Sfoglia per Rivista ACS INFECTIOUS DISEASES
1,2,3-Triazolylmethaneboronate: A Structure Activity Relationship Study of a Class of β-Lactamase Inhibitors against Acinetobacter baumannii Cephalosporinase
2020 Caselli, E.; Fini, F.; Introvigne, M. L.; Stucchi, M.; Taracila, M. A.; Fish, E. R.; Smolen, K. A.; Rather, P. N.; Powers, R. A.; Wallar, B. J.; Bonomo, R. A.; Prati, F.
Assessing Environmental Risks during the Drug Development Process for Parasitic Vector-Borne Diseases: A Critical Reflection
2024 Ilbeigi, K.; Barata, C.; Barbosa, J.; Bertram, M. G.; Caljon, G.; Costi, M. P.; Kroll, A.; Margiotta-Casaluci, L.; Thoré, E. S. J.; Bundschuh, M.
Call for Papers: One Health and Vector-Borne Parasitic Diseases
2023 Costi, Maria P.; Cordeiro-da-Silva, Anabela
Deciphering Host–Parasite Interplay in Leishmania Infection through a One Health View of Proteomics Studies on Drug Resistance
2024 Tagliazucchi, Lorenzo; Pinetti, Diego; Genovese, Filippo; Malpezzi, Giulia; Perea Martinez, Ana; Manzano, José I.; García-Hernández, Raquel; Cole, Alexander R.; Kwon, Ba Reum; Aiello, Daniele; Brooks, Bryan W.; Thoré, Eli S. J.; Bertram, Michael G.; Gamarro, Francisco; Costi, Maria Paola
Identification of Innovative Folate Inhibitors Leveraging the Amino Dihydrotriazine Motif from Cycloguanil for Their Potential as Anti-Trypanosoma brucei Agents
2024 Francesconi, Valeria; Rizzo, Marco; Pozzi, Cecilia; Tagliazucchi, Lorenzo; Konchie Simo, Claude U.; Saporito, Giulia; Landi, Giacomo; Mangani, Stefano; Carbone, Anna; Schenone, Silvia; Santarém, Nuno; Tavares, Joana; Cordeiro-da-Silva, Anabela; Costi, Maria Paola; Tonelli, Michele
Inhibiting the β-Lactamase of Mycobacterium tuberculosis (Mtb) with Novel Boronic Acid Transition-State Inhibitors (BATSIs)
2015 Kurz, Sebastian G.; Hazra, Saugata; Bethel, Christopher R.; Romagnoli, Chiara; Caselli, Emilia; Prati, Fabio; Blanchard, John S.; Bonomo, Robert A.
Inhibition of Acinetobacter -Derived Cephalosporinase: Exploring the Carboxylate Recognition Site Using Novel β-Lactamase Inhibitors
2018 Caselli, Emilia; Romagnoli, Chiara; Powers, Rachel A.; Taracila, Magdalena A.; Bouza, Alexandra A.; Swanson, Hollister C.; Smolen, Kali A.; Fini, Francesco; Wallar, Bradley J.; Bonomo, Robert A.; Prati, Fabio
Label-Free Mass Spectrometry Proteomics Reveals Different Pathways Modulated in THP-1 Cells Infected with Therapeutic Failure and Drug Resistance Leishmania infantum Clinical Isolates
2023 Tagliazucchi, Lorenzo; Perea-Martinez, Ana; Fiorini, Greta; Ignacio Manzano, José; Genovese, Filippo; García-Hernández, Raquel; Pinetti, Diego; GAMARRO CONDE, Francisco; Costi, Maria Paola
Structural Insights into the Development of Cycloguanil Derivatives as Trypanosoma brucei Pteridine-Reductase-1 Inhibitors
2019 Landi, G.; Linciano, P.; Borsari, C.; Bertolacini, C. P.; Moraes, C. B.; Cordeiro-Da-Silva, A.; Gul, S.; Witt, G.; Kuzikov, M.; Costi, M. P.; Pozzi, C.; Mangani, S.
Structure-Based Analysis of Boronic Acids as Inhibitors of Acinetobacter-Derived Cephalosporinase-7, a Unique Class C β-Lactamase
2018 Bouza, Alexandra A; Swanson, Hollister C; Smolen, Kali A; Vandine, Alison L; Taracila, Magdalena A; Romagnoli, Chiara; Caselli, Emilia; Prati, Fabio; Bonomo, Robert A; Powers, Rachel A; Wallar, Bradley J
Ten years with NDM-1 metallo β-lactamase: from structural insights to inhibitor design
2019 Linciano, Pasquale; Cendron, Laura; Gianquinto, Eleonora; Spyrakis, Francesca; Tondi, Donatella
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
1,2,3-Triazolylmethaneboronate: A Structure Activity Relationship Study of a Class of β-Lactamase Inhibitors against Acinetobacter baumannii Cephalosporinase | 1-gen-2020 | Caselli, E.; Fini, F.; Introvigne, M. L.; Stucchi, M.; Taracila, M. A.; Fish, E. R.; Smolen, K. A.; Rather, P. N.; Powers, R. A.; Wallar, B. J.; Bonomo, R. A.; Prati, F. | |
Assessing Environmental Risks during the Drug Development Process for Parasitic Vector-Borne Diseases: A Critical Reflection | 1-gen-2024 | Ilbeigi, K.; Barata, C.; Barbosa, J.; Bertram, M. G.; Caljon, G.; Costi, M. P.; Kroll, A.; Margiotta-Casaluci, L.; Thoré, E. S. J.; Bundschuh, M. | |
Call for Papers: One Health and Vector-Borne Parasitic Diseases | 1-gen-2023 | Costi, Maria P.; Cordeiro-da-Silva, Anabela | |
Deciphering Host–Parasite Interplay in Leishmania Infection through a One Health View of Proteomics Studies on Drug Resistance | 1-gen-2024 | Tagliazucchi, Lorenzo; Pinetti, Diego; Genovese, Filippo; Malpezzi, Giulia; Perea Martinez, Ana; Manzano, José I.; García-Hernández, Raquel; Cole, Alexander R.; Kwon, Ba Reum; Aiello, Daniele; Brooks, Bryan W.; Thoré, Eli S. J.; Bertram, Michael G.; Gamarro, Francisco; Costi, Maria Paola | |
Identification of Innovative Folate Inhibitors Leveraging the Amino Dihydrotriazine Motif from Cycloguanil for Their Potential as Anti-Trypanosoma brucei Agents | 1-gen-2024 | Francesconi, Valeria; Rizzo, Marco; Pozzi, Cecilia; Tagliazucchi, Lorenzo; Konchie Simo, Claude U.; Saporito, Giulia; Landi, Giacomo; Mangani, Stefano; Carbone, Anna; Schenone, Silvia; Santarém, Nuno; Tavares, Joana; Cordeiro-da-Silva, Anabela; Costi, Maria Paola; Tonelli, Michele | |
Inhibiting the β-Lactamase of Mycobacterium tuberculosis (Mtb) with Novel Boronic Acid Transition-State Inhibitors (BATSIs) | 1-gen-2015 | Kurz, Sebastian G.; Hazra, Saugata; Bethel, Christopher R.; Romagnoli, Chiara; Caselli, Emilia; Prati, Fabio; Blanchard, John S.; Bonomo, Robert A. | |
Inhibition of Acinetobacter -Derived Cephalosporinase: Exploring the Carboxylate Recognition Site Using Novel β-Lactamase Inhibitors | 1-gen-2018 | Caselli, Emilia; Romagnoli, Chiara; Powers, Rachel A.; Taracila, Magdalena A.; Bouza, Alexandra A.; Swanson, Hollister C.; Smolen, Kali A.; Fini, Francesco; Wallar, Bradley J.; Bonomo, Robert A.; Prati, Fabio | |
Label-Free Mass Spectrometry Proteomics Reveals Different Pathways Modulated in THP-1 Cells Infected with Therapeutic Failure and Drug Resistance Leishmania infantum Clinical Isolates | 1-gen-2023 | Tagliazucchi, Lorenzo; Perea-Martinez, Ana; Fiorini, Greta; Ignacio Manzano, José; Genovese, Filippo; García-Hernández, Raquel; Pinetti, Diego; GAMARRO CONDE, Francisco; Costi, Maria Paola | |
Structural Insights into the Development of Cycloguanil Derivatives as Trypanosoma brucei Pteridine-Reductase-1 Inhibitors | 1-gen-2019 | Landi, G.; Linciano, P.; Borsari, C.; Bertolacini, C. P.; Moraes, C. B.; Cordeiro-Da-Silva, A.; Gul, S.; Witt, G.; Kuzikov, M.; Costi, M. P.; Pozzi, C.; Mangani, S. | |
Structure-Based Analysis of Boronic Acids as Inhibitors of Acinetobacter-Derived Cephalosporinase-7, a Unique Class C β-Lactamase | 1-gen-2018 | Bouza, Alexandra A; Swanson, Hollister C; Smolen, Kali A; Vandine, Alison L; Taracila, Magdalena A; Romagnoli, Chiara; Caselli, Emilia; Prati, Fabio; Bonomo, Robert A; Powers, Rachel A; Wallar, Bradley J | |
Ten years with NDM-1 metallo β-lactamase: from structural insights to inhibitor design | 1-gen-2019 | Linciano, Pasquale; Cendron, Laura; Gianquinto, Eleonora; Spyrakis, Francesca; Tondi, Donatella |
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