SAPORITO, GIULIA
SAPORITO, GIULIA
Dipartimento di Scienze della Vita
Drug discovery of pyrazolo-piperidinone inhibitors targeting YAP:TEAD interaction and development of a fluorescence anisotropy assay for high-throughput screening
2025 Malpezzi, Giulia; Scalvini, Laura; Tagliazucchi, Lorenzo; Chiaravalle, Annalisa; Aiello, Daniele; Saporito, Giulia; Illuminati, Davide; Pacifico, Salvatore; Guerrini, Remo; Pozzi, Cecilia; Venturelli, Alberto; Ponterini, Glauco; Mor Sheraz Gul, Marco; Costi, Maria Paola
Identification of Innovative Folate Inhibitors Leveraging the Amino Dihydrotriazine Motif from Cycloguanil for Their Potential as Anti-Trypanosoma brucei Agents
2024 Francesconi, Valeria; Rizzo, Marco; Pozzi, Cecilia; Tagliazucchi, Lorenzo; Konchie Simo, Claude U.; Saporito, Giulia; Landi, Giacomo; Mangani, Stefano; Carbone, Anna; Schenone, Silvia; Santarém, Nuno; Tavares, Joana; Cordeiro-da-Silva, Anabela; Costi, Maria Paola; Tonelli, Michele
IDENTIFICATION OF PYRAZOLO-PIPERIDINONE DERIVATIVES TARGETING YAP-TEAD INTERFACE 3 AS ANTICANCER AGENTS THROUGH INTEGRATED VIRTUAL SCREENING AND MASS SPECTROMETRY PROTEOMICS
2025 Scalvini, Laura; Tagliazucchi, Lorenzo; Elisi, Gian Marco; Zappaterra, Dana; Moschella, Maria Gaetana; Fantini, Sebastian; Aiello, Daniele; Guerrini, Remo; Albanese, Valentina; Pacifico, Salvatore; Lopresti, Ludovica; Malpezzi, Giulia; Saporito, Giulia; Ferrari, Stefania; Lamesta, Michele; Losi, Lorena; Pozzi, Cecilia; Mangani, Stefano; Marverti, Gaetano; Venturelli, Alberto; Ponterini, Glauco; D'Arca, Domenico; Mor, Marco; Costi, Maria Paola
MS Proteomics And Biochemical Characterization Of Thymidylate Synthase Dimer Destabilizer E7 To Halt Colorectal Carcinoma
2024 Tagliazucchi, Lorenzo; DI PERSIO, Sara; Moschella, MARIA GAETANA; Malpezzi, Giulia; Aiello, Daniele; Saporito, Giulia; Bedeschi, Martina; Tesei, Anna; Passardi, Alessandro; Marverti, Gaetano; Venturelli, Alberto; D’Arca, Domenico; Costi, Maria Paola
Optimization of chemical-biological tools for characterizing the activity of dissociative inhibitor of human thymidylate synthase
2024 Saporito, Giulia; Aiello, Daniele; Malpezzi, Giulia; Tagliazucchi, Lorenzo; Venturelli, Alberto; Falchi, Federico; Ponterini, Glauco; Costi, Maria Paola
Promoting A Sustainable Medicinal Chemistry Approach With The Cost Action CA21111 - One Health Drugs Against Parasitic Vector Borne Diseases In Europe And Beyond
2024 Aiello, Daniele; Cordeiro-da-Silva, Anabela; Tagliazucchi, Lorenzo; Saporito, Giulia; Malpezzi, Giulia; Action CA2111 Members, Cost; Costi, Maria Paola
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Drug discovery of pyrazolo-piperidinone inhibitors targeting YAP:TEAD interaction and development of a fluorescence anisotropy assay for high-throughput screening | 1-gen-2025 | Malpezzi, Giulia; Scalvini, Laura; Tagliazucchi, Lorenzo; Chiaravalle, Annalisa; Aiello, Daniele; Saporito, Giulia; Illuminati, Davide; Pacifico, Salvatore; Guerrini, Remo; Pozzi, Cecilia; Venturelli, Alberto; Ponterini, Glauco; Mor Sheraz Gul, Marco; Costi, Maria Paola | |
| Identification of Innovative Folate Inhibitors Leveraging the Amino Dihydrotriazine Motif from Cycloguanil for Their Potential as Anti-Trypanosoma brucei Agents | 1-gen-2024 | Francesconi, Valeria; Rizzo, Marco; Pozzi, Cecilia; Tagliazucchi, Lorenzo; Konchie Simo, Claude U.; Saporito, Giulia; Landi, Giacomo; Mangani, Stefano; Carbone, Anna; Schenone, Silvia; Santarém, Nuno; Tavares, Joana; Cordeiro-da-Silva, Anabela; Costi, Maria Paola; Tonelli, Michele | |
| IDENTIFICATION OF PYRAZOLO-PIPERIDINONE DERIVATIVES TARGETING YAP-TEAD INTERFACE 3 AS ANTICANCER AGENTS THROUGH INTEGRATED VIRTUAL SCREENING AND MASS SPECTROMETRY PROTEOMICS | 1-gen-2025 | Scalvini, Laura; Tagliazucchi, Lorenzo; Elisi, Gian Marco; Zappaterra, Dana; Moschella, Maria Gaetana; Fantini, Sebastian; Aiello, Daniele; Guerrini, Remo; Albanese, Valentina; Pacifico, Salvatore; Lopresti, Ludovica; Malpezzi, Giulia; Saporito, Giulia; Ferrari, Stefania; Lamesta, Michele; Losi, Lorena; Pozzi, Cecilia; Mangani, Stefano; Marverti, Gaetano; Venturelli, Alberto; Ponterini, Glauco; D'Arca, Domenico; Mor, Marco; Costi, Maria Paola | |
| MS Proteomics And Biochemical Characterization Of Thymidylate Synthase Dimer Destabilizer E7 To Halt Colorectal Carcinoma | 1-gen-2024 | Tagliazucchi, Lorenzo; DI PERSIO, Sara; Moschella, MARIA GAETANA; Malpezzi, Giulia; Aiello, Daniele; Saporito, Giulia; Bedeschi, Martina; Tesei, Anna; Passardi, Alessandro; Marverti, Gaetano; Venturelli, Alberto; D’Arca, Domenico; Costi, Maria Paola | |
| Optimization of chemical-biological tools for characterizing the activity of dissociative inhibitor of human thymidylate synthase | 1-gen-2024 | Saporito, Giulia; Aiello, Daniele; Malpezzi, Giulia; Tagliazucchi, Lorenzo; Venturelli, Alberto; Falchi, Federico; Ponterini, Glauco; Costi, Maria Paola | |
| Promoting A Sustainable Medicinal Chemistry Approach With The Cost Action CA21111 - One Health Drugs Against Parasitic Vector Borne Diseases In Europe And Beyond | 1-gen-2024 | Aiello, Daniele; Cordeiro-da-Silva, Anabela; Tagliazucchi, Lorenzo; Saporito, Giulia; Malpezzi, Giulia; Action CA2111 Members, Cost; Costi, Maria Paola |
