TAIT, Annalisa

TAIT, Annalisa  

Dipartimento di Scienze della Vita  

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Titolo Data di pubblicazione Autore(i) File
(2,2-Diphenyl-[1,3]oxathiolan-5-ylmethyl)-(3-phenylpropyl)-amine: a Potent and Selective 5-HT1A Receptor Agonist 1-gen-2009 Franchini, Silvia; Tait, Annalisa; Prandi, Adolfo; Sorbi, Claudia; Gallesi, Rossella; M., Buccioni; G., Marucci; C., De Stefani; A., Cilia; Brasili, Livio
1,2,4-Benzothiadiazine derivatives as alpha(1) and 5-HT1A receptor ligands 1-gen-2005 Tait, Annalisa; Luppi, Amedeo; Franchini, Silvia; E., Preziosi; Parenti, Carlo; M., Buccioni; G., Marucci; A., Leonardi; E., Poggesi; Brasili, Livio
1,3-Dioxane as a scaffold for potent and selective 5-HT1AR agonist with in-vivo anxiolytic, anti-depressant and anti-nociceptive activity 1-gen-2019 Franchini, S.; Sorbi, C.; Linciano, P.; Carnevale, G.; Tait, A.; Ronsisvalle, S.; Buccioni, M.; Del Bello, F.; Cilia, A.; Pirona, L.; Denora, N.; Iacobazzi, R. M.; Brasili, L.
1,3-Dioxolane-Based Ligands as Rigid Analogues ofNaftopidil: Structure–Affinity/Activity Relationships at a1and 5-HT1A Receptors 1-gen-2009 Sorbi, Claudia; Franchini, Silvia; Tait, Annalisa; Prandi, Adolfo; Gallesi, Rossella; P., Angeli; G., Marucci; L., Pirona; E., Poggesi; Brasili, Livio
1,3-Dioxolane-Based Ligands Incorporating a Lactam or Imide moiety: Structure-Affinity/Activity Relationship at alpha1–Adrenoceptor subtypes and at 5-HT1A Receptors 1-gen-2010 Franchini, Silvia; Prandi, Adolfo; Baraldi, Anna Maria; Sorbi, Claudia; Tait, Annalisa; M., Buccioni; G., Marucci; A., Cilia; L., Pirona; P., Fossa; E., Cichero; Brasili, Livio
1,4-Dioxolane-triazaspirodecanone derivatives as nociceptin/orphanin FQ receptor ligands 1-gen-2014 Corrado, Sandra; Sorbi, Claudia; Tait, Annalisa; Battisti, Umberto M.; Camarda, Valeria; Malfacini, Davide; Calò, Girolamo; Brasili, Livio
2,1,3-Benzothiadiazine derivatives: synthesis and screening versus PDE4 enzyme 1-gen-2005 Tait, Annalisa; Luppi, Amedeo; Avallone, Rossella; Baraldi, Mario
Benzothiadiazine derivatives as 1 and 5-HT1A receptor ligands. 1-gen-2005 Tait, Annalisa; Franchini, Silvia; M., Buccioni; G., Marucci; A., Leonardi; E., Poggesi; Brasili, Livio
Designing Chimeric Molecules for Drug Discovery by Leveraging Chemical Biology 1-gen-2020 Borsari, C.; Trader, D. J.; Tait, A.; Costi, M. P.
Development of flavonoids derivatives as leads against Leishmaniasis and Trypanosomiasis-invited lecture 1-gen-2014 Borsari, Chiara; Luciani, Rosaria; Pozzi, Cecilia; Tait, Annalisa; Costantino, Luca; Pellati, Federica; Ferrari, Stefania; Costi, Maria Paola
Diastereoselective Synthesis of (1,3-Dioxan-4-yl)pyrimidine and Purin Nucleoside Analogues 1-gen-2015 Battisti, Umberto M.; Sorbi, Claudia; Quotadamo, Antonio; Franchini, Silvia; Tait, Annalisa; Schols, Dominique; Jeong, Lak Shin; Lee, Sang Kook; Song, Jayoung; Brasili, Livio
Discovery of a benzothiophene-flavonol halting miltefosine and antimonial drug resistance in Leishmania parasites through the application of medicinal chemistry, screening and genomics 1-gen-2019 Borsari, Chiara; Dolores Jimenez-Anton, María; Eick, Julia; Bifeld, Eugenia; Jose Torrado, Juan; Isabel Olías-Molero, Ana; Jesús Corral, María; Santarem, Nuno; Baptista, Catarina; Severi, Leda; Gul, Sheraz; Wolf, Markus; Kuzikov, Maria; Ellinger, Bernhard; Reinshagen, Jeanette; Witt, Gesa; Linciano, Pasquale; Tait, Annalisa; Costantino, Luca; Luciani, Rosaria; Tejera Nevado, Paloma; Zander-Dinse, Dorothea; Franco, Caio H.; Ferrari, Stefania; Moraes, Carolina B.; Cordeiro-da-Silva, Anabela; Ponterini, Glauco; Clos, Joachim; María Alunda, Jose; Costi, Maria Paola
Discovery of a new series of 5-HT1A receptor agonists 1-gen-2010 Franchini, Silvia; Prandi, Adolfo; Sorbi, Claudia; Tait, Annalisa; Annamaria, Baraldi; Piero, Angeli; Michela, Buccioni; Antonio, Cilia; Elena, Poggesi; Paola, Fossa; Brasili, Livio
Discovery Of New Sigma-2 Receptor Agonist Endowed With Antiproliferative Activity 1-gen-2016 Franchini, Silvia; Sorbi, Claudia; Tait, Annalisa; Benassi, Luisa; Azzoni, Paola; Vaschieri, Crisitina; Pellacani, Giovanni; Prezzavento, Orazio; Ronsisvalle, Simine; Aricò, Giuseppina; Brasili, Livio
Effect of the rigidification of propranolol, a mixed β-adrenoceptor and 5-HT1AR antagonist 1-gen-2019 Franchini, S.; Sorbi, C.; Linciano, P.; Brasili, L.; Tait, A.
Heteroarylalkanoic acids with possible antiinflammatoy activities, note IX The binding to human serum albumin 1-gen-1989 Costantino, Luca; Parenti, Carlo; Tait, Annalisa; Di Bella, M.
Heteroarylphenoxyethyl amine as selective 5-HT1A receptor ligands: synthesis and structure-activity ralationship studies. 1-gen-2010 Manasieva, LEDA IVANOVAA; Baraldi, Anna Maria; Franchini, Silvia; P., Fossa; E., Cichero; A., Cilia; E., Poggesi; Tait, Annalisa; Brasili, Livio
High-performance liquid chromatographic method for the quantification of anthranilic and 3-hydroxyanthranilic acid in rat brain dialysate 1-gen-2003 Cannazza, Giuseppe; Baraldi, Mario; Braghiroli, Daniela; Tait, Annalisa; Parenti, Carlo
IDENTIFICATION OF POTENT 1,3-DIOXOLANE-BASED 5-HT1A RECEPTOR AGONISTS FOR THE TREATMENTS OF CNS DISORDERS AND PAIN 1-gen-2019 Linciano, Pasquale; Sorbi, Claudia; Franchini, Silvia; Tait, Annalisa; Bardoni, Rita; Ronsisvalle, Simone; Denora, Nunzio; Lesniak, Anna; Bujalska-Zadrożny, Magdalena; Pawłowska, Agata; Chichero, Elena; Fossa, Paola; Brasili, Livio
Medicinal Chemistry in Parasitology: New Avenues in Drug Discovery 1-gen-2008 Tait, Annalisa