Sfoglia per Autore
Ring opening effect at alpha1-adrenoceptor subtypes and 5-HT1A receptors within a novel class of 1,3-Dioxolane-based ligands
2004 Brasili, Livio; Franchini, Silvia; Prandi, Adolfo; P., Angeli; G., Marucci; M., Buccioni; A., Leonardi; E., Poggesi
1,3-Diossolani e analoghi aperti come nuovi ligandi per il recettore Sigma
2004 Franchini, Silvia; Prandi, Adolfo; Paini, Silvia; Paini, Stefania; O., Prezzavento; G., Ronsisvalle; Brasili, Livio
Relazioni struttura-attività in una nuova serie di ligandi alpha1-adrenergici e 5-HT1A serotoninergici a struttura 2,2-difenil-[1,3]diossolanica
2004 Prandi, Adolfo; Franchini, Silvia; Sorbi, Claudia; Cancian, Laura; P., Angeli; G., Marucci; A., Leonardi; E., Poggesi; Brasili, Livio
Risoluzione della miscela racemica del (±)-(2,2-difenil-[1,3]diossolan-4-ilmetil)-(2-fenossi-etil) ammina, potente antagonista alpha1 adrenergico,
2004 Prandi, Adolfo; Franchini, Silvia; Siligardi, Cristian; P., Angeli; G., Marucci; Brasili, Livio
C3a and C3b activation products of the third component of complement (C3) are critical for normal liver recovery after toxic injury
2004 Markiewski, M. M; Mastellos, D; Tudoran, R; Deangelis, R. A; Strey, C. W; Franchini, Silvia; Wetsel, R. A; Erdei, A; Lambris, J. D.
Novel monoclonal antibodies against mouse C3 interfering with complement activation: Description of fine specificity and applications to various immunoassays
2004 Mastellos, D; Prechl, J; Lszl, G; Papp, K; Olh, E; Argyropoulos, E; Franchini, Silvia; Tudoran, R; Markiewski, M; Lambris, J. D.; Erdei, A.
Benzothiadiazine derivatives as 1 and 5-HT1A receptor ligands.
2005 Tait, Annalisa; Franchini, Silvia; M., Buccioni; G., Marucci; A., Leonardi; E., Poggesi; Brasili, Livio
SAR at alpha1-adrenoceptor subtypes and 5-HT1A receptors within a novel series of 1,3-Dioxolane-based ligands.
2005 Brasili, Livio; Franchini, Silvia; Prandi, A.; Tait, A.; Angeli, P.; Marucci, G.; Leonardi, A.; Poggesi, E.
Second Joint Italian-Swiss Meeting on Medicinal Chemistry , Italy, Modena 19-20 February 2005.
2005 Brasili, Livio; Benvenuti, Stefania; Costantino, Luca; Costi, Maria Paola; Philipp, Floersheim; Franchini, Silvia; Gamberini, Gianfranco; Parenti, Carlo; Rastelli, Giulio; Rustichelli, Cecilia; Tait, Annalisa; Tondi, Donatella
Synthesis and antimuscarinic activity of derivatives of 2-substituted-1,3-dioxolanes
2005 Marucci, G; Angeli, P; Brasili, Livio; Buccioni, M; Giardinà, D; Gulini, U; Piergentili, A; Sagratini, G; Franchini, Silvia
1,2,4-Benzothiadiazine derivatives as alpha(1) and 5-HT1A receptor ligands
2005 Tait, Annalisa; Luppi, Amedeo; Franchini, Silvia; E., Preziosi; Parenti, Carlo; M., Buccioni; G., Marucci; A., Leonardi; E., Poggesi; Brasili, Livio
Synthesis and structure-activity relationships of 1-aralkyl-4- benzylpiperidine and 1-aralkyl-4-benzylpiperazine derivatives as potent σ ligands
2005 Costantino, Luca; Gandolfi, Francesca; Sorbi, Claudia; Franchini, Silvia; Prezzavento, O; Vittorio, F; Ronsisvalle, G; Leopardi, A; Poggesi, E; Brasili, Livio
Alternative strategies in medicinal chemistry to face drug resistance in anticancer therapy.
2006 Cardinale, Daniela; Ferrari, Stefania; Franchini, Silvia; Corsini, Enrico; Battini, Renata; Costi, Maria Paola
Structure Activity Relationship at 5-HT1A receptors within a novel series of spiro-1,3-Dioxolane-based ligands
2006 Franchini, Silvia; Prandi, Adolfo; Baraldi, Anna Maria; P., Angeli; G., Marucci; M., Buccioni; A., Leonardi; E., Poggesi; G., Motta; Brasili, Livio
Synthesis and biological evaluations of 4-alkyl-1-Arylpiperazine derivatives: SAR at 5-HT1A and 1 –Adrenoreceptor
2006 Franchini, Silvia; Prandi, Adolfo; Baraldi, Anna Maria; G., Marucci; M., Buccioni; P., Angeli; A., Leonardi; E., Poggesi; G., Motta; Brasili, Livio
Synthesis and pharmacological evaluation of 1-benzylpiperazine and 4-benzylpiperidine as potent sigma ligands.
2007 Baraldi, Anna Maria; Franchini, Silvia; Prandi, Adolfo; O., Prezzavento; G., Ronsisvalle; L., Pirona; Brasili, Livio
Merging disulphide bonds for drug design Interfering with a cancer key protein
2008 Lazzari, Sandra; Venturelli, Alberto; G., Cruciani; Franchini, Silvia; S., Henrich; Genovese, Filippo; R. C., Wade; Costi, Maria Paola
Investigation within a new series of heterocyclic biaryl piperazines acting at 5-HT1A serotoninergic receptors
2008 Franchini, Silvia; M., Borriello; Prandi, Adolfo; Baraldi, Anna Maria; R., Di Fabio; Brasili, Livio
1-(1,4-Dioxa-spiro[4.5]dec-2ylmethyl)-4-(2-methoxy-phenyl)-piperazine: SAR at alpha1 and 5-HT1A Receptors.
2009 Baraldi, Anna Maria; Franchini, Silvia; Manasieva, LEDA IVANOVAA; A., Cilia; E., Poggesi; Brasili, Livio
Structure Activity Relationships at 5-HT1A receptors within a novel series of 4-alkyl-1-arylpiperazine derivatives
2009 Baraldi, Anna Maria; Franchini, Silvia; Manasieva, LEDA IVANOVAA; Sorbi, Claudia; A., Cilia; E., Poggesi; Brasili, Livio
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Ring opening effect at alpha1-adrenoceptor subtypes and 5-HT1A receptors within a novel class of 1,3-Dioxolane-based ligands | 1-gen-2004 | Brasili, Livio; Franchini, Silvia; Prandi, Adolfo; P., Angeli; G., Marucci; M., Buccioni; A., Leonardi; E., Poggesi | |
1,3-Diossolani e analoghi aperti come nuovi ligandi per il recettore Sigma | 1-gen-2004 | Franchini, Silvia; Prandi, Adolfo; Paini, Silvia; Paini, Stefania; O., Prezzavento; G., Ronsisvalle; Brasili, Livio | |
Relazioni struttura-attività in una nuova serie di ligandi alpha1-adrenergici e 5-HT1A serotoninergici a struttura 2,2-difenil-[1,3]diossolanica | 1-gen-2004 | Prandi, Adolfo; Franchini, Silvia; Sorbi, Claudia; Cancian, Laura; P., Angeli; G., Marucci; A., Leonardi; E., Poggesi; Brasili, Livio | |
Risoluzione della miscela racemica del (±)-(2,2-difenil-[1,3]diossolan-4-ilmetil)-(2-fenossi-etil) ammina, potente antagonista alpha1 adrenergico, | 1-gen-2004 | Prandi, Adolfo; Franchini, Silvia; Siligardi, Cristian; P., Angeli; G., Marucci; Brasili, Livio | |
C3a and C3b activation products of the third component of complement (C3) are critical for normal liver recovery after toxic injury | 1-gen-2004 | Markiewski, M. M; Mastellos, D; Tudoran, R; Deangelis, R. A; Strey, C. W; Franchini, Silvia; Wetsel, R. A; Erdei, A; Lambris, J. D. | |
Novel monoclonal antibodies against mouse C3 interfering with complement activation: Description of fine specificity and applications to various immunoassays | 1-gen-2004 | Mastellos, D; Prechl, J; Lszl, G; Papp, K; Olh, E; Argyropoulos, E; Franchini, Silvia; Tudoran, R; Markiewski, M; Lambris, J. D.; Erdei, A. | |
Benzothiadiazine derivatives as 1 and 5-HT1A receptor ligands. | 1-gen-2005 | Tait, Annalisa; Franchini, Silvia; M., Buccioni; G., Marucci; A., Leonardi; E., Poggesi; Brasili, Livio | |
SAR at alpha1-adrenoceptor subtypes and 5-HT1A receptors within a novel series of 1,3-Dioxolane-based ligands. | 1-gen-2005 | Brasili, Livio; Franchini, Silvia; Prandi, A.; Tait, A.; Angeli, P.; Marucci, G.; Leonardi, A.; Poggesi, E. | |
Second Joint Italian-Swiss Meeting on Medicinal Chemistry , Italy, Modena 19-20 February 2005. | 1-gen-2005 | Brasili, Livio; Benvenuti, Stefania; Costantino, Luca; Costi, Maria Paola; Philipp, Floersheim; Franchini, Silvia; Gamberini, Gianfranco; Parenti, Carlo; Rastelli, Giulio; Rustichelli, Cecilia; Tait, Annalisa; Tondi, Donatella | |
Synthesis and antimuscarinic activity of derivatives of 2-substituted-1,3-dioxolanes | 1-gen-2005 | Marucci, G; Angeli, P; Brasili, Livio; Buccioni, M; Giardinà, D; Gulini, U; Piergentili, A; Sagratini, G; Franchini, Silvia | |
1,2,4-Benzothiadiazine derivatives as alpha(1) and 5-HT1A receptor ligands | 1-gen-2005 | Tait, Annalisa; Luppi, Amedeo; Franchini, Silvia; E., Preziosi; Parenti, Carlo; M., Buccioni; G., Marucci; A., Leonardi; E., Poggesi; Brasili, Livio | |
Synthesis and structure-activity relationships of 1-aralkyl-4- benzylpiperidine and 1-aralkyl-4-benzylpiperazine derivatives as potent σ ligands | 1-gen-2005 | Costantino, Luca; Gandolfi, Francesca; Sorbi, Claudia; Franchini, Silvia; Prezzavento, O; Vittorio, F; Ronsisvalle, G; Leopardi, A; Poggesi, E; Brasili, Livio | |
Alternative strategies in medicinal chemistry to face drug resistance in anticancer therapy. | 1-gen-2006 | Cardinale, Daniela; Ferrari, Stefania; Franchini, Silvia; Corsini, Enrico; Battini, Renata; Costi, Maria Paola | |
Structure Activity Relationship at 5-HT1A receptors within a novel series of spiro-1,3-Dioxolane-based ligands | 1-gen-2006 | Franchini, Silvia; Prandi, Adolfo; Baraldi, Anna Maria; P., Angeli; G., Marucci; M., Buccioni; A., Leonardi; E., Poggesi; G., Motta; Brasili, Livio | |
Synthesis and biological evaluations of 4-alkyl-1-Arylpiperazine derivatives: SAR at 5-HT1A and 1 –Adrenoreceptor | 1-gen-2006 | Franchini, Silvia; Prandi, Adolfo; Baraldi, Anna Maria; G., Marucci; M., Buccioni; P., Angeli; A., Leonardi; E., Poggesi; G., Motta; Brasili, Livio | |
Synthesis and pharmacological evaluation of 1-benzylpiperazine and 4-benzylpiperidine as potent sigma ligands. | 1-gen-2007 | Baraldi, Anna Maria; Franchini, Silvia; Prandi, Adolfo; O., Prezzavento; G., Ronsisvalle; L., Pirona; Brasili, Livio | |
Merging disulphide bonds for drug design Interfering with a cancer key protein | 1-gen-2008 | Lazzari, Sandra; Venturelli, Alberto; G., Cruciani; Franchini, Silvia; S., Henrich; Genovese, Filippo; R. C., Wade; Costi, Maria Paola | |
Investigation within a new series of heterocyclic biaryl piperazines acting at 5-HT1A serotoninergic receptors | 1-gen-2008 | Franchini, Silvia; M., Borriello; Prandi, Adolfo; Baraldi, Anna Maria; R., Di Fabio; Brasili, Livio | |
1-(1,4-Dioxa-spiro[4.5]dec-2ylmethyl)-4-(2-methoxy-phenyl)-piperazine: SAR at alpha1 and 5-HT1A Receptors. | 1-gen-2009 | Baraldi, Anna Maria; Franchini, Silvia; Manasieva, LEDA IVANOVAA; A., Cilia; E., Poggesi; Brasili, Livio | |
Structure Activity Relationships at 5-HT1A receptors within a novel series of 4-alkyl-1-arylpiperazine derivatives | 1-gen-2009 | Baraldi, Anna Maria; Franchini, Silvia; Manasieva, LEDA IVANOVAA; Sorbi, Claudia; A., Cilia; E., Poggesi; Brasili, Livio |
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