PINZI, LUCA

PINZI, LUCA  

Dipartimento di Scienze della Vita  

Mostra records
Risultati 1 - 20 di 47 (tempo di esecuzione: 0.029 secondi).
Titolo Data di pubblicazione Autore(i) File
2-Phenyloxazole-4-carboxamide as a Scaffold for Selective Inhibition of Human Monoamine Oxidase B 1-gen-2019 Di Paolo, M. L.; Christodoulou, M. S.; Calogero, A. M.; Pinzi, L.; Rastelli, G.; Passarella, D.; Cappelletti, G.; Dalla Via, L.
An unexpected reversal in the pharmacological stereoselectivity of benzothiadiazine AMPA positive allosteric modulators 1-gen-2016 Battisti, UMBERTO MARIA; Citti, Cinzia; Rastelli, Giulio; Pinzi, Luca; Puja, Giulia; Ravazzini, Federica; Ciccarella, Giuseppe; Braghiroli, Daniela; Cannazza, Giuseppe
Antifungal Activity and DNA Topoisomerase Inhibition of Hydrolysable Tannins from Punica granatum L. 1-gen-2021 Brighenti, V.; Iseppi, R.; Pinzi, L.; Mincuzzi, A.; Ippolito, A.; Messi, P.; Sanzani, S. M.; Rastelli, G.; Pellati, F.
Chemoinformatics Analyses of Tau Ligands Reveal Key Molecular Requirements for the Identification of Potential Drug Candidates against Tauopathies 1-gen-2021 Pinzi, Luca; Tinivella, Annachiara; Rastelli, Giulio
Computational polypharmacology comes of age 1-gen-2015 Rastelli, Giulio; Pinzi, Luca
Design and Synthesis of Hsp90 Inhibitors with B-Raf and PDHK1 Multi-Target Activity 1-gen-2021 Pinzi, L.; Foschi, F.; Christodoulou, M. S.; Passarella, D.; Rastelli, G.
Design of dual inhibitors of histone deacetylase 6 and heat shock protein 90 1-gen-2020 Pinzi, L.; Benedetti, R.; Altucci, L.; Rastelli, G.
Design, synthesis, biological evaluation and crystal structure determination of dual modulators of carbonic anhydrases and estrogen receptors 1-gen-2023 Tinivella, Annachiara; Nwachukwu, J. C.; Angeli, A.; Foschi, F.; Benatti, Annalaura; Pinzi, Luca; Izard, T.; Ferraroni, M.; Erumbi, R.; Christodoulou, M. S.; Passarella, D.; Supuran, C.; Nettles, K. W.; Rastelli, Giulio
Development and application of LigAdvisor, a user-friendly web-platform for polypharmacology and drug repurposing 1-gen-2021 Pinzi, Luca; Tinivella, Annachiara; Rastelli, Giulio
Development of machine learning classifers to predict compound activity on prostate cancer cell lines. 1-gen-2022 Bonanni, Davide; Pinzi, Luca; Rastelli, Giulio
Discovery of potent pyrrolo-pyrimidine and purine HDAC inhibitors for the treatment of advanced prostate cancer 1-gen-2023 Moi, Davide; Bonanni, Davide; Belluti, Silvia; Linciano, Pasquale; Citarella, Andrea; Franchini, Silvia; Sorbi, Claudia; Imbriano, Carol; Pinzi, Luca; Rastelli, Giulio
Drug Repurposing and Polypharmacology to Fight SARS-CoV-2 Through Inhibition of the Main Protease 1-gen-2021 Pinzi, Luca; Tinivella, Annachiara; Caporuscio, Fabiana; Rastelli, Giulio
Dual Targeting Strategies On Histone Deacetylase 6 (HDAC6) And Heat Shock Protein 90 (Hsp90) 1-gen-2022 Bonanni, Davide; Citarella, Andrea; Moi, Davide; Pinzi, Luca; Bergamini, Elisa; Rastelli, Giulio
Evaluation of Amides, Carbamates, Sulfonamides, and Ureas of 4-Prop-2-ynylidenecycloalkylamine as Potent, Selective, and Bioavailable Negative Allosteric Modulators of Metabotropic Glutamate Receptor 5 1-gen-2019 Graziani, Davide; Caligari, Silvia; Callegari, Elisa; De Toma, Carlo; Longhi, Matteo; Frigerio, Fabio; Dilernia, Roberto; Menegon, Sergio; Pinzi, Luca; Pirona, Lorenza; Tazzari, Valerio; Valsecchi, Anna Elisa; Vistoli, Giulio; Rastelli, Giulio; Ruga Riva, Carlo
Heat shock protein 90 and serine/threonine kinase B-Raf inhibitors have overlapping chemical space 1-gen-2017 Anighoro, A.; Pinzi, Luca; Marverti, Gaetano; Bajorath, J; Rastelli, Giulio
Hydroxamic Acid Derivatives: From Synthetic Strategies to Medicinal Chemistry Applications 1-gen-2021 Citarella, A.; Moi, D.; Pinzi, L.; Bonanni, D.; Rastelli, G.
Identification of 4-aryl-1H-pyrrole[2,3-b]pyridine derivatives for the development of new B-Raf inhibitors 1-gen-2018 Pinzi, Luca; Anighoro, Andrew; Bajorath, Jürgen; Rastelli, Giulio
Identification of potential biological targets of oxindole scaffolds via in silico repositioning strategies 1-gen-2022 Tinivella, Annachiara; Pinzi, Luca; Gambacorta, Guido; Baxendale, Ian; Rastelli, Giulio
Identification of Promising Drug Candidates against Prostate Cancer through Computationally-Driven Drug Repurposing 1-gen-2023 Bernal, Leonardo; Pinzi, Luca; Rastelli, Giulio
Identification of small-molecule EGFR allosteric inhibitors by high-Throughput docking 1-gen-2018 Caporuscio, Fabiana; Tinivella, Annachiara; Restelli, Valentina; Semrau, Marta S; Pinzi, Luca; Storici, Paola; Broggini, Massimo; Rastelli, Giulio