SAXENA, PUNEET
Dettaglio
SAXENA, PUNEET
Dipartimento di Scienze della Vita
Pubblicazioni
Risultati 1 - 14 di 14 (tempo di esecuzione: 0.0 secondi).
Titolo | Data di pubblicazione | Autore(i) | |
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1 | 2-Carboxyquinoxalines Kill Mycobacterium tuberculosis through Noncovalent Inhibition of DprE1 | 2015 | Neres, João; Hartkoorn, Ruben C.; Chiarelli, Laurent R.; Gadupudi, Ramakrishna; Pasca, Maria Rosalia; Mori, Giorgia; Venturelli, Alberto; Savina, Svetlana; Makarov, Vadim; Kolly, Gaelle S.; Molteni, Elisabetta; Binda, Claudia; Dhar, Neeraj; Ferrari, Stefania; Brodin, Priscille; Delorme, Vincent; Landry, Valérie; de Jesus Lopes Ribeiro, Ana Luisa; Farina, Davide Salvatore Francesco; Saxena, Puneet; Pojer, Florence; Carta, Antonio; Luciani, Rosaria; Porta, Alessio; Zanoni, Giuseppe; De Rossi, Edda; Costi, Maria Paola; Riccardi, Giovanna; Cole, Stewart T. |
2 | Alanine Mutants of the Interface Residues of Human Thymidylate Synthase Decode Key Features of the Binding Mode of Allosteric Anticancer Peptides | 2015 | Tochowicz, Anna Maria; Santucci, Matteo; Saxena, Puneet; Guaitoli, Giambattista; Costi, Maria Paola |
3 | Computational Insights into ADAMTS4, ADAMTS5 andMMP13 Inhibitor Selectivity | 2012 | FILOMIA, Federico; SAXENA, PUNEET; DURANTE, Caterina; DE RIENZO, Francesca; COCCHI, Marina; MENZIANI, Maria Cristina |
4 | Conformational Propensity and Biological Studies of Proline Mutated LR Peptides Inhibiting Human Thymidylate Synthase and Ovarian Cancer Cell Growth | 2018 | Saxena, Puneet; Severi, Leda; Santucci, Matteo; Taddia, Laura; Ferrari, Stefania; Luciani, Rosaria; Marverti, Gaetano; Marraccini, Chiara; Tondi, Donatella; Mor, Marco; Laura, Scalvini; Vitiello, Simone; Losi, Lorena; Fonda, Sergio; Pacifico, Salvatore; Guerrini, Remo; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola |
5 | Cyclic Peptides Acting as Allosteric Inhibitors of Human Thymidylate Synthase and Cancer Cell Growth | 2019 | Pacifico, Salvatore; Santucci, Matteo; Luciani, Rosaria; Saxena, Puneet; Linciano, Pasquale; Ponterini, Glauco; Lauriola, Angela; D'Arca, Domenico; Marverti, Gaetano; Guerrini, Remo; Costi, Maria Paola |
6 | Exploiting the 2-Amino-1,3,4-thiadiazole Scaffold To InhibitTrypanosoma bruceiPteridine Reductase in Support of Early-Stage Drug Discovery | 2017 | Linciano, Pasquale; Dawson, Alice; Pöhner, Ina; Costa, David M; Sá, Monica S; Cordeiro-da-Silva, Anabela; Luciani, Rosaria; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Gribbon, Philip; Reinshagen, Jeanette; Wolf, Markus; Behrens, Birte; Hannaert, Véronique; Michels, Paul A M; Nerini, Erika; Pozzi, Cecilia; di Pisa, Flavio; Landi, Giacomo; Santarem, Nuno; Ferrari, Stefania; Saxena, Puneet; Lazzari, Sandra; Cannazza, Giuseppe; Freitas-Junior, Lucio H; Moraes, Carolina B; Pascoalino, Bruno S; Alcântara, Laura M; Bertolacini, Claudia P; Fontana, Vanessa; Wittig, Ulrike; Müller, Wolfgang; Wade, Rebecca C; Hunter, William N; Mangani, Stefano; Costantino, Luca; Costi, Maria P |
7 | Hotspots in an obligate homodimeric anticancer target. structural and functional effects of interfacial mutations in human thymidylate synthase | 2015 | Salo Ahen, Outi M. H.; Tochowicz, Anna; Pozzi, Cecilia; Cardinale, Daniela; Ferrari, Stefania; Boum, Yap; Mangani, Stefano; Stroud, Robert M.; Saxena, Puneet; Myllykallio, Hannu; Costi, Maria Paola; Ponterini, Glauco; Wade, Rebecca C. |
8 | Maxwell A: F1000Prime Recommendation of Evaluation [Neres J et al., ACS Chem Biol 2014]. In F1000Prime, 09 Jan 2015; DOI: 10.3410/f.725248139.793502885. F1000Prime.com/725248139#eval793502885 | 2015 | Maxwell, Anthony; Neres, J; Hartkoorn, Rc; Chiarelli, Lr; Gadupudi, Ramakrishna; Pasca, Mr; Mori, G; Venturelli, Alberto; Savina, S; Makarov, V; Kolly, Gs; Molteni, E; Binda, C; Dhar, N; Ferrari, Stefania; Brodin, P; Delorme, V; Landry, V; de Jesus Lopes Ribeiro, Al; Farina, Davide Salvatore Francesco; Saxena, Puneet; Pojer, F; Carta, Antonello; Luciani, Rosaria; Porta, Andrea; Zanoni, G; De Rossi, E; Costi, Maria Paola; Riccardi, G. |
9 | Optimization of Peptides That Target Human Thymidylate Synthase to Inhibit Ovarian Cancer Cell Growth | 2014 | M., Pelà; Saxena, Puneet; Luciani, Rosaria; Santucci, Matteo; Ferrari, Stefania; Marverti, Gaetano; Marraccini, Chiara; Martello, Andrea; Pirondi, Silvia; Genovese, Filippo; S., Salvadori; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola; R., Guerrini |
10 | Progress Towards the Identification of New Aggrecanase Inhibitors | 2009 | DE RIENZO, Francesca; Saxena, Puneet; Filomia, Federico; G., Caselli; F., Colace; L., Stasi; A., Giordani; Menziani, Maria Cristina |
11 | QUINOXALINE DERIVATIVES AS ANTITUBERCULOSIS AGENTS | - | Costi, Maria Paola; Ferrari, Stefania; Saxena, Puneet; Venturelli, Alberto; Farina, Davide Salvatore Francesco; Luciani, Rosaria; Gadupudi, Ramakrishna |
12 | Structure-Based Selectivity Optimization of Piperidine–Pteridine Derivatives as Potent Leishmania Pteridine Reductase Inhibitors | 2012 | Paola, Corona; Gibellini, Federica; Saxena, Puneet; Luciani, Rosaria; Guerrieri, Davide; Nerini, Erika; Ferrari, Stefania; Costi, Maria Paola |
13 | Targeting the trypanosomatidic enzymes pteridine reductase and dihydrofolate reductase. | 2012 | Ferrari, Stefania; Valeria, Losasso; Saxena, Puneet; Costi, Maria Paola |
14 | Virtual Screening and X-ray Crystallography Identify Non-Substrate Analog Inhibitors of Flavin-Dependent Thymidylate Synthase | 2016 | Luciani, Rosaria; Saxena, Puneet; Surade, Sachin; Santucci, Matteo; Venturelli, Alberto; Borsari, Chiara; Marverti, Gaetano; Ponterini, Glauco; Ferrari, Stefania; Blundell, Tom L; Costi, Maria Paola |