Sfoglia per Autore
Structure-Activity Relationship in Dihydropteroate Synthase Inhibition by Sulfanilamides. Comparison with the Antibacterial Activity.
1981 DE BENEDETTI, Pier Giuseppe; Rastelli, Augusto; Frassineti, Chiara; Cennamo, Carlo
A Theoretical Study of the Structure-Activity Relationship in Diarylsulphones. Comparison with Sulfa Drugs.
1983 DE BENEDETTI, Pier Giuseppe; Frassineti, Chiara
Experimental and Theoretical Study of Electronic Substituent Effects in 4-Aminoaryl (4-Substituted Aryl) Sulphones.
1985 DE BENEDETTI, Pier Giuseppe; Folli, Ugo; Iarossi, Dario; Frassineti, Chiara
A Quantum Chemical QSAR Study of Carbonic Anhydrase Inhibition by Sulfonamides.
1985 DE BENEDETTI, Pier Giuseppe; Menziani, Maria Cristina; Frassineti, Chiara
A Quantum Chemical QSAR Analysis of Carbonic Anhydrase Inhibition by Heterocyclic Sulfonamides.
1987 DE BENEDETTI, Pier Giuseppe; Menziani, Maria Cristina; Cocchi, Marina; Frassineti, Chiara
Quantitative Structure-Activity Analysis in Dihydropteroate Synthase Inhibition by Sulphones. Comparison with Sulfanilamides.
1987 DE BENEDETTI, Pier Giuseppe; Iarossi, Dario; Menziani, Maria Cristina; V., Caiolfa; Frassineti, Chiara; Cennamo, Carlo
Multinuclear NMR and Vibrational Spectroscopy Studies of the Substituent Effects in Benzensulfonamide Inhibitors of the Enzyme Carbonic Anhydrase.
1988 DE BENEDETTI, Pier Giuseppe; Iarossi, Dario; Menziani, Maria Cristina; Frassineti, Chiara; Benedetti, Adriano
A Theoretical Study of Conformation-Electronic Structure Relationships in Benzensulfonamide Inhibitors of Carbonic Anhydrase Enzyme.
1989 DE BENEDETTI, Pier Giuseppe; Menziani, Maria Cristina; Cocchi, Marina; Frassineti, Chiara
Comparative QSAR Analysis in Dihydropteroate Synthase Inhibition by Sulphones. Design of Some New Derivatives with Improved Petency.
1989 DE BENEDETTI, Pier Giuseppe; Iarossi, Dario; Frassineti, Chiara; Menziani, Maria Cristina; Cocchi, Marina; Cennamo, Carlo
Quantitative Structure-Activity Relationships in Dihydropteroate Synthase Inhibition by Multisubstituted Sulfones. Design and Synthesis of Some New Derivatives with Improved Potency.
1989 DE BENEDETTI, Pier Giuseppe; Iarossi, Dario; Folli, Ugo; Frassineti, Chiara; Menziani, Maria Cristina; Cennamo, Carlo
The binding of benzenesulfonamides to carbonic anhydrase enzyme. A molecular mechanics study and quantitative structure-activity relationships
1989 Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe; F., Gago; W. G., Richards
QSAR analysis in 2,4-diamino-6,7-dimethoxy quinoline derivatives - α1-adrenoceptor antagonists - using the partial least squares (PLS) method and theoretical molecular descriptors
1990 Cocchi, Marina; Menziani, Maria Cristina; Rastelli, Giulio; DE BENEDETTI, Pier Giuseppe
Direct and Indirect Theoretical QSAR Modelling in Sulfonamide Carbonic Anhydrase Inhibitors
1991 Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe
QSAR Analysis Using Theoretical Molecular Descriptors in 2,4-Diamino-6,7-Dimethoxy Quinazoline 1-Adrenoceptor Antagonists.
1991 DE BENEDETTI, Pier Giuseppe; Menziani, Maria Cristina; Rastelli, Giulio; Cocchi, Marina
MOLECULAR-ORBITAL STUDY OF THE NITROGEN BASICITY OF PRAZOSIN ANALOGS IN RELATION TO THEIR ALPHA-1-ADRENOCEPTOR BINDING-AFFINITY
1991 DE BENEDETTI, Pier Giuseppe; Menziani, Maria Cristina; Rastelli, Giulio; Cocchi, Marina
Theoretical conformational analysis, electronic structure and molecular modelling studies in dihydropteroate synthase in hibition by multisubstituted s
1991 Sokolov, Yu. A.; Menziani, M. C.; Cocchi, M.; De Benedetti, P. G.
Correlation and Multivariate Analyses of the Spectroscopic Data in 4'-Substituted 4-Nitro-difhenylsulfones
1991 Cocchi, Marina; Iarossi, Dario; Frassineti, Chiara; Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe
Conformational analysis, molecular modeling and quantitative structure-activity relationships studies of 2,4-diamino-6,7-dimethoxy-2-substituted quinazoline α1-adrenergic antagonists
1991 Rastelli, Giulio; Fanelli, Francesca; Menziani, Maria Cristina; Cocchi, Marina; DE BENEDETTI, Pier Giuseppe
A THEORETICAL-STUDY OF THE STRUCTURE OF BIG ENDOTHELIN
1991 Menziani, Maria Cristina; Cocchi, Marina; DE BENEDETTI, Pier Giuseppe; Gilbert, Rg; Richards, Wg; Zamai, M; Caiolfa, Vr
Molecular mechanics and quantum chemical qsar analysis in carbonic anhydrase-heterocyclic sulfonamide interactions
1992 Menziani, Maria Cristina; DE BENEDETTI, Pier Giuseppe
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