Sfoglia per Autore
Update on antifolate drugs targets
2001 Costi, Maria Paola; Ferrari, Stefania
Dal Ligand based design di inibitori della Timidilato Sintasi all'Analisi Comparativa dei Complessi Enzima-Inibitore
2002 Costi, Maria Paola; Ferrari, Stefania; Pecorari, Piergiorgio; Rinaldi, Marcella; Tondi, Donatella; Venturelli, Alberto; Wade, R. C.
From ligand-based design to Hit validation of new thymidylate synthase inhibitors
2003 Costi, Maria Paola; Ferrari, Stefania; Rinaldi, Marcella; Tondi, Donatella; Wade, R. C.
Inhibitor Specificity via Protein Dynamics. Insights from the Design of Antibacterial Agents Targeted Against Thymidylate Synthase
2003 Ferrari, Stefania; Costi, Maria Paola; Wade, R. C.
Rapid-Throughput Technologies Applied to the Discovery of New Hits against Thymidylate synthase Enzymes
2004 Ferrari, Stefania; Malaguti, E; Calò, S; Tondi, Donatella; Venturelli, Alberto; Costi, Maria Paola
Medicinal chemistry in parasitology
2004 Costi, Maria Paola; Ferrari, Stefania; Rastelli, Giulio
Aza-boronic acids as non-beta-lactam inhibitors of AmpC-beta-lactamase
2004 Buzzoni, V.; Blazquez, J.; Ferrari, Stefania; Calo, S.; Venturelli, A.; Costi, Maria Paola
“A step further in the discovery of phthalein derivatives as Thymidylate Synthase inhibitors”
2004 Calo', Samuele; Tondi, Donatella; Venturelli, A.; Ferrari, Stefania; Pecorari, Piergiorgio; Rinaldi, Marcella; Ghelli, S.; Costi, Maria Paola
The structure of Cryptococcus neoformans thymidylate synthase suggests strategies for using target dynamics for species-specific inhibition
2005 JS Finer, Moore; Ac, Anderson; Rh, O'Neil; Costi, Maria Paola; Ferrari, Stefania; J., Krucinski; Rm, Stroud
Thymidylate synthase structure, function and implication in drug discovery
2005 Costi, Maria Paola; Ferrari, Stefania; Venturelli, A; Calo, S; Tondi, Donatella; Barlocco, D.
Improving specificity vs bacterial thymidylate synthases through N-dansyl modulation of didansyltyrosine
2005 Tondi, Donatella; Venturelli, A.; Ferrari, Stefania; Ghelli, S.; Costi, Maria Paola
Alternative strategies in medicinal chemistry to face drug resistance in anticancer therapy.
2006 Cardinale, Daniela; Ferrari, Stefania; Franchini, Silvia; Corsini, Enrico; Battini, Renata; Costi, Maria Paola
Antibacterial agent discovery using thymidylate synthase biolibrary screening
2006 Costi, Maria Paola; A., Gelain; D., Barlocco; S., Ghelli; Soragni, Fabrizia; F., Reniero; Rossi, Tiziana; Ruberto, Ippazio Antonio; C., Guillou; A., Cavazzuti; Casolari, Chiara; Ferrari, Stefania
Novel 3-benzoyl-2-piperazinylquinoxaline derivatives as potential antitumor agents
2006 S., Piras; M., Loriga; A., Carta; G., Paglietti; Costi, Maria Paola; Ferrari, Stefania
Congress on - Medicinal Chemistry in parasitology: new avenues in drug discovery-organised in Modena in 2007.
2007 Costi, Maria Paola; Ferrari, Stefania; Taramelli, D.; D., Gonzales Pacnowska
Interfering with Human Thymidylate Synthase Dimerization against ovarian human carcinoma
2007 Costi, Maria Paola; Cardinale, Daniela; Guaitoli, Giambattista; Tondi, Donatella; Ferrari, Stefania; Salo Ahen, O; Wade, R.
Interfering with Human Thymidylate Synthase Dimerization anti peptide design in the search of anticancer agents against ovarian human carcinoma
2007 Cardinale, Daniela; Salo Ahen, O; Guaitoli, Giambattista; Tondi, Donatella; Ferrari, Stefania; Wade, R; Costi, Maria Paola
Anti-Parasitic drugsDiscovery of potent pteridine reductase inhibitors to guide antiparasite drug development.
2008 Costi, Maria Paola; Ferrari, Stefania; Cavazzuti, Antonio
FRET-based assay for sensing a cancer key protein functional state and inhibition by oligopeptides: Sitespecific Protein Chemical Modifications
2008 Genovese, Filippo; M., Vargiu; M. A., Ariza Mateos; Guaitoli, Giambattista; Ferrari, Stefania; Ponterini, Glauco; Costi, Maria Paola
Discovery of potent pteridine reductase inhibitors to guide antiparasite drug development
2008 Cavazzuti, Antonio; Paglietti, G.; Hunter, W. N.; Gamarro, F.; Piras, S.; Loriga, M.; Alleca, S.; Corona, P.; Mcluskey, K.; Tulloch, L.; Gibellini, Federica; Ferrari, Stefania; Costi, Maria Paola
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Update on antifolate drugs targets | 1-gen-2001 | Costi, Maria Paola; Ferrari, Stefania | |
Dal Ligand based design di inibitori della Timidilato Sintasi all'Analisi Comparativa dei Complessi Enzima-Inibitore | 1-gen-2002 | Costi, Maria Paola; Ferrari, Stefania; Pecorari, Piergiorgio; Rinaldi, Marcella; Tondi, Donatella; Venturelli, Alberto; Wade, R. C. | |
From ligand-based design to Hit validation of new thymidylate synthase inhibitors | 1-gen-2003 | Costi, Maria Paola; Ferrari, Stefania; Rinaldi, Marcella; Tondi, Donatella; Wade, R. C. | |
Inhibitor Specificity via Protein Dynamics. Insights from the Design of Antibacterial Agents Targeted Against Thymidylate Synthase | 1-gen-2003 | Ferrari, Stefania; Costi, Maria Paola; Wade, R. C. | |
Rapid-Throughput Technologies Applied to the Discovery of New Hits against Thymidylate synthase Enzymes | 1-gen-2004 | Ferrari, Stefania; Malaguti, E; Calò, S; Tondi, Donatella; Venturelli, Alberto; Costi, Maria Paola | |
Medicinal chemistry in parasitology | 1-gen-2004 | Costi, Maria Paola; Ferrari, Stefania; Rastelli, Giulio | |
Aza-boronic acids as non-beta-lactam inhibitors of AmpC-beta-lactamase | 1-gen-2004 | Buzzoni, V.; Blazquez, J.; Ferrari, Stefania; Calo, S.; Venturelli, A.; Costi, Maria Paola | |
“A step further in the discovery of phthalein derivatives as Thymidylate Synthase inhibitors” | 1-gen-2004 | Calo', Samuele; Tondi, Donatella; Venturelli, A.; Ferrari, Stefania; Pecorari, Piergiorgio; Rinaldi, Marcella; Ghelli, S.; Costi, Maria Paola | |
The structure of Cryptococcus neoformans thymidylate synthase suggests strategies for using target dynamics for species-specific inhibition | 1-gen-2005 | JS Finer, Moore; Ac, Anderson; Rh, O'Neil; Costi, Maria Paola; Ferrari, Stefania; J., Krucinski; Rm, Stroud | |
Thymidylate synthase structure, function and implication in drug discovery | 1-gen-2005 | Costi, Maria Paola; Ferrari, Stefania; Venturelli, A; Calo, S; Tondi, Donatella; Barlocco, D. | |
Improving specificity vs bacterial thymidylate synthases through N-dansyl modulation of didansyltyrosine | 1-gen-2005 | Tondi, Donatella; Venturelli, A.; Ferrari, Stefania; Ghelli, S.; Costi, Maria Paola | |
Alternative strategies in medicinal chemistry to face drug resistance in anticancer therapy. | 1-gen-2006 | Cardinale, Daniela; Ferrari, Stefania; Franchini, Silvia; Corsini, Enrico; Battini, Renata; Costi, Maria Paola | |
Antibacterial agent discovery using thymidylate synthase biolibrary screening | 1-gen-2006 | Costi, Maria Paola; A., Gelain; D., Barlocco; S., Ghelli; Soragni, Fabrizia; F., Reniero; Rossi, Tiziana; Ruberto, Ippazio Antonio; C., Guillou; A., Cavazzuti; Casolari, Chiara; Ferrari, Stefania | |
Novel 3-benzoyl-2-piperazinylquinoxaline derivatives as potential antitumor agents | 1-gen-2006 | S., Piras; M., Loriga; A., Carta; G., Paglietti; Costi, Maria Paola; Ferrari, Stefania | |
Congress on - Medicinal Chemistry in parasitology: new avenues in drug discovery-organised in Modena in 2007. | 1-gen-2007 | Costi, Maria Paola; Ferrari, Stefania; Taramelli, D.; D., Gonzales Pacnowska | |
Interfering with Human Thymidylate Synthase Dimerization against ovarian human carcinoma | 1-gen-2007 | Costi, Maria Paola; Cardinale, Daniela; Guaitoli, Giambattista; Tondi, Donatella; Ferrari, Stefania; Salo Ahen, O; Wade, R. | |
Interfering with Human Thymidylate Synthase Dimerization anti peptide design in the search of anticancer agents against ovarian human carcinoma | 1-gen-2007 | Cardinale, Daniela; Salo Ahen, O; Guaitoli, Giambattista; Tondi, Donatella; Ferrari, Stefania; Wade, R; Costi, Maria Paola | |
Anti-Parasitic drugsDiscovery of potent pteridine reductase inhibitors to guide antiparasite drug development. | 1-gen-2008 | Costi, Maria Paola; Ferrari, Stefania; Cavazzuti, Antonio | |
FRET-based assay for sensing a cancer key protein functional state and inhibition by oligopeptides: Sitespecific Protein Chemical Modifications | 1-gen-2008 | Genovese, Filippo; M., Vargiu; M. A., Ariza Mateos; Guaitoli, Giambattista; Ferrari, Stefania; Ponterini, Glauco; Costi, Maria Paola | |
Discovery of potent pteridine reductase inhibitors to guide antiparasite drug development | 1-gen-2008 | Cavazzuti, Antonio; Paglietti, G.; Hunter, W. N.; Gamarro, F.; Piras, S.; Loriga, M.; Alleca, S.; Corona, P.; Mcluskey, K.; Tulloch, L.; Gibellini, Federica; Ferrari, Stefania; Costi, Maria Paola |
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