta-substituted aspartates | 1-gen-1997 | Antolini, Luciano; Bucciarelli, Maria; Caselli, Emilia; Davoli, Paolo; Forni, Arrigo; Moretti, Irene; Prati, Fabio; Torre, Giovanni | |
Structure-Based Design and In Parallel Synthesis of Boronic Acid Inhibitors of AmpC 61538;-Lactamase | 1-gen-2000 | Tondi, Donatella; Powers, R.; Caselli, Emilia; Costi, Maria Paola; Shoichet, B. K. | |
Structure-based design and solid phase synthesis of novel AmpC b-lactamase inhibitors | 1-gen-2001 | Tondi, Donatella; Powers, R.; Caselli, E.; Costi, M. P.; Shoichet, B. K. | |
Progettazione, Sintesi ed Attività di Acidi 1-Acilamminoalcanboronici Inibitori di beta-Lattamasi | 1-gen-2001 | Caselli, Emilia; Forni, Arrigo; SHOICHET B., K; Prati, Fabio | |
Energetic, structural, and antimicrobial analyses of beta-lactam side chain recognition by beta-lactamases | 1-gen-2001 | Caselli, Emilia; Powers, Ra; Blasczcak, Lc; Wu, Cye; Prati, Fabio; Shoichet, Bk | |
Structure-based design and in-parallel synthesis of inhibitors of AmpC β-lactamase | 1-gen-2001 | Tondi, Donatella; Ra, Powers; Caselli, Emilia; Mc, Negri; J., Blazquez; Costi, Maria Paola; Bk, Shoichet | |
The structures of Ceftazidime and Its Transition State Analog in Complex with AmpC-beta-lactamase: Implication for Resistance Mutation and Inhibitor Design | 1-gen-2001 | R. A., Powers; Caselli, Emilia; P. J., Focia; Prati, Fabio; B. K., Shoichet | |
Highly enantioselective reduction of ethyl 4-chloro-3-oxobutanoate to L-and D-3-hydroxyesters with baker`s yeast | 1-gen-2002 | Forni, Arrigo; Caselli, Emilia; Prati, Fabio; Bucciarelli, Maria; Torre, Giovanni | |
Lipase-Catalyzed Resolution and Desymmetrization of 2-Hydroxymethylaziridines | 1-gen-2002 | Davoli, Paolo; Caselli, Emilia; Bucciarelli, Maria; Forni, Arrigo; Torre, Giovanni; Prati, Fabio | |
A Common Mechanism Underlying Promiscuous Inhibitors from Virtual and High-Throughput Screening | 1-gen-2002 | Susan L., Mcgovern; Caselli, Emilia; Nikolaus, Grigorieff; Brian K., Shoichet | |
Acido alfa-Acetammido-alfa-Fenilmetanboronico come Agente Derivatizzante Chirale per la Determinazione dell’Eccesso Enantiomerico di 1,2-Dioli | 1-gen-2003 | B., Bonfiglio; Caselli, Emilia; Forni, Arrigo; Danieli, Chiara; Prati, Fabio | |
Sintesi Stereoselettiva di Acidi Boronici Inibitori di beta-Lattamasi | 1-gen-2003 | Morandi, Stefania; Caselli, Emilia; S., Baldini; Prati, Fabio | |
Recognition and resistance in TEM beta-lactamase | 1-gen-2003 | Xj, Wang; G., Minasov; J., Blazquez; Caselli, Emilia; Prati, Fabio; Bk, Shoichet | |
Nanomolar inhibitors of AmpC beta-lactamase | 1-gen-2003 | Morandi, Federica; Caselli, Emilia; Morandi, Stefania; P. J., Focia; J., Blazquez; B. K., Shoichet; Prati, Fabio | |
(S)-(+)-N-acetylphenylglycineboronic acid: A chiral derivatizing agent for Ee determination of 1,2-diols | 1-gen-2003 | Caselli, Emilia; Danieli, Chiara; Morandi, Stefania; B., Bonfiglio; Forni, Arrigo; Prati, Fabio | |
Chemo-enzymatic synthesis of levodropropizine | 1-gen-2003 | Caselli, Emilia; Tosi, Giovanni; Forni, Arrigo; Bucciarelli, Maria; Prati, Fabio | |
Biocatalytic asymmetric synthesis of (S)- and (R)-Timolol | 1-gen-2004 | Tosi, Giovanni; F., Zironi; Caselli, Emilia; Forni, Arrigo; Prati, Fabio | |
Enantiomeric excess of 1,2-diols by formation of cyclic boronates: an improved method | 1-gen-2005 | Morandi, Stefania; Caselli, Emilia; Forni, Arrigo; Bucciarelli, Maria; Torre, Giovanni; Prati, Fabio | |
Using Boronic Acid Transition State Inhibitors to understand the extended spectrum (ES) and carbapenemase phenotypes of class A beta-lactamases in Klebsiella pneumoniae | 1-gen-2007 | BETHEL C., R; Prati, Fabio; Caselli, Emilia; Bonomo, R. A. | |
Structure-based optimization of cephalotin analogue boronic acids as beta-lactamase inhibitors | 1-gen-2008 | Morandi, Stefania; Morandi, Federica; Caselli, Emilia; B. K., Shoichet; Prati, Fabio |
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