Sfoglia per Autore
Collateral sensitivity to novel thymidylate synthase inhibitors correlates with folate cycle enzymes impairment in cisplatin-resistant human ovarian cancer cells
2009 Marverti, Gaetano; Ligabue, Alessio; G., Paglietti; P., Corona; S., Piras; G., Vitale; Guerrieri, Davide; Luciani, Rosaria; Costi, Maria Paola; Frassineti, Chiara; Moruzzi, Maria Stella
Ligand-Based Virtual Screening and ADME-Tox Guided Approach to Identify Triazolo-quinoxalines as Folate Cycle Inhibitors.
2010 E., Carosati; G., Sforna; M., Pippi; Marverti, Gaetano; Ligabue, Alessio; Guerrieri, Davide; S., Piras; Guaitoli, Giambattista; Luciani, Rosaria; Costi, Maria Paola; G., Cruciani
Crystal Structure of histidine-tagged human thymidylate synthase
2011 Pozzi, Cristina; Cardinale, Daniela; Guaitoli, G.; Tondi, Donatella; Luciani, Rosaria; Myllykallio, H.; Ferrari, Stefania; Costi, Maria Paola; Mangani, S.
Crystal Structure of human thymidylate synthase bound to a peptide inhibitor
2011 Pozzi, Cristina; Cardinale, Daniela; Guaitoli, G.; Tondi, Donatella; Luciani, Rosaria; Myllykallio, H.; Ferrari, Stefania; Costi, Maria Paola; Mangani, S.
Identification of the binding modes of N-phenylphthalimides inhibiting bacterial thymidylate synthase through X-ray crystallography screening.
2011 Mangani, S; Cancian, Laura; Leone, R; Pozzi, C; Lazzari, Sandra; Luciani, Rosaria; Ferrari, Stefania; Costi, Maria Paola
Virtual screening identification of nonfolate compounds, including a CNS drug, as antiparasitic agents inhibiting pteridine reductase
2011 Ferrari, Stefania; Morandi, Federica; Motiejunas, D.; Nerini, Erika; Henrich, S.; Luciani, Rosaria; Venturelli, Alberto; Lazzari, Sandra; Calo', Samuele; Gupta, S.; Hannaert, V.; Michels, P. A. M.; Wade, R. C.; Costi, Maria Paola
Erratum: Protein-protein interface-binding peptides inhibit the cancer therapy target human thymidylate synthase (Proceedings of the National Academy of Sciences of the United States of America (2011) 108, 34 (E542-E549) DOI: 10.1073/pnas.1104829108)
2011 Cardinale, D.; Guaitoli, G.; Tondi, D.; Luciani, R.; Henrich, S.; Salo-Ahen, O. M. H.; Ferrari, S.; Marverti, G.; Guerrieri, D.; Ligabue, A.; Frassineti, C.; Pozzi, C.; Mangani, S.; Fessas, D.; Guerrini, R.; Ponterini, G.; Wade, R. C.; Costi, M. P.
Protein–protein interface-binding peptides inhibit the cancer therapy target human thymidylate synthase
2011 Cardinale, Daniela; Guaitoli, Giambattista; Tondi, Donatella; Luciani, Rosaria; S., Henrich; O. M. H., Salo Ahen; Ferrari, Stefania; Marverti, Gaetano; Guerrieri, Davide; Ligabue, Alessio; Frassineti, Chiara; C., Pozzi; S., Mangani; D., Fessas; R., Guerrini; Ponterini, Glauco; R. C., Wade; Costi, Maria Paola
The structure of Enterococcus faecalis thymidylate synthase provides clues about folate bacterial metabolism
2012 C., Pozzi; Ferrari, Stefania; D., Cortesi; Luciani, Rosaria; R. M., Stroud; A., Catalano; Costi, Maria Paola; S., Mangani
Inhibitor of Ovarian Cancer Cells growth by Virtual Screening: A New Thiazole Derivative Targeting Human Thymidylate Synthase
2012 Emanuele, Carosati; Anna, Tochowicz; Marverti, Gaetano; Giambattista, Guaitoli; Paolo, Benedetti; Ferrari, Stefania; Robert M., Stroud; Janet Sue Finer, Moore; Luciani, Rosaria; Davide, Farina; Gabriele, Cruciani; Costi, Maria Paola
Structure-Based Selectivity Optimization of Piperidine–Pteridine Derivatives as Potent Leishmania Pteridine Reductase Inhibitors
2012 Paola, Corona; Gibellini, Federica; Saxena, Puneet; Luciani, Rosaria; Guerrieri, Davide; Nerini, Erika; Ferrari, Stefania; Costi, Maria Paola
2′-Deoxyuridine 5′-Monophosphate Substrate Displacement in Thymidylate Synthase through 6-Hydroxy-2H-naphtho[1,8-bc]furan-2-one Derivatives
2013 Ferrari, Stefania; Calò, S; Leone, R; Luciani, Rosaria; Costantino, Luca; Sammak, Susan; Di Pisa, F; Pozzi, C; Mangani, S; Costi, Maria Paola
Discovery of highly potent acid ceramidase inhibitors with in vitro tumor chemosensitizing activity
2013 Natalia, Realini; Carlos, Solorzano; Chiara, Pagliuca; Daniela, Pizzirani; Andrea, Armirotti; Luciani, Rosaria; Costi, Maria Paola; Tiziano, Bandiera; Daniele, Piomelli
NUOVE MOLECOLE, PER USO COME AGENTI ANTITUMORALI
2013 Costi, Maria Paola; Costantino, Luca; Sammak, Susan; Ponterini, Glauco; Ferrari, Stefania; Luciani, Rosaria; Farina, Davide Salvatore Francesco; Franchini, Silvia; Santucci, Matteo; Gabriele, Cruciani; Emanuele, Carosati
Development of flavonoids derivatives as leads against Leishmaniasis and Trypanosomiasis-invited lecture
2014 Borsari, Chiara; Luciani, Rosaria; Pozzi, Cecilia; Tait, Annalisa; Costantino, Luca; Pellati, Federica; Ferrari, Stefania; Costi, Maria Paola
2-[N-Alkyl(R-phenyl)-aminomethyl]-3-phenyl-7-trifluoromethylquinoxalines as anticancer agents inhibitors of folate enzymes
2014 Piras, Sandra; Carta, Antonio; Briguglio, Irene; Corona, Paola; Paglietti, Giuseppe; Luciani, Rosaria; Costi, Maria Paola; Ferrari, Stefania
Optimization of Peptides That Target Human Thymidylate Synthase to Inhibit Ovarian Cancer Cell Growth
2014 M., Pelà; Saxena, Puneet; Luciani, Rosaria; Santucci, Matteo; Ferrari, Stefania; Marverti, Gaetano; Marraccini, Chiara; Martello, Andrea; Pirondi, Silvia; Genovese, Filippo; S., Salvadori; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola; R., Guerrini
ANTICANCER DRUGS
2015 Costantino, Luca; Costi, Maria Paola; Ponterini, Glauco; Marverti, Gaetano; Franchini, Silvia; Tondi, Donatella; D'Arca, Domenico; Ferrari, Stefania; Luciani, Rosaria; Venturelli, Alberto; Sammak, Susan; Lauriola, Angela; Gozzi, Gaia
Maxwell A: F1000Prime Recommendation of Evaluation [Neres J et al., ACS Chem Biol 2014]. In F1000Prime, 09 Jan 2015; DOI: 10.3410/f.725248139.793502885. F1000Prime.com/725248139#eval793502885
2015 Maxwell, Anthony; Neres, J; Hartkoorn, Rc; Chiarelli, Lr; Gadupudi, Ramakrishna; Pasca, Mr; Mori, G; Venturelli, Alberto; Savina, S; Makarov, V; Kolly, Gs; Molteni, E; Binda, C; Dhar, N; Ferrari, Stefania; Brodin, P; Delorme, V; Landry, V; de Jesus Lopes Ribeiro, Al; Farina, Davide Salvatore Francesco; Saxena, Puneet; Pojer, F; Carta, Antonello; Luciani, Rosaria; Porta, Andrea; Zanoni, G; De Rossi, E; Costi, Maria Paola; Riccardi, G.
Characterization of 2,4-Diamino-6-oxo-1,6-dihydropyrimidin-5-yl Ureido Based Inhibitors of Trypanosoma brucei FolD and Testing for Antiparasitic Activity
2015 Eadsforth, T. C.; Pinto, A.; Luciani, R.; Tamborini, L.; Cullia, G.; De Micheli, C.; Marinelli, L.; Cosconati, S.; Novellino, E.; Lo Presti, L.; Cordeiro Da Silva, A.; Conti, P.; Hunter, W. N.; Costi, M. P.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Collateral sensitivity to novel thymidylate synthase inhibitors correlates with folate cycle enzymes impairment in cisplatin-resistant human ovarian cancer cells | 1-gen-2009 | Marverti, Gaetano; Ligabue, Alessio; G., Paglietti; P., Corona; S., Piras; G., Vitale; Guerrieri, Davide; Luciani, Rosaria; Costi, Maria Paola; Frassineti, Chiara; Moruzzi, Maria Stella | |
Ligand-Based Virtual Screening and ADME-Tox Guided Approach to Identify Triazolo-quinoxalines as Folate Cycle Inhibitors. | 1-gen-2010 | E., Carosati; G., Sforna; M., Pippi; Marverti, Gaetano; Ligabue, Alessio; Guerrieri, Davide; S., Piras; Guaitoli, Giambattista; Luciani, Rosaria; Costi, Maria Paola; G., Cruciani | |
Crystal Structure of histidine-tagged human thymidylate synthase | 1-gen-2011 | Pozzi, Cristina; Cardinale, Daniela; Guaitoli, G.; Tondi, Donatella; Luciani, Rosaria; Myllykallio, H.; Ferrari, Stefania; Costi, Maria Paola; Mangani, S. | |
Crystal Structure of human thymidylate synthase bound to a peptide inhibitor | 1-gen-2011 | Pozzi, Cristina; Cardinale, Daniela; Guaitoli, G.; Tondi, Donatella; Luciani, Rosaria; Myllykallio, H.; Ferrari, Stefania; Costi, Maria Paola; Mangani, S. | |
Identification of the binding modes of N-phenylphthalimides inhibiting bacterial thymidylate synthase through X-ray crystallography screening. | 1-gen-2011 | Mangani, S; Cancian, Laura; Leone, R; Pozzi, C; Lazzari, Sandra; Luciani, Rosaria; Ferrari, Stefania; Costi, Maria Paola | |
Virtual screening identification of nonfolate compounds, including a CNS drug, as antiparasitic agents inhibiting pteridine reductase | 1-gen-2011 | Ferrari, Stefania; Morandi, Federica; Motiejunas, D.; Nerini, Erika; Henrich, S.; Luciani, Rosaria; Venturelli, Alberto; Lazzari, Sandra; Calo', Samuele; Gupta, S.; Hannaert, V.; Michels, P. A. M.; Wade, R. C.; Costi, Maria Paola | |
Erratum: Protein-protein interface-binding peptides inhibit the cancer therapy target human thymidylate synthase (Proceedings of the National Academy of Sciences of the United States of America (2011) 108, 34 (E542-E549) DOI: 10.1073/pnas.1104829108) | 1-gen-2011 | Cardinale, D.; Guaitoli, G.; Tondi, D.; Luciani, R.; Henrich, S.; Salo-Ahen, O. M. H.; Ferrari, S.; Marverti, G.; Guerrieri, D.; Ligabue, A.; Frassineti, C.; Pozzi, C.; Mangani, S.; Fessas, D.; Guerrini, R.; Ponterini, G.; Wade, R. C.; Costi, M. P. | |
Protein–protein interface-binding peptides inhibit the cancer therapy target human thymidylate synthase | 1-gen-2011 | Cardinale, Daniela; Guaitoli, Giambattista; Tondi, Donatella; Luciani, Rosaria; S., Henrich; O. M. H., Salo Ahen; Ferrari, Stefania; Marverti, Gaetano; Guerrieri, Davide; Ligabue, Alessio; Frassineti, Chiara; C., Pozzi; S., Mangani; D., Fessas; R., Guerrini; Ponterini, Glauco; R. C., Wade; Costi, Maria Paola | |
The structure of Enterococcus faecalis thymidylate synthase provides clues about folate bacterial metabolism | 1-gen-2012 | C., Pozzi; Ferrari, Stefania; D., Cortesi; Luciani, Rosaria; R. M., Stroud; A., Catalano; Costi, Maria Paola; S., Mangani | |
Inhibitor of Ovarian Cancer Cells growth by Virtual Screening: A New Thiazole Derivative Targeting Human Thymidylate Synthase | 1-gen-2012 | Emanuele, Carosati; Anna, Tochowicz; Marverti, Gaetano; Giambattista, Guaitoli; Paolo, Benedetti; Ferrari, Stefania; Robert M., Stroud; Janet Sue Finer, Moore; Luciani, Rosaria; Davide, Farina; Gabriele, Cruciani; Costi, Maria Paola | |
Structure-Based Selectivity Optimization of Piperidine–Pteridine Derivatives as Potent Leishmania Pteridine Reductase Inhibitors | 1-gen-2012 | Paola, Corona; Gibellini, Federica; Saxena, Puneet; Luciani, Rosaria; Guerrieri, Davide; Nerini, Erika; Ferrari, Stefania; Costi, Maria Paola | |
2′-Deoxyuridine 5′-Monophosphate Substrate Displacement in Thymidylate Synthase through 6-Hydroxy-2H-naphtho[1,8-bc]furan-2-one Derivatives | 1-gen-2013 | Ferrari, Stefania; Calò, S; Leone, R; Luciani, Rosaria; Costantino, Luca; Sammak, Susan; Di Pisa, F; Pozzi, C; Mangani, S; Costi, Maria Paola | |
Discovery of highly potent acid ceramidase inhibitors with in vitro tumor chemosensitizing activity | 1-gen-2013 | Natalia, Realini; Carlos, Solorzano; Chiara, Pagliuca; Daniela, Pizzirani; Andrea, Armirotti; Luciani, Rosaria; Costi, Maria Paola; Tiziano, Bandiera; Daniele, Piomelli | |
NUOVE MOLECOLE, PER USO COME AGENTI ANTITUMORALI | 1-gen-2013 | Costi, Maria Paola; Costantino, Luca; Sammak, Susan; Ponterini, Glauco; Ferrari, Stefania; Luciani, Rosaria; Farina, Davide Salvatore Francesco; Franchini, Silvia; Santucci, Matteo; Gabriele, Cruciani; Emanuele, Carosati | |
Development of flavonoids derivatives as leads against Leishmaniasis and Trypanosomiasis-invited lecture | 1-gen-2014 | Borsari, Chiara; Luciani, Rosaria; Pozzi, Cecilia; Tait, Annalisa; Costantino, Luca; Pellati, Federica; Ferrari, Stefania; Costi, Maria Paola | |
2-[N-Alkyl(R-phenyl)-aminomethyl]-3-phenyl-7-trifluoromethylquinoxalines as anticancer agents inhibitors of folate enzymes | 1-gen-2014 | Piras, Sandra; Carta, Antonio; Briguglio, Irene; Corona, Paola; Paglietti, Giuseppe; Luciani, Rosaria; Costi, Maria Paola; Ferrari, Stefania | |
Optimization of Peptides That Target Human Thymidylate Synthase to Inhibit Ovarian Cancer Cell Growth | 1-gen-2014 | M., Pelà; Saxena, Puneet; Luciani, Rosaria; Santucci, Matteo; Ferrari, Stefania; Marverti, Gaetano; Marraccini, Chiara; Martello, Andrea; Pirondi, Silvia; Genovese, Filippo; S., Salvadori; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola; R., Guerrini | |
ANTICANCER DRUGS | 1-gen-2015 | Costantino, Luca; Costi, Maria Paola; Ponterini, Glauco; Marverti, Gaetano; Franchini, Silvia; Tondi, Donatella; D'Arca, Domenico; Ferrari, Stefania; Luciani, Rosaria; Venturelli, Alberto; Sammak, Susan; Lauriola, Angela; Gozzi, Gaia | |
Maxwell A: F1000Prime Recommendation of Evaluation [Neres J et al., ACS Chem Biol 2014]. In F1000Prime, 09 Jan 2015; DOI: 10.3410/f.725248139.793502885. F1000Prime.com/725248139#eval793502885 | 1-gen-2015 | Maxwell, Anthony; Neres, J; Hartkoorn, Rc; Chiarelli, Lr; Gadupudi, Ramakrishna; Pasca, Mr; Mori, G; Venturelli, Alberto; Savina, S; Makarov, V; Kolly, Gs; Molteni, E; Binda, C; Dhar, N; Ferrari, Stefania; Brodin, P; Delorme, V; Landry, V; de Jesus Lopes Ribeiro, Al; Farina, Davide Salvatore Francesco; Saxena, Puneet; Pojer, F; Carta, Antonello; Luciani, Rosaria; Porta, Andrea; Zanoni, G; De Rossi, E; Costi, Maria Paola; Riccardi, G. | |
Characterization of 2,4-Diamino-6-oxo-1,6-dihydropyrimidin-5-yl Ureido Based Inhibitors of Trypanosoma brucei FolD and Testing for Antiparasitic Activity | 1-gen-2015 | Eadsforth, T. C.; Pinto, A.; Luciani, R.; Tamborini, L.; Cullia, G.; De Micheli, C.; Marinelli, L.; Cosconati, S.; Novellino, E.; Lo Presti, L.; Cordeiro Da Silva, A.; Conti, P.; Hunter, W. N.; Costi, M. P. |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile