Sfoglia per Autore
Molecular structure and dynamics of some potent 5-HT3 receptor antagonists. Insight into the interaction with the receptor
1996 Cappelli, A; Donati, A; Anzini, M; Vomero, S; DE BENEDETTI, Pier Giuseppe; Menziani, Maria Cristina; Langer, T.
Computational simulations of stem-cell factor c-Kit receptor interaction
1996 Menziani, Maria Cristina; Fanelli, Francesca; DE BENEDETTI, Pier Giuseppe
Synthesis, biological evaluation, and quantitative receptor docking simulations of 2-[(acylamino)ethyl]-1,4-benzodiazepines as novel tifluadom-like ligands with high affinity and selectivity for kappa-opioid receptors
1996 Cappelli, A; Anzini, M; Vomero, S; Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe; Sbacchi, M; Clarke, Gd; Mennuni, L.
Alpha 1-adrenoceptor subtype selectivity: Molecular modelling and theoretical quantitative structure-affinity relationships
1997 DE BENEDETTI, Pier Giuseppe; Fanelli, Francesca; Menziani, Maria Cristina; Cocchi, Marina; R., Testa; A., Leonardi
Conformational analysis and theoretical quantitative size and shape-affinity relationships of N-4-protonated N-1-arylpiperazine 5-HT1A serotoninergic ligands
1997 Cocchi, Marina; Fanelli, Francesca; Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe
Theoretical investigation of IL-6 multiprotein receptor assembly
1997 Menziani, Maria Cristina; Fanelli, Francesca; DE BENEDETTI, Pier Giuseppe
Molecular dynamics of guest radicals in urea inclusion compounds
1997 Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe; Segre, Ulderico; Brustolon, M.
Constitutively active α1B-adrenergic receptor mutants: potential mechanisms underlying receptor activation
1997 A., Scheer; Fanelli, Francesca; T., Costa; DE BENEDETTI, Pier Giuseppe; S., Cotecchia
Theoretical descriptors in quantitative structure - Affinity and selectivity relationship study of potent N4-substituted arylpiperazine 5-HT1(Alpha) receptor antagonists
1998 Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe; Karelson, M.
Ab initio modeling and molecular dynamics simulation of the alpha 1b-adrenergic receptor activation
1998 Fanelli, Francesca; Menziani, Maria Cristina; A., Scheer; S., Cotecchia; DE BENEDETTI, Pier Giuseppe
Novel potent and selective central 5-HT3 receptor ligands provided with different intrinsic efficacy. 1. Mapping the central 5-HT3 receptor binding site by arylpiperazine derivatives
1998 Cappelli, A; Anzini, M; Vomero, S; Mennuni, L; Makovec, F; Doucet, E; Hamon, M; Bruni, G; Romeo, Mr; Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe; Langer, T.
Molecular mechanisms involved in the activation and regulation of the alpha 1-adrenergic receptor subtypes
1998 S., Cotecchia; A., Scheer; D., Diviani; Fanelli, Francesca; DE BENEDETTI, Pier Giuseppe
Computer modeling of size and shape descriptors of alpha 1-adrenergic receptor antagonists and quantitative structure-affinity/selectivity relationships
1998 Montorsi, Monia; Menziani, Maria Cristina; Cocchi, Marina; Fanelli, Francesca; DE BENEDETTI, Pier Giuseppe
Use of the supermolecule approach to derive molecular similarity descriptors for QSAR analysis.
1998 Cocchi, Marina; DE BENEDETTI, Pier Giuseppe
Constitutively active receptor mutants as probes for studying the mechanisms underlying G protein-coupled receptor activation
1999 S., Cotecchia; Fanelli, Francesca; A., Scheer; DE BENEDETTI, Pier Giuseppe
Structure-function relationships of the alpha(1b)-adrenergic receptor
1999 A., Scheer; Fanelli, Francesca; D., Diviani; DE BENEDETTI, Pier Giuseppe; S., Cotecchia
Relevance of theoretical molecular descriptors in quantitative structure-activity relationship analysis of alpha 1-adrenergic receptor antagonists
1999 Menziani, Maria Cristina; Montorsi, Monia; DE BENEDETTI, Pier Giuseppe; Karelson, M.
Activation mechanism of human oxytocin receptor: A combined study of experimental and computer-simulated mutagenesis
1999 Fanelli, Francesca; P., Barbier; D., Zanchetta; DE BENEDETTI, Pier Giuseppe; B., Chini
Novel potent and selective central 5-HT3 receptor ligands provided with different intrinsic efficacy. 2. Molecular basis of the intrinsic efficacy of arylpiperazine derivatives at the central 5-HT3 receptors
1999 Cappelli, A; Anzini, M; Vomero, S; Canullo, L; Mennuni, L; Makovec, F; Doucet, E; Hamon, M; Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe; Bruni, G; Romeo, Mr; Giorgi, G; Donati, A.
Synthesis, pharmacological evaluation, and structure-activity relationship and quantitative structure-activity relationship studies on novel derivatives of 2,4-diamino-6,7-dimethoxyquinazoline alpha(1)-adrenoceptor antagonists
1999 Leonardi, A; Motta, G; Boi, C; Testa, R; Poggesi, E; DE BENEDETTI, Pier Giuseppe; Menziani, Maria Cristina
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