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Conformational analysis, molecular modeling and quantitative structure-activity relationships studies of 2,4-diamino-6,7-dimethoxy-2-substituted quinazoline α1-adrenergic antagonists 1-gen-1991 Rastelli, Giulio; Fanelli, Francesca; Menziani, Maria Cristina; Cocchi, Marina; DE BENEDETTI, Pier Giuseppe
Molecular modeling and quantitaive structure activity relationship analysis using theoretical descriptors of 1,4-benzodioxan (WB-4101) related-compounds alpha-1-adrenergic antagonists 1-gen-1992 P., Venturelli; Menziani, Maria Cristina; Cocchi, Marina; Fanelli, Francesca; DE BENEDETTI, Pier Giuseppe
Three dimensional molecular modeling of the α1a-adrenoceptor. Direct 3D-QSAR modeling of selective antagonists 1-gen-1993 Fanelli, Francesca; Menziani, Maria Cristina; Cocchi, Marina; DE BENEDETTI, Pier Giuseppe
The heuristic-direct approach to quantitative structure-activity relationship analysis 1-gen-1993 DE BENEDETTI, Pier Giuseppe; Menziani, Maria Cristina; Fanelli, Francesca; Cocchi, Marina
Theoretical quantitative structure-activity analysis and pharmacophore modelling of selective non congeneric α1a-adrenergic antagonists 1-gen-1993 DE BENEDETTI, Pier Giuseppe; Cocchi, Marina; Menziani, Maria Cristina; Fanelli, Francesca
Theoretical quantitative structure-activity analysis of quinuclidine-based muscarinic cholinergic receptor ligands 1-gen-1993 Fanelli, Francesca; Menziani, Maria Cristina; Carotti, A; DE BENEDETTI, Pier Giuseppe
Enantiomeric resolution of sulfoxides on a DACH‐DNB chiral stationary phase: A quantitative structure–enantioselective retention relationship (QSERR) study 1-gen-1993 C., Altomare; A., Carotti; S., Cellamare; Fanelli, Francesca; F., Gasparrini; C., Villani; P. A., Carrupt; B., Testa
Theoretical Quantitative Structure-Activity Relationship Analysis on Three Dimensional Models of Ligand-m1 Muscarinic Receptor Complexes 1-gen-1994 Fanelli, Francesca; Menziani, Maria Cristina; A., Carotti; P. G., DE BENEDETTI
The heuristic-direct approach to theoretical quantitative structure activity relationship analysis of α1- adrenoceptor ligands 1-gen-1994 Fanelli, Francesca; Menziani, Maria Cristina; Cocchi, Marina; A., Leonardi; DE BENEDETTI, Pier Giuseppe
Theoretical quantitative size and shape activity and selectivity analyses of 5-HT1A serotonin and α1-adrenergic receptor ligands 1-gen-1994 DE BENEDETTI, Pier Giuseppe; Cocchi, Marina; Menziani, Maria Cristina; Fanelli, Francesca
The Heuristic-Direct Approach to QSAR Analysis of Ligand-G-Protein Coupled Receptor Complexes 1-gen-1995 DE BENEDETTI, Pier Giuseppe; Menziani, Maria Cristina; Fanelli, Francesca; Cocchi, Marina
Theoretical QSAR analysis on three dimensional models of the complexes between peptide and non-peptide antagonists with the ETA and ETB receptors 1-gen-1995 Menziani, Maria Cristina; Cocchi, Marina; Fanelli, Francesca; DE BENEDETTI, Pier Giuseppe
Computer simulations of signal transduction mechanism in alpha 1B-adrenergic and m3-muscarinic receptors 1-gen-1995 Fanelli, Francesca; Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe
Comparative molecular dynamics study of the seven-helix bundle arrangement of G-protein coupled receptors 1-gen-1995 Fanelli, Francesca; Menziani, Maria Cristina; Cocchi, Marina; DE BENEDETTI, Pier Giuseppe
Quantitative structure-affinity/selectivity relationship analysis on three-dimensional models of the complexes between the ETA and ETB receptors and C-terminal endothelin hexapeptide antagonists 1-gen-1995 Menziani, Maria Cristina; Cocchi, Marina; Fanelli, Francesca; DE BENEDETTI, Pier Giuseppe
Prototropic molecular forms and theoretical descriptors in QSAR analysis 1-gen-1995 DE BENEDETTI, Pier Giuseppe; Menziani, Maria Cristina; Cocchi, Marina; Fanelli, Francesca
Molecular dynamics simulations of m3-muscarinic receptor activation and QSAR analysis 1-gen-1995 Fanelli, Francesca; Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe
Theoretical quantitative structure-activity relationship analysis of congeneric and non-congeneric α1-adrenoceptor antagonists: a chemometric study 1-gen-1995 Cocchi, Marina; Menziani, Maria Cristina; Fanelli, Francesca; DE BENEDETTI, Pier Giuseppe
The Heuristic-Direct approach to Quantitative Structure-Activity Relationship Analysis of Ligand-G Protein Coupled Receptor Complexes 1-gen-1996 Menziani, Maria Cristina; Fanelli, Francesca; Cocchi, Marina; DE BENEDETTI, Pier Giuseppe
Constitutively active mutants of the alpha 1B-adrenergic receptor: role of highly conserved polar amino acids in receptor activation 1-gen-1996 Scheer, A.; Fanelli, Francesca; Costa, T.; DE BENEDETTI, P. G.; Cotecchia, S.
Mostrati risultati da 1 a 20 di 165
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