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Conformational analysis of phthalein derivatives acting as thymidylate synthase inhibitors by means of 1H NMR and quantum chemical calculations 1-gen-1996 S., Ghelli; Rastelli, Giulio; D., Barlocco; M., Rinaldi; Tondi, Donatella; P., Pecorari; Costi, Maria Paola
Naphthalimido Derivatives as Antifolate Thymidylate Synthase Inhibitors 1-gen-1996 Costi, Mp; Tondi, Donatella; Rinaldi, M; Barlocco, D; Cignarella, G; Santi, Dv; Musiu, C; Pudu, I; Vacca, G; Lacolla, P.
"Structure-Based Discovery & In parallel Optimization of Novel Inhibitors of Thymidylate Synthase" 1-gen-1997 Tondi, D.; Slomczynska, U.; Ghelli, S.; Wattweson, D. M.; Costi, M. P.; Shoichet, B. K.
1H-NMR conformational studies of some phtalein derivatives acting as thymidylate synthase inhibitors 1-gen-1997 S., Ghelli; Costi, Maria Paola; D., Barlocco; M., Rinaldi; Tondi, Donatella; P., Pecorari; Rastelli, Giulio
Mono- and Disubstituted-3,8-diazabicyclo[3.2.1]octane Derivatives as Analgesics Structurally Related to Epibatidine: Synthesis, Activity, and Modeling. 1-gen-1998 Barlocco, Daniela; Cignarella, Giorgio; Tondi, Donatella; Vianello, Paola; Villa, Stefania; Bartolini, Alessandro; Ghelardini, Carla; Galeotti, Nicoletta; ANDERSON DAVID, J. KUNTZWEILER THERESA A.; Colombo, Diego; Toma, Lucio
3-Aminophenylboronic acid derivative inhibitors of beta-lactamases, their preparation, and their therapeutic use. 16-dic-1998 SHOICHET BRIAN, K.; Costi, Maria Paola; Tondi, Donatella
Structure-based discovery and combinatorial optimization of novel competitive inhibitors of thymidylate synthase 1-gen-1999 Sholchet, Bk; Tondi, Donatella; Slomczynska, U.
Thymidylate Synthase as a potential new target in drug resistance antimicrobial therapy. 1-gen-1999 Costi, Maria Paola; A., Gelain; I., Cardilicchio; Soragni, Fabrizia; Rinaldi, Marcella; Pecorari, Piergiorgio; Tondi, Donatella; D. V., Santi
Structure based design and combinatorial optimization of novel Thymidylate synthase inhibitors. Meeting Abstract : 217th ACS National Meeting, Chicago March 1999 1-gen-1999 Tondi, Donatella; Slomcynska, U.; Ghelli, Stefano; Watterson, D. M.; Costi, Maria Paola; Shoichet, B. K.
Structure-based design of inhibitors specific for bacterial thymidylate synthase 1-gen-1999 Tj, Stout; Tondi, Donatella; Rinaldi, Marcella; Barlocco, Daniela; Pecorari, Piergiorgio; Dv, Santi; I., Kuntz; Rm, Stroud; Costi, Maria Paola; Bk, Shoichet
Separation, structural determination and biological evaluation of the thymidylate synthase inhibitor 3,3-di(4'-hydroxyphenyl)-6(7)-chloro-1-oxo-1H,3H-naphtho[1,8-cd]pyran 1-gen-1999 Costi, Maria Paola; Tondi, Donatella; Pecorari, Piergiorgio; Rinaldi, M; Celentano, G; Ghelli, Stefano; Antolini, L; Barlocco, Daniela
Phthalein derivatives as a new tool for selectivity in thymidylate synthase inhibition 1-gen-1999 Costi, Maria Paola; Rinaldi, Marcella; Tondi, Donatella; Pecorari, Piergiorgio; Barlocco, Daniela; Ghelli, Stefano; Rm, Stroud; Dv, Santi; Tj, Stout; C., Musiu; Em, Marangiu; A., Pani; D., Congiu; Ga, Loi; P., La Colla
Structure-based discovery and in-parallel optimization of novel competitive inhibitors of thymidylate synthase 1-gen-1999 Tondi, Donatella; U., Slomczynska; Costi, Maria Paola; Dm, Watterson; Ghelli, Stefano; Bk, Shoichet
Sulfonamide Boronic Acid Inhibitors of AmpC b-lactamase to Reverse Bacterial Resistance to b-lactam Antibiotics. 16-dic-1999 Shoichet, B. K.; Tondi, Donatella; Costi, Maria Paola; M., P.
Amide Boronic Acid Inhibitors of AmpC b-lactamase to Reverse Bacterial Resistance to b-lactam Antibiotics. 16-dic-1999 Shoichet, B. K.; Tondi, Donatella; Costi, Maria Paola; M., P.
Phenylboronic acid derivative inhibitors of β-lactamases, their preparation, pharmaceutical compositions, and therapeutic use 16-dic-1999 Shoichet, B K; Costi, Maria Paola; Tondi, Donatella
Structure-Based Design and In Parallel Synthesis of Boronic Acid Inhibitors of AmpC 61538;-Lactamase 1-gen-2000 Tondi, Donatella; Powers, R.; Caselli, Emilia; Costi, Maria Paola; Shoichet, B. K.
Studi termodinamici e strutturali dell’interazione tra derivati densilici e Timidilato Sintasi Batteriche 1-gen-2000 Tondi, Donatella; Venturelli, Alberto; Skinner, M. A.; Brown, K.; Costi, Maria Paola
Phenylboronic acid derivative inhibitors of ?-lactamases, their preparation, pharmaceutical compositions, and therapeutic use. 1-gen-2000 Shoichet, B. K.; Costi, Maria Paola; Tondi, Donatella
3-Aminophenylboronic acid derivative inhibitors of β-lactamases, their preparation, and their therapeutic use 22-giu-2000 Shoichet, B. K.; Costi, Maria Paola; Tondi, Donatella
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