Sfoglia per Autore
On-line racemization by high-performance liquid chromatography
2009 Cannazza, Giuseppe; Carrozzo, Marina Maria; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Parenti, Carlo
Simultaneous Determination of Enantiomerizationand Hydrolysis Kinetic Parameters of ChiralN-Alkylbenzothiadiazine Derivatives
2010 Carrozzo, Marina Maria; Cannazza, Giuseppe; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Parenti, Carlo
Quantitative analysis of acetylcholine in rat brain microdialysates by liquid chromatography coupled with electrospray ionization tandem mass spectrometry
2010 Carrozzo, Marina Maria; Cannazza, Giuseppe; Pinetti, Diego; DI VIESTI, Vittoria; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Parenti, Carlo; Baraldi, Mario
Epimerization and hydrolysis of 3,6-dimethyl-2,3,5,6-tetrahydro[1,2,4]thiadiazino[6,5,4-hi]indole 1,1-dioxide
2010 Carrozzo, Marina Maria; Cannazza, Giuseppe; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Troisi, Luigino; Parenti, Carlo
Determination of kinetic parameters of enantiomerization of benzothiadiazines by DCXplorer
2010 CANNAZZA, Giuseppe; CARROZZO, Marina Maria; BATTISTI, UMBERTO MARIA; BRAGHIROLI, Daniela; PARENTI, Carlo; Troisi, Alessandro; Troisi, Luigino
Regioselective reduction of 3-substituted 2,3-dihydrobenzothiadiazines with borohydrides
2010 Battisti, UMBERTO MARIA; Cannazza, Giuseppe; M. M., Carrozzo; Braghiroli, Daniela; Parenti, Carlo; F., Rosato; L., Troisi
Molecular modeling studies, synthesis, configurational stability and biological activity of 8-chloro-2,3,5,6-tetrahydro-3,6-dimethyl-pyrrolo[1,2,3-de]-1,2,4-benzothiadiazine 1,1-dioxide
2011 Battisti, UMBERTO MARIA; Carrozzo, Marina Maria; Cannazza, Giuseppe; Puja, Giulia; Giulia, ; L., Troisi; Braghiroli, Daniela; Parenti, Carlo; K., Jozwiak
Evaluation of stereo and chemical stability of chiral compounds
2011 Cannazza, Giuseppe; Battisti, UMBERTO MARIA; Carrozzo, Marina Maria; Brasili, Livio; Braghiroli, Daniela; Parenti, Carlo
Regioselective cyclization of chloroacylaminobenzenesulfonamide derivatives
2012 Carrozzo, Marina Maria; Battisti, UMBERTO MARIA; Cannazza, Giuseppe; C., Citti; Parenti, Carlo; L., Troisi
Efficient synthesis of 5,6-dihydro-8H-[1,2,4]thiadiazino[6,5,4-de] phenanthridine 4,4-dioxide and 5,6-dihydro-8H-[1,2,4]-thiadiazino[6,5,4-ij] thieno[2,3-c]quinoline 4,4-dioxide
2012 Battisti, UMBERTO MARIA; Carrozzo, Marina Maria; Cannazza, Giuseppe; Braghiroli, Daniela; Parenti, Carlo; Brasili, Livio; Cinzia, Citti; Luigino, Troisi
Structure-affinity/activity relationships of 1,4-dioxa-spiro[4.5]decane based ligands at α1 and 5-HT1A receptors
2014 Franchini, Silvia; Battisti, UMBERTO MARIA; Baraldi, Anna Maria; Prandi, Adolfo; Fossa, Paola; Cichero, Elena; Tait, Annalisa; Sorbi, Claudia; Marucci, Gabriella; Cilia, Antonio; Pirona, Lorenza; Brasili, Livio
Design, stereoselective synthesis, configurational stability and biological activity of 7-chloro-9-(furan-3-yl)-2,3,3a,4-tetrahydro-1H-benzo[e]pyrrolo[2,1-c][1,2,4]thiadiazine 5,5-dioxide
2014 Carrozzo, Marina Maria; Battisti, UMBERTO MARIA; Cannazza, Giuseppe; Puja, Giulia; Ravazzini, Federica; Falchicchio, Aurelia; Perrone, Serena; Citti, Cinzia; Jozwiak, Krzysztof; Braghiroli, Daniela; Parenti, Carlo; Troisi, Luigino
Transacetalization of Acetals with Butane-1,2,4-triol Using Cobalt(II) Chloride and Chlorotrimethylsilane
2014 Battisti, UMBERTO MARIA; Sorbi, Claudia; Franchini, Silvia; Tait, Annalisa; Brasili, Livio
A New and Versatile Synthesis of 1,3-Dioxan-5-yl-pyrimidine and Purine Nucleoside Analogues
2015 Sorbi, Claudia; Prandi, Adolfo; Battisti, UMBERTO MARIA; Franchini, Silvia; Cornia, Andrea; Balzarini, Jan; Jeong, Lak Shin; Lee, Sang Kook; Song, Jayoung; Brasili, Livio
Synthesis of Heteroaryl ortho-Phenoxyethylamines via Suzuki Cross-Coupling: Easy Access to New Potential Scaffolds in Medicinal Chemistry
2015 Manasieva, Leda Ivanova; Battisti, UMBERTO MARIA; Prandi, Adolfo; Brasili, Livio; Franchini, Silvia
Enantiomeric resolution of [(2,2-diphenyl-1,3-dioxolan-4-yl)methyl](2-phenoxyethyl)amine, a potent α1and 5-HT1Areceptor ligand: an in vitro and computational study
2015 Franchini, Silvia; Baraldi, Anna Maria; Sorbi, Claudia; Pellati, Federica; Cichero, Elena; Battisti, UMBERTO MARIA; Angeli, Piero; Cilia, Antonio; Brasili, Livio
Synthesis, biological evaluation and molecular modelling of 1-oxa-4-thiaspiro- and 1,4-dithiaspiro[4.5]decane derivatives as potent and selective 5-HT1A receptor agonists
2016 Sorbi, Claudia; Franchini, Silvia; Manasieva, Leda Ivanova; Battisti, UMBERTO MARIA; Fossa, Paola; Cichero, Elena; Denora, Nunzio; Iacobazzi, Rosa Maria; Cilia, Antonio; Pirona, Lorenza; Brasili, Livio
An unexpected reversal in the pharmacological stereoselectivity of benzothiadiazine AMPA positive allosteric modulators
2016 Battisti, UMBERTO MARIA; Citti, Cinzia; Rastelli, Giulio; Pinzi, Luca; Puja, Giulia; Ravazzini, Federica; Ciccarella, Giuseppe; Braghiroli, Daniela; Cannazza, Giuseppe
Scouting new sigma receptor ligands: Synthesis, pharmacological evaluation and molecular modeling of 1,3-dioxolane-based structures and derivatives
2016 Franchini, Silvia; Battisti, UMBERTO MARIA; Prandi, Adolfo; Tait, Annalisa; Borsari, Chiara; Cichero, Elena; Fossa, Paola; Cilia, Antonio; Prezzavento, Orazio; Ronsisvalle, Simone; Aricò, Giuseppina; Parenti, Carmela; Brasili, Livio
7-Chloro-5-(furan-3-yl)-3-methyl-4H-benzo[e][1,2,4]thiadiazine 1,1-Dioxide as Positive Allosteric Modulator of α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor. The End of the Unsaturated-Inactive Paradigm?
2016 Citti, Cinzia; Battisti, UMBERTO MARIA; Cannazza, Giuseppe; Jozwiak, Krzysztof; Stasiak, Natalia; Puja, Giulia; Ravazzini, Federica; Ciccarella, Giuseppe; Braghiroli, Daniela; Parenti, Carlo; Troisi, Luigino; Zoli, Michele
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
On-line racemization by high-performance liquid chromatography | 1-gen-2009 | Cannazza, Giuseppe; Carrozzo, Marina Maria; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Parenti, Carlo | |
Simultaneous Determination of Enantiomerizationand Hydrolysis Kinetic Parameters of ChiralN-Alkylbenzothiadiazine Derivatives | 1-gen-2010 | Carrozzo, Marina Maria; Cannazza, Giuseppe; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Parenti, Carlo | |
Quantitative analysis of acetylcholine in rat brain microdialysates by liquid chromatography coupled with electrospray ionization tandem mass spectrometry | 1-gen-2010 | Carrozzo, Marina Maria; Cannazza, Giuseppe; Pinetti, Diego; DI VIESTI, Vittoria; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Parenti, Carlo; Baraldi, Mario | |
Epimerization and hydrolysis of 3,6-dimethyl-2,3,5,6-tetrahydro[1,2,4]thiadiazino[6,5,4-hi]indole 1,1-dioxide | 1-gen-2010 | Carrozzo, Marina Maria; Cannazza, Giuseppe; Battisti, UMBERTO MARIA; Braghiroli, Daniela; Troisi, Luigino; Parenti, Carlo | |
Determination of kinetic parameters of enantiomerization of benzothiadiazines by DCXplorer | 1-gen-2010 | CANNAZZA, Giuseppe; CARROZZO, Marina Maria; BATTISTI, UMBERTO MARIA; BRAGHIROLI, Daniela; PARENTI, Carlo; Troisi, Alessandro; Troisi, Luigino | |
Regioselective reduction of 3-substituted 2,3-dihydrobenzothiadiazines with borohydrides | 1-gen-2010 | Battisti, UMBERTO MARIA; Cannazza, Giuseppe; M. M., Carrozzo; Braghiroli, Daniela; Parenti, Carlo; F., Rosato; L., Troisi | |
Molecular modeling studies, synthesis, configurational stability and biological activity of 8-chloro-2,3,5,6-tetrahydro-3,6-dimethyl-pyrrolo[1,2,3-de]-1,2,4-benzothiadiazine 1,1-dioxide | 1-gen-2011 | Battisti, UMBERTO MARIA; Carrozzo, Marina Maria; Cannazza, Giuseppe; Puja, Giulia; Giulia, ; L., Troisi; Braghiroli, Daniela; Parenti, Carlo; K., Jozwiak | |
Evaluation of stereo and chemical stability of chiral compounds | 1-gen-2011 | Cannazza, Giuseppe; Battisti, UMBERTO MARIA; Carrozzo, Marina Maria; Brasili, Livio; Braghiroli, Daniela; Parenti, Carlo | |
Regioselective cyclization of chloroacylaminobenzenesulfonamide derivatives | 1-gen-2012 | Carrozzo, Marina Maria; Battisti, UMBERTO MARIA; Cannazza, Giuseppe; C., Citti; Parenti, Carlo; L., Troisi | |
Efficient synthesis of 5,6-dihydro-8H-[1,2,4]thiadiazino[6,5,4-de] phenanthridine 4,4-dioxide and 5,6-dihydro-8H-[1,2,4]-thiadiazino[6,5,4-ij] thieno[2,3-c]quinoline 4,4-dioxide | 1-gen-2012 | Battisti, UMBERTO MARIA; Carrozzo, Marina Maria; Cannazza, Giuseppe; Braghiroli, Daniela; Parenti, Carlo; Brasili, Livio; Cinzia, Citti; Luigino, Troisi | |
Structure-affinity/activity relationships of 1,4-dioxa-spiro[4.5]decane based ligands at α<alpha>1 and 5-HT1A receptors | 1-gen-2014 | Franchini, Silvia; Battisti, UMBERTO MARIA; Baraldi, Anna Maria; Prandi, Adolfo; Fossa, Paola; Cichero, Elena; Tait, Annalisa; Sorbi, Claudia; Marucci, Gabriella; Cilia, Antonio; Pirona, Lorenza; Brasili, Livio | |
Design, stereoselective synthesis, configurational stability and biological activity of 7-chloro-9-(furan-3-yl)-2,3,3a,4-tetrahydro-1H-benzo[e]pyrrolo[2,1-c][1,2,4]thiadiazine 5,5-dioxide | 1-gen-2014 | Carrozzo, Marina Maria; Battisti, UMBERTO MARIA; Cannazza, Giuseppe; Puja, Giulia; Ravazzini, Federica; Falchicchio, Aurelia; Perrone, Serena; Citti, Cinzia; Jozwiak, Krzysztof; Braghiroli, Daniela; Parenti, Carlo; Troisi, Luigino | |
Transacetalization of Acetals with Butane-1,2,4-triol Using Cobalt(II) Chloride and Chlorotrimethylsilane | 1-gen-2014 | Battisti, UMBERTO MARIA; Sorbi, Claudia; Franchini, Silvia; Tait, Annalisa; Brasili, Livio | |
A New and Versatile Synthesis of 1,3-Dioxan-5-yl-pyrimidine and Purine Nucleoside Analogues | 1-gen-2015 | Sorbi, Claudia; Prandi, Adolfo; Battisti, UMBERTO MARIA; Franchini, Silvia; Cornia, Andrea; Balzarini, Jan; Jeong, Lak Shin; Lee, Sang Kook; Song, Jayoung; Brasili, Livio | |
Synthesis of Heteroaryl ortho-Phenoxyethylamines via Suzuki Cross-Coupling: Easy Access to New Potential Scaffolds in Medicinal Chemistry | 1-gen-2015 | Manasieva, Leda Ivanova; Battisti, UMBERTO MARIA; Prandi, Adolfo; Brasili, Livio; Franchini, Silvia | |
Enantiomeric resolution of [(2,2-diphenyl-1,3-dioxolan-4-yl)methyl](2-phenoxyethyl)amine, a potent α1and 5-HT1Areceptor ligand: an in vitro and computational study | 1-gen-2015 | Franchini, Silvia; Baraldi, Anna Maria; Sorbi, Claudia; Pellati, Federica; Cichero, Elena; Battisti, UMBERTO MARIA; Angeli, Piero; Cilia, Antonio; Brasili, Livio | |
Synthesis, biological evaluation and molecular modelling of 1-oxa-4-thiaspiro- and 1,4-dithiaspiro[4.5]decane derivatives as potent and selective 5-HT1A receptor agonists | 1-gen-2016 | Sorbi, Claudia; Franchini, Silvia; Manasieva, Leda Ivanova; Battisti, UMBERTO MARIA; Fossa, Paola; Cichero, Elena; Denora, Nunzio; Iacobazzi, Rosa Maria; Cilia, Antonio; Pirona, Lorenza; Brasili, Livio | |
An unexpected reversal in the pharmacological stereoselectivity of benzothiadiazine AMPA positive allosteric modulators | 1-gen-2016 | Battisti, UMBERTO MARIA; Citti, Cinzia; Rastelli, Giulio; Pinzi, Luca; Puja, Giulia; Ravazzini, Federica; Ciccarella, Giuseppe; Braghiroli, Daniela; Cannazza, Giuseppe | |
Scouting new sigma receptor ligands: Synthesis, pharmacological evaluation and molecular modeling of 1,3-dioxolane-based structures and derivatives | 1-gen-2016 | Franchini, Silvia; Battisti, UMBERTO MARIA; Prandi, Adolfo; Tait, Annalisa; Borsari, Chiara; Cichero, Elena; Fossa, Paola; Cilia, Antonio; Prezzavento, Orazio; Ronsisvalle, Simone; Aricò, Giuseppina; Parenti, Carmela; Brasili, Livio | |
7-Chloro-5-(furan-3-yl)-3-methyl-4H-benzo[e][1,2,4]thiadiazine 1,1-Dioxide as Positive Allosteric Modulator of α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor. The End of the Unsaturated-Inactive Paradigm? | 1-gen-2016 | Citti, Cinzia; Battisti, UMBERTO MARIA; Cannazza, Giuseppe; Jozwiak, Krzysztof; Stasiak, Natalia; Puja, Giulia; Ravazzini, Federica; Ciccarella, Giuseppe; Braghiroli, Daniela; Parenti, Carlo; Troisi, Luigino; Zoli, Michele |
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