Sfoglia per Autore
Rational design of dual inhibitors of Hsp90 and B-Raf as a novel pharmacological approach against melanomas
2015 Pinzi, Luca; Rastelli, Giulio
Rational design of dual inhibitors of Hsp90 and Braf as a novel pharmacological approach against melanomas
2015 Pinzi, Luca; Rastelli, Giulio
Computational polypharmacology comes of age
2015 Rastelli, Giulio; Pinzi, Luca
Polypharmacology predictions in the Protein Data Bank
2016 Pinzi, Luca; Rastelli, Giulio
Predicting drug polypharmacology using structural databases
2016 Pinzi, Luca; Rastelli, Giulio
An unexpected reversal in the pharmacological stereoselectivity of benzothiadiazine AMPA positive allosteric modulators
2016 Battisti, UMBERTO MARIA; Citti, Cinzia; Rastelli, Giulio; Pinzi, Luca; Puja, Giulia; Ravazzini, Federica; Ciccarella, Giuseppe; Braghiroli, Daniela; Cannazza, Giuseppe
Heat shock protein 90 and serine/threonine kinase B-Raf inhibitors have overlapping chemical space
2017 Anighoro, A.; Pinzi, Luca; Marverti, Gaetano; Bajorath, J; Rastelli, Giulio
On the integration of in silico drug design methods for drug repurposing
2017 MARCH VILA, Eric; Pinzi, Luca; Sturm, Noã; Tinivella, Annachiara; Engkvist, Ola; Chen, Hongming; Rastelli, Giulio
Identification of 4-aryl-1H-pyrrole[2,3-b]pyridine derivatives for the development of new B-Raf inhibitors
2018 Pinzi, Luca; Anighoro, Andrew; Bajorath, Jürgen; Rastelli, Giulio
Identification of small-molecule EGFR allosteric inhibitors by high-Throughput docking
2018 Caporuscio, Fabiana; Tinivella, Annachiara; Restelli, Valentina; Semrau, Marta S; Pinzi, Luca; Storici, Paola; Broggini, Massimo; Rastelli, Giulio
Structure–Activity Relationships of Hexahydrocyclopenta[c]quinoline Derivatives as Allosteric Inhibitors of CDK2 and EGFR
2018 Carlino, Luca; Christodoulou, Michael S.; Restelli, Valentina; Caporuscio, Fabiana; Foschi, FRANCESCA MADDALENA; Semrau, MARTA STEFANIA; Costanzi, Elisa; Tinivella, Annachiara; Pinzi, Luca; Lo Presti, Leonardo; Battistutta, Roberto; Storici, Paola; Broggini, Massimo; Passarella, Daniele; Rastelli, Giulio
Selection of protein conformations for structure-based polypharmacology studies
2018 Pinzi, Luca; Caporuscio, Fabiana; Rastelli, Giulio
Unveiling target associations for polypharmacology from analysis of crystallographic ligands in the Protein Data Bank
2019 Pinzi, Luca; Rastelli, Giulio
Evaluation of Amides, Carbamates, Sulfonamides, and Ureas of 4-Prop-2-ynylidenecycloalkylamine as Potent, Selective, and Bioavailable Negative Allosteric Modulators of Metabotropic Glutamate Receptor 5
2019 Graziani, Davide; Caligari, Silvia; Callegari, Elisa; De Toma, Carlo; Longhi, Matteo; Frigerio, Fabio; Dilernia, Roberto; Menegon, Sergio; Pinzi, Luca; Pirona, Lorenza; Tazzari, Valerio; Valsecchi, Anna Elisa; Vistoli, Giulio; Rastelli, Giulio; Ruga Riva, Carlo
In silico repositioning of cannabigerol as a novel inhibitor of the enoyl acyl carrier protein (ACP) reductase (INHA)
2019 Pinzi, L.; Lherbet, C.; Baltas, M.; Pellati, F.; Rastelli, G.
Refinement and rescoring of virtual screening results
2019 Rastelli, G.; Pinzi, L.
2-Phenyloxazole-4-carboxamide as a Scaffold for Selective Inhibition of Human Monoamine Oxidase B
2019 Di Paolo, M. L.; Christodoulou, M. S.; Calogero, A. M.; Pinzi, L.; Rastelli, G.; Passarella, D.; Cappelletti, G.; Dalla Via, L.
Molecular docking: Shifting paradigms in drug discovery
2019 Pinzi, L.; Rastelli, G.
Virtual screening for dual Hsp90/B-Raf inhibitors
2019 Anighoro, A.; Pinzi, L.; Rastelli, G.; Bajorath, J.
Repositioning natural products in drug discovery
2020 Rastelli, G.; Pellati, F.; Pinzi, L.; Gamberini, M. C.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Rational design of dual inhibitors of Hsp90 and B-Raf as a novel pharmacological approach against melanomas | 1-gen-2015 | Pinzi, Luca; Rastelli, Giulio | |
Rational design of dual inhibitors of Hsp90 and Braf as a novel pharmacological approach against melanomas | 1-gen-2015 | Pinzi, Luca; Rastelli, Giulio | |
Computational polypharmacology comes of age | 1-gen-2015 | Rastelli, Giulio; Pinzi, Luca | |
Polypharmacology predictions in the Protein Data Bank | 1-gen-2016 | Pinzi, Luca; Rastelli, Giulio | |
Predicting drug polypharmacology using structural databases | 1-gen-2016 | Pinzi, Luca; Rastelli, Giulio | |
An unexpected reversal in the pharmacological stereoselectivity of benzothiadiazine AMPA positive allosteric modulators | 1-gen-2016 | Battisti, UMBERTO MARIA; Citti, Cinzia; Rastelli, Giulio; Pinzi, Luca; Puja, Giulia; Ravazzini, Federica; Ciccarella, Giuseppe; Braghiroli, Daniela; Cannazza, Giuseppe | |
Heat shock protein 90 and serine/threonine kinase B-Raf inhibitors have overlapping chemical space | 1-gen-2017 | Anighoro, A.; Pinzi, Luca; Marverti, Gaetano; Bajorath, J; Rastelli, Giulio | |
On the integration of in silico drug design methods for drug repurposing | 1-gen-2017 | MARCH VILA, Eric; Pinzi, Luca; Sturm, Noã; Tinivella, Annachiara; Engkvist, Ola; Chen, Hongming; Rastelli, Giulio | |
Identification of 4-aryl-1H-pyrrole[2,3-b]pyridine derivatives for the development of new B-Raf inhibitors | 1-gen-2018 | Pinzi, Luca; Anighoro, Andrew; Bajorath, Jürgen; Rastelli, Giulio | |
Identification of small-molecule EGFR allosteric inhibitors by high-Throughput docking | 1-gen-2018 | Caporuscio, Fabiana; Tinivella, Annachiara; Restelli, Valentina; Semrau, Marta S; Pinzi, Luca; Storici, Paola; Broggini, Massimo; Rastelli, Giulio | |
Structure–Activity Relationships of Hexahydrocyclopenta[c]quinoline Derivatives as Allosteric Inhibitors of CDK2 and EGFR | 1-gen-2018 | Carlino, Luca; Christodoulou, Michael S.; Restelli, Valentina; Caporuscio, Fabiana; Foschi, FRANCESCA MADDALENA; Semrau, MARTA STEFANIA; Costanzi, Elisa; Tinivella, Annachiara; Pinzi, Luca; Lo Presti, Leonardo; Battistutta, Roberto; Storici, Paola; Broggini, Massimo; Passarella, Daniele; Rastelli, Giulio | |
Selection of protein conformations for structure-based polypharmacology studies | 1-gen-2018 | Pinzi, Luca; Caporuscio, Fabiana; Rastelli, Giulio | |
Unveiling target associations for polypharmacology from analysis of crystallographic ligands in the Protein Data Bank | 1-gen-2019 | Pinzi, Luca; Rastelli, Giulio | |
Evaluation of Amides, Carbamates, Sulfonamides, and Ureas of 4-Prop-2-ynylidenecycloalkylamine as Potent, Selective, and Bioavailable Negative Allosteric Modulators of Metabotropic Glutamate Receptor 5 | 1-gen-2019 | Graziani, Davide; Caligari, Silvia; Callegari, Elisa; De Toma, Carlo; Longhi, Matteo; Frigerio, Fabio; Dilernia, Roberto; Menegon, Sergio; Pinzi, Luca; Pirona, Lorenza; Tazzari, Valerio; Valsecchi, Anna Elisa; Vistoli, Giulio; Rastelli, Giulio; Ruga Riva, Carlo | |
In silico repositioning of cannabigerol as a novel inhibitor of the enoyl acyl carrier protein (ACP) reductase (INHA) | 1-gen-2019 | Pinzi, L.; Lherbet, C.; Baltas, M.; Pellati, F.; Rastelli, G. | |
Refinement and rescoring of virtual screening results | 1-gen-2019 | Rastelli, G.; Pinzi, L. | |
2-Phenyloxazole-4-carboxamide as a Scaffold for Selective Inhibition of Human Monoamine Oxidase B | 1-gen-2019 | Di Paolo, M. L.; Christodoulou, M. S.; Calogero, A. M.; Pinzi, L.; Rastelli, G.; Passarella, D.; Cappelletti, G.; Dalla Via, L. | |
Molecular docking: Shifting paradigms in drug discovery | 1-gen-2019 | Pinzi, L.; Rastelli, G. | |
Virtual screening for dual Hsp90/B-Raf inhibitors | 1-gen-2019 | Anighoro, A.; Pinzi, L.; Rastelli, G.; Bajorath, J. | |
Repositioning natural products in drug discovery | 1-gen-2020 | Rastelli, G.; Pellati, F.; Pinzi, L.; Gamberini, M. C. |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile