Sfoglia per Autore
An Improved Synthesis of CENTA, a Chromogenic Substrate for β-Lactamases
2016 QUOTADAMO, ANTONIO; LINCIANO, PASQUALE; DAVOLI, Paolo; TONDI, Donatella; COSTI, Maria Paola; VENTURELLI, Alberto
A multidisciplinary approach to the design of novel inhibitors for KPC-2
2017 Celenza, Giuseppe; Bellio, Pierangelo; Linciano, Pasquale; Perilli, Mariagrazia; Cendron, Laura; Tondi, Donatella
Exploiting the 2-Amino-1,3,4-thiadiazole Scaffold To InhibitTrypanosoma bruceiPteridine Reductase in Support of Early-Stage Drug Discovery
2017 Linciano, Pasquale; Dawson, Alice; Pöhner, Ina; Costa, David M; Sá, Monica S; Cordeiro-da-Silva, Anabela; Luciani, Rosaria; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Gribbon, Philip; Reinshagen, Jeanette; Wolf, Markus; Behrens, Birte; Hannaert, Véronique; Michels, Paul A M; Nerini, Erika; Pozzi, Cecilia; di Pisa, Flavio; Landi, Giacomo; Santarem, Nuno; Ferrari, Stefania; Saxena, Puneet; Lazzari, Sandra; Cannazza, Giuseppe; Freitas-Junior, Lucio H; Moraes, Carolina B; Pascoalino, Bruno S; Alcântara, Laura M; Bertolacini, Claudia P; Fontana, Vanessa; Wittig, Ulrike; Müller, Wolfgang; Wade, Rebecca C; Hunter, William N; Mangani, Stefano; Costantino, Luca; Costi, Maria P
Methoxylated 2'-hydroxychalcones as antiparasitic hit compounds
2017 Borsari, Chiara; Santarem, Nuno; Torrado, Juan; Olías, Ana Isabel; Corral, María Jesús; Baptista, Catarina; Gul, Sheraz; Wolf, Markus; Kuzikov, Maria; Ellinger, Bernhard; Witt, Gesa; Gribbon, Philip; Reinshagen, Jeanette; Linciano, Pasquale; Tait, Annalisa; Costantino, Luca; Freitas-Junior, Lucio H.; Moraes, Carolina B.; Bruno dos Santos, Pascoalino; Alcântara, Laura Maria; Franco, Caio Haddad; Bertolacini, Claudia Danielli; Fontana, Vanessa; Tejera Nevado, Paloma; Clos, Joachim; Alunda, José María; Cordeiro-da-Silva, Anabela; Ferrari, Stefania; Costi, Maria Paola
New weapons against antimicrobial resistance: Targeting SOS response to recover b actericidal activity of antibiotics
2018 Maso, Lorenzo; Bellio, Pierangelo; Linciano, Pasquale; D’Acunto, Maria; Celenza, Giuseppe; Tondi, Donatella; Cendron, Laura
In silico identification and experimental validation of hits active against KPC-2 β-lactamase
2018 Klein, Raphael; Linciano, Pasquale; Celenza, Giuseppe; Bellio, Pierangelo; Papaioannou, Sofia; Blazquez, Jesus; Cendron, Laura; Brenk, Ruth; Tondi, Donatella
Phenyl boronic acids development led to validated leads active in clinical strains overexpressing KPC-2: a step against bacterial resistance.
2018 Celenza, Giuseppe; Vicario, Mattia; Bellio, Pierangelo; Linciano, Pasquale; Perilli, Mariagrazia; Oliver, Antonio; Blazquez, Jesús; Cendron, Laura; Tondi, Donatella
Aryl thiosemicarbazones for the treatment of trypanosomatidic infections
2018 Linciano, Pasquale; Moraes, Carolina B.; Alcantara, Laura M.; Franco, Caio H.; Pascoalino, Bruno; Freitas-Junior, Lucio H.; Macedo, Sara; Santarem, Nuno; Cordeiro-da-Silva, Anabela; Gul, Sheraz; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Ferrari, Stefania; Luciani, Rosaria; Quotadamo, Antonio; Costantino, Luca; Costi, Maria Paola
Scouting Sigma Receptor Ligands As New Tools For The Treatment Of Neurodegenerative Diseases And Cancer
2019 Sorbi, C.; Linciano, P.; Tait, A.; Atene, C. G.; Guglielmo, L.; Di Rocco, G.; Ronsisvalle, S.; Denora, N.; Imbriano, C.; Rigillo, G.; Fossa, P.; Cichero, E.; Benassi, L.; Vaschieri, C.; Marocchi, F.; Lanfrancone, M. L.; Brasili, L.; Franchini, S.
IDENTIFICATION OF POTENT 1,3-DIOXOLANE-BASED 5-HT1A RECEPTOR AGONISTS FOR THE TREATMENTS OF CNS DISORDERS AND PAIN
2019 Linciano, Pasquale; Sorbi, Claudia; Franchini, Silvia; Tait, Annalisa; Bardoni, Rita; Ronsisvalle, Simone; Denora, Nunzio; Lesniak, Anna; Bujalska-Zadrożny, Magdalena; Pawłowska, Agata; Chichero, Elena; Fossa, Paola; Brasili, Livio
Hits and Lead Discovery in the Identification of New Drugs against the Trypanosomatidic Infections
2019 Calogeropoulou, Theodora; Magoulas, George E.; Pöhner, Ina; Wade, Rebecca C.; Panecka-Hofman, Joanna; Linciano, Pasquale; Ferrari, Stefania; Costi, Maria Paola; Santarem, Nuno; Dolores Jiménez-Antón, Ma; Isabel Olías-Molero, Ana; Cordeiro da Silva and José María Alunda, Anabela
Development of therapeutic agents blocking SOS activation.
2019 Maso, L.; Bellio, P.; Linciano, P.; D' Acunto, M.; Celenza, G.; Tondi, Donatella; Cendron, L.
Effect of the rigidification of propranolol, a mixed β-adrenoceptor and 5-HT1AR antagonist
2019 Franchini, S.; Sorbi, C.; Linciano, P.; Brasili, L.; Tait, A.
Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform
2019 Moraes, Carolina B.; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Calogeropoulou, Theodora; Prousis, Kyriakos C.; Mangani, Stefano; Di Pisa, Flavio; Landi, Giacomo; Iacono, Lucia Dello; Pozzi, Cecilia; Freitas-Junior, Lucio H.; dos Santos Pascoalino, Bruno; Bertolacini, Claudia P.; Behrens, Birte; Keminer, Oliver; Leu, Jennifer; Wolf, Markus; Reinshagen, Jeanette; Cordeiro-da-Silva, Anabela; Santarem, Nuno; Venturelli, Alberto; Wrigley, Stephen; Karunakaran, Deepa; Kebede, Bethlehem; Pöhner, Ina; Müller, Wolfgang; Panecka-Hofman, Joanna; Wade, Rebecca C.; Fenske, Martina; Clos, Joachim; Alunda, José María; Corral, María Jesús; Uliassi, Elisa; Bolognesi, Maria Laura; Linciano, Pasquale; Quotadamo, Antonio; Ferrari, Stefania; Santucci, Matteo; Borsari, Chiara; Costi, Maria Paola; Gul, Sheraz
A novel phytocannabinoid isolated from Cannabis sativa L. with an in vivo cannabimimetic activity higher than Δ9-tetrahydrocannabinol: Δ9-Tetrahydrocannabiphorol
2019 Citti, C.; Linciano, P.; Russo, F.; Luongo, L.; Iannotta, M.; Maione, S.; Lagana, A.; Capriotti, A. L.; Forni, F.; Vandelli, M. A.; Gigli, G.; Cannazza, G.
Analysis of impurities of cannabidiol from hemp. Isolation, characterization and synthesis of cannabidibutol, the novel cannabidiol butyl analog
2019 Citti, C.; Linciano, P.; Forni, F.; Vandelli, M. A.; Gigli, G.; Lagana, A.; Cannazza, G.
Cyclic Peptides Acting as Allosteric Inhibitors of Human Thymidylate Synthase and Cancer Cell Growth
2019 Pacifico, Salvatore; Santucci, Matteo; Luciani, Rosaria; Saxena, Puneet; Linciano, Pasquale; Ponterini, Glauco; Lauriola, Angela; D'Arca, Domenico; Marverti, Gaetano; Guerrini, Remo; Costi, Maria Paola
First virtual screening and experimental validation of inhibitors targeting GES-5 carbapenemase
2019 Spyrakis, Francesca; Bellio, Pierangelo; Quotadamo, Antonio; Linciano, Pasquale; Benedetti, Paolo; D’Arrigo, Giulia; Baroni, Massimo; Cendron, Laura; Celenza, Giuseppe; Tondi, Donatella
Excited-state intramolecular proton transfer in a bioactive flavonoid provides fluorescence observables for recognizing its engagement with target proteins
2019 Vanossi, D.; Caselli, M.; Pavesi, G.; Borsari, C.; Linciano, P.; Costi, M. P.; Ponterini, G.
Optimization of N-alkylation in the Synthesis of Methotrexate and Pteridine-based Derivatives Under Microwave-Irradiation
2019 Quotadamo, A.; Linciano, P.; Costi, M. P.; Venturelli, A.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
An Improved Synthesis of CENTA, a Chromogenic Substrate for β-Lactamases | 1-gen-2016 | QUOTADAMO, ANTONIO; LINCIANO, PASQUALE; DAVOLI, Paolo; TONDI, Donatella; COSTI, Maria Paola; VENTURELLI, Alberto | |
A multidisciplinary approach to the design of novel inhibitors for KPC-2 | 1-gen-2017 | Celenza, Giuseppe; Bellio, Pierangelo; Linciano, Pasquale; Perilli, Mariagrazia; Cendron, Laura; Tondi, Donatella | |
Exploiting the 2-Amino-1,3,4-thiadiazole Scaffold To InhibitTrypanosoma bruceiPteridine Reductase in Support of Early-Stage Drug Discovery | 1-gen-2017 | Linciano, Pasquale; Dawson, Alice; Pöhner, Ina; Costa, David M; Sá, Monica S; Cordeiro-da-Silva, Anabela; Luciani, Rosaria; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Gribbon, Philip; Reinshagen, Jeanette; Wolf, Markus; Behrens, Birte; Hannaert, Véronique; Michels, Paul A M; Nerini, Erika; Pozzi, Cecilia; di Pisa, Flavio; Landi, Giacomo; Santarem, Nuno; Ferrari, Stefania; Saxena, Puneet; Lazzari, Sandra; Cannazza, Giuseppe; Freitas-Junior, Lucio H; Moraes, Carolina B; Pascoalino, Bruno S; Alcântara, Laura M; Bertolacini, Claudia P; Fontana, Vanessa; Wittig, Ulrike; Müller, Wolfgang; Wade, Rebecca C; Hunter, William N; Mangani, Stefano; Costantino, Luca; Costi, Maria P | |
Methoxylated 2'-hydroxychalcones as antiparasitic hit compounds | 1-gen-2017 | Borsari, Chiara; Santarem, Nuno; Torrado, Juan; Olías, Ana Isabel; Corral, María Jesús; Baptista, Catarina; Gul, Sheraz; Wolf, Markus; Kuzikov, Maria; Ellinger, Bernhard; Witt, Gesa; Gribbon, Philip; Reinshagen, Jeanette; Linciano, Pasquale; Tait, Annalisa; Costantino, Luca; Freitas-Junior, Lucio H.; Moraes, Carolina B.; Bruno dos Santos, Pascoalino; Alcântara, Laura Maria; Franco, Caio Haddad; Bertolacini, Claudia Danielli; Fontana, Vanessa; Tejera Nevado, Paloma; Clos, Joachim; Alunda, José María; Cordeiro-da-Silva, Anabela; Ferrari, Stefania; Costi, Maria Paola | |
New weapons against antimicrobial resistance: Targeting SOS response to recover b actericidal activity of antibiotics | 1-gen-2018 | Maso, Lorenzo; Bellio, Pierangelo; Linciano, Pasquale; D’Acunto, Maria; Celenza, Giuseppe; Tondi, Donatella; Cendron, Laura | |
In silico identification and experimental validation of hits active against KPC-2 β-lactamase | 1-gen-2018 | Klein, Raphael; Linciano, Pasquale; Celenza, Giuseppe; Bellio, Pierangelo; Papaioannou, Sofia; Blazquez, Jesus; Cendron, Laura; Brenk, Ruth; Tondi, Donatella | |
Phenyl boronic acids development led to validated leads active in clinical strains overexpressing KPC-2: a step against bacterial resistance. | 1-gen-2018 | Celenza, Giuseppe; Vicario, Mattia; Bellio, Pierangelo; Linciano, Pasquale; Perilli, Mariagrazia; Oliver, Antonio; Blazquez, Jesús; Cendron, Laura; Tondi, Donatella | |
Aryl thiosemicarbazones for the treatment of trypanosomatidic infections | 1-gen-2018 | Linciano, Pasquale; Moraes, Carolina B.; Alcantara, Laura M.; Franco, Caio H.; Pascoalino, Bruno; Freitas-Junior, Lucio H.; Macedo, Sara; Santarem, Nuno; Cordeiro-da-Silva, Anabela; Gul, Sheraz; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Ferrari, Stefania; Luciani, Rosaria; Quotadamo, Antonio; Costantino, Luca; Costi, Maria Paola | |
Scouting Sigma Receptor Ligands As New Tools For The Treatment Of Neurodegenerative Diseases And Cancer | 1-gen-2019 | Sorbi, C.; Linciano, P.; Tait, A.; Atene, C. G.; Guglielmo, L.; Di Rocco, G.; Ronsisvalle, S.; Denora, N.; Imbriano, C.; Rigillo, G.; Fossa, P.; Cichero, E.; Benassi, L.; Vaschieri, C.; Marocchi, F.; Lanfrancone, M. L.; Brasili, L.; Franchini, S. | |
IDENTIFICATION OF POTENT 1,3-DIOXOLANE-BASED 5-HT1A RECEPTOR AGONISTS FOR THE TREATMENTS OF CNS DISORDERS AND PAIN | 1-gen-2019 | Linciano, Pasquale; Sorbi, Claudia; Franchini, Silvia; Tait, Annalisa; Bardoni, Rita; Ronsisvalle, Simone; Denora, Nunzio; Lesniak, Anna; Bujalska-Zadrożny, Magdalena; Pawłowska, Agata; Chichero, Elena; Fossa, Paola; Brasili, Livio | |
Hits and Lead Discovery in the Identification of New Drugs against the Trypanosomatidic Infections | 1-gen-2019 | Calogeropoulou, Theodora; Magoulas, George E.; Pöhner, Ina; Wade, Rebecca C.; Panecka-Hofman, Joanna; Linciano, Pasquale; Ferrari, Stefania; Costi, Maria Paola; Santarem, Nuno; Dolores Jiménez-Antón, Ma; Isabel Olías-Molero, Ana; Cordeiro da Silva and José María Alunda, Anabela | |
Development of therapeutic agents blocking SOS activation. | 1-gen-2019 | Maso, L.; Bellio, P.; Linciano, P.; D' Acunto, M.; Celenza, G.; Tondi, Donatella; Cendron, L. | |
Effect of the rigidification of propranolol, a mixed β-adrenoceptor and 5-HT1AR antagonist | 1-gen-2019 | Franchini, S.; Sorbi, C.; Linciano, P.; Brasili, L.; Tait, A. | |
Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform | 1-gen-2019 | Moraes, Carolina B.; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Calogeropoulou, Theodora; Prousis, Kyriakos C.; Mangani, Stefano; Di Pisa, Flavio; Landi, Giacomo; Iacono, Lucia Dello; Pozzi, Cecilia; Freitas-Junior, Lucio H.; dos Santos Pascoalino, Bruno; Bertolacini, Claudia P.; Behrens, Birte; Keminer, Oliver; Leu, Jennifer; Wolf, Markus; Reinshagen, Jeanette; Cordeiro-da-Silva, Anabela; Santarem, Nuno; Venturelli, Alberto; Wrigley, Stephen; Karunakaran, Deepa; Kebede, Bethlehem; Pöhner, Ina; Müller, Wolfgang; Panecka-Hofman, Joanna; Wade, Rebecca C.; Fenske, Martina; Clos, Joachim; Alunda, José María; Corral, María Jesús; Uliassi, Elisa; Bolognesi, Maria Laura; Linciano, Pasquale; Quotadamo, Antonio; Ferrari, Stefania; Santucci, Matteo; Borsari, Chiara; Costi, Maria Paola; Gul, Sheraz | |
A novel phytocannabinoid isolated from Cannabis sativa L. with an in vivo cannabimimetic activity higher than Δ9-tetrahydrocannabinol: Δ9-Tetrahydrocannabiphorol | 1-gen-2019 | Citti, C.; Linciano, P.; Russo, F.; Luongo, L.; Iannotta, M.; Maione, S.; Lagana, A.; Capriotti, A. L.; Forni, F.; Vandelli, M. A.; Gigli, G.; Cannazza, G. | |
Analysis of impurities of cannabidiol from hemp. Isolation, characterization and synthesis of cannabidibutol, the novel cannabidiol butyl analog | 1-gen-2019 | Citti, C.; Linciano, P.; Forni, F.; Vandelli, M. A.; Gigli, G.; Lagana, A.; Cannazza, G. | |
Cyclic Peptides Acting as Allosteric Inhibitors of Human Thymidylate Synthase and Cancer Cell Growth | 1-gen-2019 | Pacifico, Salvatore; Santucci, Matteo; Luciani, Rosaria; Saxena, Puneet; Linciano, Pasquale; Ponterini, Glauco; Lauriola, Angela; D'Arca, Domenico; Marverti, Gaetano; Guerrini, Remo; Costi, Maria Paola | |
First virtual screening and experimental validation of inhibitors targeting GES-5 carbapenemase | 1-gen-2019 | Spyrakis, Francesca; Bellio, Pierangelo; Quotadamo, Antonio; Linciano, Pasquale; Benedetti, Paolo; D’Arrigo, Giulia; Baroni, Massimo; Cendron, Laura; Celenza, Giuseppe; Tondi, Donatella | |
Excited-state intramolecular proton transfer in a bioactive flavonoid provides fluorescence observables for recognizing its engagement with target proteins | 1-gen-2019 | Vanossi, D.; Caselli, M.; Pavesi, G.; Borsari, C.; Linciano, P.; Costi, M. P.; Ponterini, G. | |
Optimization of N-alkylation in the Synthesis of Methotrexate and Pteridine-based Derivatives Under Microwave-Irradiation | 1-gen-2019 | Quotadamo, A.; Linciano, P.; Costi, M. P.; Venturelli, A. |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile