MALPEZZI, GIULIA
MALPEZZI, GIULIA
Dipartimento di Scienze Biomediche, Metaboliche e Neuroscienze
A toolbox of biophysical and analytical assays helps to confirm the activity of novel hTS dimer disrupters (Ddis) with anticancer properties
2022 Tagliazucchi, Lorenzo; Venturelli, Alberto; Malpezzi, Giulia; Moschella, MARIA GAETANA; Aiello, Daniele; Lopresti, Ludovica; Pozzi, Cecilia; Marverti, Gaetano; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola
Applying optical tweezers technology to reveal Thymidylate Synthase interactions with its consensus mRNA
2023 Malpezzi, Giulia; Viader, Xvaier; Zaltron, Annamaria; Neri, Benedetta; di Felice, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Moschella, MARIA GAETANA; Costi, Maria Paola; D'Arca, Domenico; Cecconi, Ciro
Current Treatments to Control African Trypanosomiasis and One Health Perspective
2022 Venturelli, Alberto; Tagliazucchi, Lorenzo; Lima, Clara; Venuti, Federica; Malpezzi, Giulia; Magoulas, George E.; Santarem, Nuno; Calogeropoulou, Theodora; Cordeiro-da-Silva, Anabela; Costi, Maria Paola
design, synthesis and biological evaluation of novel YAP:TEAD complex disruptors for thetreatment of colorectal cancer
2023 Tagliazucchi, Lorenzo; Venturelli, Alberto; Malpezzi, Giulia; Zappaterra, Dana; Aiello, Daniele; Elisi, GIAN MARCO; Mor, Marco; Moschella, MARIA GAETANA; Marverti, Gaetano; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola
Designing selective Cys-ligands to unpair the binding of the Human Transcription Enhancer Associated Domain 4 (hTEAD-4) with its modulators to halt cancer cell growth
2021 Tagliazucchi, Lorenzo; Malpezzi, Giulia; Pozzi, Cecilia; Lopresti, Ludovica; Venturelli, Alberto; D'Arca, Domenico; Marverti, Gaetano; Cecconi, Ciro; Ponterini, Glauco; Costi, Maria Paola
Development of a novel class of YAP:TEAD interface-3 molecular disruptors to treat colorectal carcinoma
2023 Tagliazucchi, Lorenzo; Malpezzi, Giulia; Aiello, Daniele; Zappaterra, Dana; Elisi, GIAN MARCO; Venturelli, Alberto; Moschella, MARIA GAETANA; D'Arca, Domenico; Marverti, Gaetano; Lopresti, Ludovica; Pozzi, Cecilia; Pacifico, Salvatore; Guerrini, Remo; Ponterini, Glauco; Costi, Maria Paola
Exploiting Forster Resonance Energy Transfer (FRET) in the characterization of YAP:TEAD complex disruption
2022 Tagliazucchi, Lorenzo; Rossi, Marianna; Malpezzi, Giulia; Zappaterra, Dana; Aiello, Daniele; Pozzi, Cecilia; Pacifico, Salvatore; Guerrini, Remo; Venturelli, Alberto; Ponterini, Glauco; Costi, Maria Paola
Exploiting the Optical Tweezer technology to reveal thymidylate synthase interactions with its consensus mRNA
2023 Malpezzi, Giulia; Viander, Xavier; Zaltron, Annamaria; Neri, Benedetta; Di Felice, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Moschella, MARIA GAETANA; Costi, Maria Paola; D'Arca, Domenico; Cecconi, Ciro
EXPLOITING THE OPTICAL TWEEZER, A SINGLE MOLECULE TECHNOLOGY, TO REVEAL THYMIDYLATE SYNTHASE INTERACTIONS WITH ITS CONSENSUS mRNA
2023 Malpezzi, Giulia; Viander, Xavier; Zaltron, Annamaria; Neri, Benedetta; Di Felice, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Moschella, Maria; Costi, Maria Paola; D’Arcae, Domenico; Cecconi, Ciro
Insights into host-target interaction from the proteome modulation analysis through untargeted LC-MS/MS Proteomics of drug resistant L infantum-THP1 infected cells
2023 Tagliazucchi, Lorenzo; Malpezzi, Giulia; Perea Martinez, Ana; Ignacio Manzano, José; Garcia-Hernandez, Raquel; Pinetti, Diego; Genovese, Filippo; Thorè, Eli; Brooks, Bryan W.; Bertram, Michael G.; Gamarro, Francisco; Costi, Maria Paola
Investigating the mechanism of action of the antiparasitic agent H80 through imaging techniques
2023 Malpezzi, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Venturelli, Alberto; CORDEIRO DA SILVA, Anabela; Santarem, Nuno; Ponterini, Glauco; Costi, Maria Paola
LC-MS/MS proteomics for the rapid and selective screening of drug resistances in Leishmania infantum clinical isolates
2023 Tagliazucchi, Lorenzo; Malpezzi, Giulia; Perea Martinez, Ana; Ignacio Manzano, José; Garcia-Hernandez, Raquel; Pinetti, Diego; Genovese, Filippo; Costi, Maria Paola
Lead optimization of human thymidylate synthase dimer disrupters: from computational studies to evaluation of their biological profiles
2023 Aiello, Daniele; Malpezzi, Giulia; Tagliazucchi, Lorenzo; Moschella, MARIA GAETANA; Giulia, Saporito; Venturelli, Alberto; Gluaco, Ponterini; D'Arca, Domenico; Marverti, Gaetano; Federico, Falchi; Costi, Maria Paola
Lead-optimization process and characterization of the dissociative effect applied to new dimer disrupters of human Thymidylate Synthase
2022 Aiello, Daniele; Ascione, Cristian; Tagliazucchi, Lorenzo; Malpezzi, Giulia; Cassanelli, Valentina; Ponterini, Glauco; D'Arca, Domenico; Marverti, Gaetano; Moschella, MARIA GAETANA; Falchi, Federico; Venturelli, Alberto; Costi, Maria Paola
Leveraging proteomic, bioinformatic and ecotoxicology models to select new targets overcoming L. Infantum drug resistent
2024 Tagliazucchi, Lorenzo; Malpezzi, Giulia; Brooks, Brain V.; Thorè, Eli S. J.; Bertram, Michael G.; Gammarro, Francisco; Costi, Maria Paola
Leveraging proteomics, bioinformatics, and ecotoxicology models to select new targets overcoming L infantum drug resistance.
2024 Tagliazucchi, Lorenzo; Malpezzi, Giulia; Brooks, Bryan W.; Thoré, Eli S. J.; Bertram, Michael G.; Gamarro, Francisco; Costi, Maria Paola
Targeting of the Cysteines Surface domain of the Transcriptional Enhancer Associate Domain (TEAD) for anticancer drug discovery
2021 Tagliazucchi, Lorenzo; Malpezzi, Giulia; Mangani, Stefano; Lopresti, Ludovica; Pozzi, Cecilia; Ponterini, Glauco; Venturelli, Alberto; Costi, Maria Paola
UHPLC-MS/MS screening of the hTEAD surface for the identification of novel allosteric inhibitors with anticancer activity
2021 Tagliazucchi, Lorenzo; Malpezzi, Giulia; Pozzi, Cecilia; Lopresti, Ludovica; Mangani, Stefano; ABDEL LATIF, Andrea; Ponterini, Glauco; Venturelli, Alberto; Costi, Maria Paola
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A toolbox of biophysical and analytical assays helps to confirm the activity of novel hTS dimer disrupters (Ddis) with anticancer properties | 1-gen-2022 | Tagliazucchi, Lorenzo; Venturelli, Alberto; Malpezzi, Giulia; Moschella, MARIA GAETANA; Aiello, Daniele; Lopresti, Ludovica; Pozzi, Cecilia; Marverti, Gaetano; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola | |
Applying optical tweezers technology to reveal Thymidylate Synthase interactions with its consensus mRNA | 1-gen-2023 | Malpezzi, Giulia; Viader, Xvaier; Zaltron, Annamaria; Neri, Benedetta; di Felice, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Moschella, MARIA GAETANA; Costi, Maria Paola; D'Arca, Domenico; Cecconi, Ciro | |
Current Treatments to Control African Trypanosomiasis and One Health Perspective | 1-gen-2022 | Venturelli, Alberto; Tagliazucchi, Lorenzo; Lima, Clara; Venuti, Federica; Malpezzi, Giulia; Magoulas, George E.; Santarem, Nuno; Calogeropoulou, Theodora; Cordeiro-da-Silva, Anabela; Costi, Maria Paola | |
design, synthesis and biological evaluation of novel YAP:TEAD complex disruptors for thetreatment of colorectal cancer | 1-gen-2023 | Tagliazucchi, Lorenzo; Venturelli, Alberto; Malpezzi, Giulia; Zappaterra, Dana; Aiello, Daniele; Elisi, GIAN MARCO; Mor, Marco; Moschella, MARIA GAETANA; Marverti, Gaetano; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola | |
Designing selective Cys-ligands to unpair the binding of the Human Transcription Enhancer Associated Domain 4 (hTEAD-4) with its modulators to halt cancer cell growth | 1-gen-2021 | Tagliazucchi, Lorenzo; Malpezzi, Giulia; Pozzi, Cecilia; Lopresti, Ludovica; Venturelli, Alberto; D'Arca, Domenico; Marverti, Gaetano; Cecconi, Ciro; Ponterini, Glauco; Costi, Maria Paola | |
Development of a novel class of YAP:TEAD interface-3 molecular disruptors to treat colorectal carcinoma | 1-gen-2023 | Tagliazucchi, Lorenzo; Malpezzi, Giulia; Aiello, Daniele; Zappaterra, Dana; Elisi, GIAN MARCO; Venturelli, Alberto; Moschella, MARIA GAETANA; D'Arca, Domenico; Marverti, Gaetano; Lopresti, Ludovica; Pozzi, Cecilia; Pacifico, Salvatore; Guerrini, Remo; Ponterini, Glauco; Costi, Maria Paola | |
Exploiting Forster Resonance Energy Transfer (FRET) in the characterization of YAP:TEAD complex disruption | 1-gen-2022 | Tagliazucchi, Lorenzo; Rossi, Marianna; Malpezzi, Giulia; Zappaterra, Dana; Aiello, Daniele; Pozzi, Cecilia; Pacifico, Salvatore; Guerrini, Remo; Venturelli, Alberto; Ponterini, Glauco; Costi, Maria Paola | |
Exploiting the Optical Tweezer technology to reveal thymidylate synthase interactions with its consensus mRNA | 1-gen-2023 | Malpezzi, Giulia; Viander, Xavier; Zaltron, Annamaria; Neri, Benedetta; Di Felice, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Moschella, MARIA GAETANA; Costi, Maria Paola; D'Arca, Domenico; Cecconi, Ciro | |
EXPLOITING THE OPTICAL TWEEZER, A SINGLE MOLECULE TECHNOLOGY, TO REVEAL THYMIDYLATE SYNTHASE INTERACTIONS WITH ITS CONSENSUS mRNA | 1-gen-2023 | Malpezzi, Giulia; Viander, Xavier; Zaltron, Annamaria; Neri, Benedetta; Di Felice, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Moschella, Maria; Costi, Maria Paola; D’Arcae, Domenico; Cecconi, Ciro | |
Insights into host-target interaction from the proteome modulation analysis through untargeted LC-MS/MS Proteomics of drug resistant L infantum-THP1 infected cells | 1-gen-2023 | Tagliazucchi, Lorenzo; Malpezzi, Giulia; Perea Martinez, Ana; Ignacio Manzano, José; Garcia-Hernandez, Raquel; Pinetti, Diego; Genovese, Filippo; Thorè, Eli; Brooks, Bryan W.; Bertram, Michael G.; Gamarro, Francisco; Costi, Maria Paola | |
Investigating the mechanism of action of the antiparasitic agent H80 through imaging techniques | 1-gen-2023 | Malpezzi, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Venturelli, Alberto; CORDEIRO DA SILVA, Anabela; Santarem, Nuno; Ponterini, Glauco; Costi, Maria Paola | |
LC-MS/MS proteomics for the rapid and selective screening of drug resistances in Leishmania infantum clinical isolates | 1-gen-2023 | Tagliazucchi, Lorenzo; Malpezzi, Giulia; Perea Martinez, Ana; Ignacio Manzano, José; Garcia-Hernandez, Raquel; Pinetti, Diego; Genovese, Filippo; Costi, Maria Paola | |
Lead optimization of human thymidylate synthase dimer disrupters: from computational studies to evaluation of their biological profiles | 1-gen-2023 | Aiello, Daniele; Malpezzi, Giulia; Tagliazucchi, Lorenzo; Moschella, MARIA GAETANA; Giulia, Saporito; Venturelli, Alberto; Gluaco, Ponterini; D'Arca, Domenico; Marverti, Gaetano; Federico, Falchi; Costi, Maria Paola | |
Lead-optimization process and characterization of the dissociative effect applied to new dimer disrupters of human Thymidylate Synthase | 1-gen-2022 | Aiello, Daniele; Ascione, Cristian; Tagliazucchi, Lorenzo; Malpezzi, Giulia; Cassanelli, Valentina; Ponterini, Glauco; D'Arca, Domenico; Marverti, Gaetano; Moschella, MARIA GAETANA; Falchi, Federico; Venturelli, Alberto; Costi, Maria Paola | |
Leveraging proteomic, bioinformatic and ecotoxicology models to select new targets overcoming L. Infantum drug resistent | 1-gen-2024 | Tagliazucchi, Lorenzo; Malpezzi, Giulia; Brooks, Brain V.; Thorè, Eli S. J.; Bertram, Michael G.; Gammarro, Francisco; Costi, Maria Paola | |
Leveraging proteomics, bioinformatics, and ecotoxicology models to select new targets overcoming L infantum drug resistance. | 1-gen-2024 | Tagliazucchi, Lorenzo; Malpezzi, Giulia; Brooks, Bryan W.; Thoré, Eli S. J.; Bertram, Michael G.; Gamarro, Francisco; Costi, Maria Paola | |
Targeting of the Cysteines Surface domain of the Transcriptional Enhancer Associate Domain (TEAD) for anticancer drug discovery | 1-gen-2021 | Tagliazucchi, Lorenzo; Malpezzi, Giulia; Mangani, Stefano; Lopresti, Ludovica; Pozzi, Cecilia; Ponterini, Glauco; Venturelli, Alberto; Costi, Maria Paola | |
UHPLC-MS/MS screening of the hTEAD surface for the identification of novel allosteric inhibitors with anticancer activity | 1-gen-2021 | Tagliazucchi, Lorenzo; Malpezzi, Giulia; Pozzi, Cecilia; Lopresti, Ludovica; Mangani, Stefano; ABDEL LATIF, Andrea; Ponterini, Glauco; Venturelli, Alberto; Costi, Maria Paola |