Sfoglia per Autore
MOLECULAR PROPERTIES OF THE ADRENERGIC a-RECEPTORIII - Origin of topographicol duqlism in the reaction of a receptor thiolwith symmetrical and unsymmetrical polyamine disulfides.
1978 C., Melchiorre; D., Giardina; Brasili, Livio; B., Belleau
THE CATECHOLAMINE Alpha--RECEPTOR AS A POLYANIONIC CYSTEINE PROTEIN.SELECTIVE COVALENT OCCUPANCY BY POLYAMINEDISULFIDES
1979 Carlo, Melchiorre; MAN SEN, Yong; Bruno, Benfey; Brasili, Livio; Gordon, Bolger; Bernard, Belleau
MOLECULAR REQUIREMENTS OF THE ACTIVE SITESOF THE CHOLINERGIC RECEPTORSXII (*) - 3-Methyl-2-oxo-L-dimethylaminomethylcyclopentane methiodideas a new selective agonist for the nicotinic receptorM. GIANNELLA, P. ANGELI, C. MELCHIORRE, L. BRASILI
1980 M., Giannella; P., Angeli; C., Melchiorre; Brasili, Livio
MOLECULAR REQUIREMENTS OF THE ACTIVE SITESOF THE CHOLINERGIC RECEPTORSXI - Synthesis and biological evaluation of isomuscarine and itsisomers
1980 M., Pigini; R., Ballini; F., Gualtieri; Brasili, Livio
Potentiation and inhibition ofnicotinic effects on striated muscle by the tetramlne disulfide benextramineB. G. Benfey, L. Brasili, C. Melchiorre, B. Belleau
1980 B. G., Benfey; Brasili, Livio; C., Melchiorre; B., Belleau
Reactivation by cysteamine of vascular alpha-adrenoceptors blocked by the tetraminedisulfide benextramine and interaction of benextramine with phenoxybenzamine
1980 Brasili, Livio; C., Melchiorre; B., Belleau; B. G., Benfey
Irreversible alfa-adrenoceptor blocking effects and irreversible muscarinic blocking and nicotinic blocking effect of tetramine disulfides on heart B. G. Benfey, B. Belleau, L. Brasili, M. Giannella, C. Melchiorre
1980 B. G., Benfey; B., Belleau; Brasili, Livio; M., Giannella; C., Melchiorre
MOLECULAR REQUIREMENTS OF THE ACTIVE SITESOF THE CHOLINERGIC RECEPTORSXVI (x) - Synthesis qnd cholinergic activity ol 2- or 5-alkyl or 5-phenyl--4-methyl-3-oxo-1 -dimethylaminomethylcy clopentane methiodide.
1981 M., Pigini; Brasili, Livio
Structural requirements for adrenergic alpha-receptorcovalent occupancy by chiral tetramine disulfides
1981 Brasili, Livio; Mario, Giannella; Carlo, Melchiorre; Bernard, Belleau; Bruno G., Benfey
Molecular properties of the adrenergic alpha-receptor6. - Optimum carbon chain-length between the inner nitrogenand the sulfur of tetramine disulfides
1981 Dario, Giardinà; Brasili, Livio; Carlo, Melchiorre; Bernard, Belleau; Bruno G., Benfey
Molecular requirements of the active sites of thecholinergic receptors XVII. 1,3-oxathiolane nucleus as a carrier of the active moeties
1981 Maria, Pigini; Brasili, Livio; Mario, Giannella; Fulvio, Gualtieri
Molecular properties of the adrenergic alpha-receptors.4.Topographical and structural differences betweentissue-specific binding sites as revealedby benextramine and analogues.
1981 Carlo, Melchiorre; Mario, Giannella; Brasili, Livio; Bruno G., Benfey; Bernard, Belleau
Molecular Requirements of the Active Site of CholinergicReceptors XV: Synthesis and Biological Activity of2, 3 -Dehydrodeoxamuscarone and 2,3 -Dehydrodeoxamuscarines
1981 Piero, Angeli; Brasili, Livio; Dario, Giardinà; Carlo, Melchiorre
MOLECULAR REQUIREMENTS OF THE ACTIVE SITESOF THE CHOLINERGIC RECEPTORS
1982 F., Gualtieri; Brasili, Livio; M., Giannella; M., Pigini
MOLECULAR. REQUIR.EMENTS OF THE ACTIVE SITESOF THE CHOLINERGIC RECEPTORS
1982 Brasili, Livio; M., Leonelli; M., Giannella
Structural requirements for competitive s-adrenoceptor occupancy bycyclic and opened analogues of WB 4I0I
1982 Carlo, Melchiorre; Dario, Giardina'; Patrizia, Gallucci; Brasili, Livio
SYNTHESIS AND PHARMACOLOGICAL EVALUATIONOF PROPRANOLOL-CYCLIC ANALOGUES
1983 E., Castagnino; S., Corsano; G., Strappaghetti; Brasili, Livio; P., Gallucci
SYNTHESIS AND PHARMACOLOGICAL EVALUATIONOF SOME V/84101 ANALOGUES BEARING ANAPHTODIOXANIC NUCLEUS
1984 E., Castagnino; G., Strappaghetti; S., Corsano; P., Gallucci; Brasili, Livio; D., Giardina
Correlation hetween adrenergic alpha-receptorantagonists of tetramine disulfidesand benzodioxanes classes
1984 Carlo, Melchiorre; Ugo, Gulini; Dario, Giardina'; Patrizia, Gallucci; Brasili, Livio
2-{[(2-(2,6-Dimethoxyphenoxy)ethyl]}-1,4-benzoxathiano:A New Antagonist With High Potency and Selectivity Toward alpha1-Adrenoreceptors.
1984 Melchiorre, C.; Brasili, Livio; Giardin, D.; Pigini, M.; Strappaghetti, G.
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