Sfoglia per Autore
Synthesis, biological evaluation, and quantitative receptor docking simulations of 2-[(acylamino)ethyl]-1,4-benzodiazepines as novel tifluadom-like ligands with high affinity and selectivity for kappa-opioid receptors
1996 Cappelli, A; Anzini, M; Vomero, S; Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe; Sbacchi, M; Clarke, Gd; Mennuni, L.
Molecular structure and dynamics of some potent 5-HT3 receptor antagonists. Insight into the interaction with the receptor
1996 Cappelli, A; Donati, A; Anzini, M; Vomero, S; DE BENEDETTI, Pier Giuseppe; Menziani, Maria Cristina; Langer, T.
The Heuristic-Direct approach to Quantitative Structure-Activity Relationship Analysis of Ligand-G Protein Coupled Receptor Complexes
1996 Menziani, Maria Cristina; Fanelli, Francesca; Cocchi, Marina; DE BENEDETTI, Pier Giuseppe
Molecular dynamics of guest radicals in urea inclusion compounds
1997 Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe; Segre, Ulderico; Brustolon, M.
Mapping the peripheral benzodiazepine receptor binding site by conformationally restrained derivatives of 1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)-3-isoquinolinecarboxamide (PK11195)
1997 Cappelli, A; Anzini, M; Vomero, S; Debenedetti, Pg; Menziani, Maria Cristina; Giorgi, G; Manzoni, C.
Alpha 1-adrenoceptor subtype selectivity: Molecular modelling and theoretical quantitative structure-affinity relationships
1997 DE BENEDETTI, Pier Giuseppe; Fanelli, Francesca; Menziani, Maria Cristina; Cocchi, Marina; R., Testa; A., Leonardi
Theoretical investigation of IL-6 multiprotein receptor assembly
1997 Menziani, Maria Cristina; Fanelli, Francesca; DE BENEDETTI, Pier Giuseppe
Conformational analysis and theoretical quantitative size and shape-affinity relationships of N-4-protonated N-1-arylpiperazine 5-HT1A serotoninergic ligands
1997 Cocchi, Marina; Fanelli, Francesca; Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe
Computer modeling of size and shape descriptors of alpha 1-adrenergic receptor antagonists and quantitative structure-affinity/selectivity relationships
1998 Montorsi, Monia; Menziani, Maria Cristina; Cocchi, Marina; Fanelli, Francesca; DE BENEDETTI, Pier Giuseppe
Ab initio modeling and molecular dynamics simulation of the alpha 1b-adrenergic receptor activation
1998 Fanelli, Francesca; Menziani, Maria Cristina; A., Scheer; S., Cotecchia; DE BENEDETTI, Pier Giuseppe
Theoretical descriptors in quantitative structure - Affinity and selectivity relationship study of potent N4-substituted arylpiperazine 5-HT1(Alpha) receptor antagonists
1998 Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe; Karelson, M.
Novel potent and selective central 5-HT3 receptor ligands provided with different intrinsic efficacy. 1. Mapping the central 5-HT3 receptor binding site by arylpiperazine derivatives
1998 Cappelli, A; Anzini, M; Vomero, S; Mennuni, L; Makovec, F; Doucet, E; Hamon, M; Bruni, G; Romeo, Mr; Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe; Langer, T.
Theoretical study on the electrostatically driven step of receptor-G protein recognition
1999 Fanelli, Francesca; Menziani, Maria Cristina; A., Scheer; Cotecchia, S.; DE BENEDETTI, Pier Giuseppe
Relevance of theoretical molecular descriptors in quantitative structure-activity relationship analysis of alpha 1-adrenergic receptor antagonists
1999 Menziani, Maria Cristina; Montorsi, Monia; DE BENEDETTI, Pier Giuseppe; Karelson, M.
Novel potent and selective central 5-HT3 receptor ligands provided with different intrinsic efficacy. 2. Molecular basis of the intrinsic efficacy of arylpiperazine derivatives at the central 5-HT3 receptors
1999 Cappelli, A; Anzini, M; Vomero, S; Canullo, L; Mennuni, L; Makovec, F; Doucet, E; Hamon, M; Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe; Bruni, G; Romeo, Mr; Giorgi, G; Donati, A.
Synthesis, pharmacological evaluation, and structure-activity relationship and quantitative structure-activity relationship studies on novel derivatives of 2,4-diamino-6,7-dimethoxyquinazoline alpha(1)-adrenoceptor antagonists
1999 Leonardi, A; Motta, G; Boi, C; Testa, R; Poggesi, E; DE BENEDETTI, Pier Giuseppe; Menziani, Maria Cristina
Theoretical study on receptor-G protein recognition: new insights into the mechanism of the α1b-adrenergic receptor activation
1999 Fanelli, Francesca; Menziani, Maria Cristina; A., Scheer; S., Cotecchia; DE BENEDETTI, Pier Giuseppe
Theoretical investigation of substrate specificity for cytochromes p450 IA2, p450 IID6 and p450 IIIA4
2000 DE RIENZO, Francesca; Fanelli, Francesca; Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe
Molecular dynamics simulations of alumina addition in sodium silicate glasses
2000 Montorsi, Monia; Menziani, Maria Cristina; Leonelli, Cristina; Pellacani, Gian Carlo; A. N., Cormack
The ad hoc supermolecule approach to receptor ligand design
2000 DE BENEDETTI, Pier Giuseppe; Fanelli, Francesca; Menziani, Maria Cristina; Cocchi, Marina
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