TAIT, Annalisa
Dettaglio
TAIT, Annalisa
Dipartimento di Scienze della Vita
Pubblicazioni
Risultati 1 - 20 di 43 (tempo di esecuzione: 0.0 secondi).
Titolo | Data di pubblicazione | Autore(i) | |
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1 | 1,2,4-Benzothiadiazine derivatives as alpha(1) and 5-HT1A receptor ligands | 2005 | Tait, Annalisa; Luppi, Amedeo; Franchini, Silvia; E., Preziosi; Parenti, Carlo; M., Buccioni; G., Marucci; A., Leonardi; E., Poggesi; Brasili, Livio |
2 | 1,3-Dioxane as a scaffold for potent and selective 5-HT1AR agonist with in-vivo anxiolytic, anti-depressant and anti-nociceptive activity | 2019 | Franchini, S.; Sorbi, C.; Linciano, P.; Carnevale, G.; Tait, A.; Ronsisvalle, S.; Buccioni, M.; Del Bello, F.; Cilia, A.; Pirona, L.; Denora, N.; Iacobazzi, R. M.; Brasili, L. |
3 | 1,3-Dioxolane-Based Ligands as Rigid Analogues ofNaftopidil: Structure–Affinity/Activity Relationships at a1and 5-HT1A Receptors | 2009 | Sorbi, Claudia; Franchini, Silvia; Tait, Annalisa; Prandi, Adolfo; Gallesi, Rossella; P., Angeli; G., Marucci; L., Pirona; E., Poggesi; Brasili, Livio |
4 | 1,3-Dioxolane-Based Ligands Incorporating a Lactam or Imide moiety: Structure-Affinity/Activity Relationship at alpha1–Adrenoceptor subtypes and at 5-HT1A Receptors | 2010 | Franchini, Silvia; Prandi, Adolfo; Baraldi, Anna Maria; Sorbi, Claudia; Tait, Annalisa; M., Buccioni; G., Marucci; A., Cilia; L., Pirona; P., Fossa; E., Cichero; Brasili, Livio |
5 | 1,4-Dioxolane-triazaspirodecanone derivatives as nociceptin/orphanin FQ receptor ligands | 2014 | Corrado, Sandra; Sorbi, Claudia; Tait, Annalisa; Battisti, Umberto M.; Camarda, Valeria; Malfacini, Davide; Calò, Girolamo; Brasili, Livio |
6 | 2,1,3-Benzothiadiazine derivatives: synthesis and screening versus PDE4 enzyme | 2005 | Tait, Annalisa; Luppi, Amedeo; Avallone, Rossella; Baraldi, Mario |
7 | (2,2-Diphenyl-[1,3]oxathiolan-5-ylmethyl)-(3-phenylpropyl)-amine: a Potent and Selective 5-HT1A Receptor Agonist | 2009 | Franchini, Silvia; Tait, Annalisa; Prandi, Adolfo; Sorbi, Claudia; Gallesi, Rossella; M., Buccioni; G., Marucci; C., De Stefani; A., Cilia; Brasili, Livio |
8 | Benzothiadiazine derivatives as 1 and 5-HT1A receptor ligands. | 2005 | Tait, Annalisa; Franchini, Silvia; M., Buccioni; G., Marucci; A., Leonardi; E., Poggesi; Brasili, Livio |
9 | Designing Chimeric Molecules for Drug Discovery by Leveraging Chemical Biology | 2020 | Borsari, C.; Trader, D. J.; Tait, A.; Costi, M. P. |
10 | Development of flavonoids derivatives as leads against Leishmaniasis and Trypanosomiasis-invited lecture | 2014 | Borsari, Chiara; Luciani, Rosaria; Pozzi, Cecilia; Tait, Annalisa; Costantino, Luca; Pellati, Federica; Ferrari, Stefania; Costi, Maria Paola |
11 | Diastereoselective Synthesis of (1,3-Dioxan-4-yl)pyrimidine and Purin Nucleoside Analogues | 2015 | Battisti, Umberto M.; Sorbi, Claudia; Quotadamo, Antonio; Franchini, Silvia; Tait, Annalisa; Schols, Dominique; Jeong, Lak Shin; Lee, Sang Kook; Song, Jayoung; Brasili, Livio |
12 | Discovery of a benzothiophene-flavonol halting miltefosine and antimonial drug resistance in Leishmania parasites through the application of medicinal chemistry, screening and genomics | 2019 | Borsari, Chiara; Dolores Jimenez-Anton, María; Eick, Julia; Bifeld, Eugenia; Jose Torrado, Juan; Isabel Olías-Molero, Ana; Jesús Corral, María; Santarem, Nuno; Baptista, Catarina; Severi, Leda; Gul, Sheraz; Wolf, Markus; Kuzikov, Maria; Ellinger, Bernhard; Reinshagen, Jeanette; Witt, Gesa; Linciano, Pasquale; Tait, Annalisa; Costantino, Luca; Luciani, Rosaria; Tejera Nevado, Paloma; Zander-Dinse, Dorothea; Franco, Caio H.; Ferrari, Stefania; Moraes, Carolina B.; Cordeiro-da-Silva, Anabela; Ponterini, Glauco; Clos, Joachim; María Alunda, Jose; Costi, Maria Paola |
13 | Discovery of a new series of 5-HT1A receptor agonists | 2010 | Franchini, Silvia; Prandi, Adolfo; Sorbi, Claudia; Tait, Annalisa; Annamaria, Baraldi; Piero, Angeli; Michela, Buccioni; Antonio, Cilia; Elena, Poggesi; Paola, Fossa; Brasili, Livio |
14 | Discovery Of New Sigma-2 Receptor Agonist Endowed With Antiproliferative Activity | 2016 | Franchini, Silvia; Sorbi, Claudia; Tait, Annalisa; Benassi, Luisa; Azzoni, Paola; Vaschieri, Crisitina; Pellacani, Giovanni; Prezzavento, Orazio; Ronsisvalle, Simine; Aricò, Giuseppina; Brasili, Livio |
15 | Effect of the rigidification of propranolol, a mixed β-adrenoceptor and 5-HT1AR antagonist | 2019 | Franchini, S.; Sorbi, C.; Linciano, P.; Brasili, L.; Tait, A. |
16 | Heteroarylalkanoic acids with possible antiinflammatoy activities, note IX The binding to human serum albumin | 1989 | Costantino, Luca; Parenti, Carlo; Tait, Annalisa; Di Bella, M. |
17 | Heteroarylphenoxyethyl amine as selective 5-HT1A receptor ligands: synthesis and structure-activity ralationship studies. | 2010 | Manasieva, LEDA IVANOVAA; Baraldi, Anna Maria; Franchini, Silvia; P., Fossa; E., Cichero; A., Cilia; E., Poggesi; Tait, Annalisa; Brasili, Livio |
18 | High-performance liquid chromatographic method for the quantification of anthranilic and 3-hydroxyanthranilic acid in rat brain dialysate | 2003 | Cannazza, Giuseppe; Baraldi, Mario; Braghiroli, Daniela; Tait, Annalisa; Parenti, Carlo |
19 | IDENTIFICATION OF POTENT 1,3-DIOXOLANE-BASED 5-HT1A RECEPTOR AGONISTS FOR THE TREATMENTS OF CNS DISORDERS AND PAIN | 2019 | Linciano, Pasquale; Sorbi, Claudia; Franchini, Silvia; Tait, Annalisa; Bardoni, Rita; Ronsisvalle, Simone; Denora, Nunzio; Lesniak, Anna; Bujalska-Zadrożny, Magdalena; Pawłowska, Agata; Chichero, Elena; Fossa, Paola; Brasili, Livio |
20 | Medicinal Chemistry in Parasitology: New Avenues in Drug Discovery | 2007 | Tait, Annalisa |