Sfoglia per Autore
On the development of B-Raf inhibitors acting through innovative mechanisms
2022 Pinzi, L.
Development of machine learning classifiers to predict compound activity on prostate cancer cell lines
2022 Bonanni, Davide; Pinzi, Luca; Rastelli, Giulio
Dual Targeting Strategies On Histone Deacetylase 6 (HDAC6) And Heat Shock Protein 90 (Hsp90)
2022 Bonanni, Davide; Citarella, Andrea; Moi, Davide; Pinzi, Luca; Bergamini, Elisa; Rastelli, Giulio
Structure-activity exploration of a small-molecule allosteric inhibitor of T790M/L858R double mutant EGFR
2023 Foschi, FRANCESCA MADDALENA; Tinivella, Annachiara; Crippa, Valeria; Pinzi, Luca; Mologni, Luca; Passarella, Daniele; Rastelli, Giulio
Discovery of potent pyrrolo-pyrimidine and purine HDAC inhibitors for the treatment of advanced prostate cancer
2023 Moi, Davide; Bonanni, Davide; Belluti, Silvia; Linciano, Pasquale; Citarella, Andrea; Franchini, Silvia; Sorbi, Claudia; Imbriano, Carol; Pinzi, Luca; Rastelli, Giulio
Insights into the Structural Conformations of the Tau Protein in Different Aggregation Status
2023 Pinzi, L.; Bisi, N.; Sorbi, C.; Franchini, S.; Tonali, N.; Rastelli, G.
Design, synthesis, biological evaluation and crystal structure determination of dual modulators of carbonic anhydrases and estrogen receptors
2023 Tinivella, Annachiara; Nwachukwu, J. C.; Angeli, A.; Foschi, F.; Benatti, Annalaura; Pinzi, Luca; Izard, T.; Ferraroni, M.; Erumbi, R.; Christodoulou, M. S.; Passarella, D.; Supuran, C.; Nettles, K. W.; Rastelli, Giulio
Identification of Promising Drug Candidates against Prostate Cancer through Computationally-Driven Drug Repurposing
2023 Bernal, Leonardo; Pinzi, Luca; Rastelli, Giulio
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
On the development of B-Raf inhibitors acting through innovative mechanisms | 1-gen-2022 | Pinzi, L. | |
Development of machine learning classifiers to predict compound activity on prostate cancer cell lines | 1-gen-2022 | Bonanni, Davide; Pinzi, Luca; Rastelli, Giulio | |
Dual Targeting Strategies On Histone Deacetylase 6 (HDAC6) And Heat Shock Protein 90 (Hsp90) | 1-gen-2022 | Bonanni, Davide; Citarella, Andrea; Moi, Davide; Pinzi, Luca; Bergamini, Elisa; Rastelli, Giulio | |
Structure-activity exploration of a small-molecule allosteric inhibitor of T790M/L858R double mutant EGFR | 1-gen-2023 | Foschi, FRANCESCA MADDALENA; Tinivella, Annachiara; Crippa, Valeria; Pinzi, Luca; Mologni, Luca; Passarella, Daniele; Rastelli, Giulio | |
Discovery of potent pyrrolo-pyrimidine and purine HDAC inhibitors for the treatment of advanced prostate cancer | 1-gen-2023 | Moi, Davide; Bonanni, Davide; Belluti, Silvia; Linciano, Pasquale; Citarella, Andrea; Franchini, Silvia; Sorbi, Claudia; Imbriano, Carol; Pinzi, Luca; Rastelli, Giulio | |
Insights into the Structural Conformations of the Tau Protein in Different Aggregation Status | 1-gen-2023 | Pinzi, L.; Bisi, N.; Sorbi, C.; Franchini, S.; Tonali, N.; Rastelli, G. | |
Design, synthesis, biological evaluation and crystal structure determination of dual modulators of carbonic anhydrases and estrogen receptors | 1-gen-2023 | Tinivella, Annachiara; Nwachukwu, J. C.; Angeli, A.; Foschi, F.; Benatti, Annalaura; Pinzi, Luca; Izard, T.; Ferraroni, M.; Erumbi, R.; Christodoulou, M. S.; Passarella, D.; Supuran, C.; Nettles, K. W.; Rastelli, Giulio | |
Identification of Promising Drug Candidates against Prostate Cancer through Computationally-Driven Drug Repurposing | 1-gen-2023 | Bernal, Leonardo; Pinzi, Luca; Rastelli, Giulio |
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