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Comparing Drug Images and Repurposing Drugs with BioGPS and FLAPdock: The Thymidylate Synthase Case 1-gen-2016 Siragusa, Lydia; Luciani, Rosaria; Borsari, Chiara; Ferrari, Stefania; Costi, Maria Paola; Cruciani, Gabriele; Spyrakis, Francesca
Virtual Screening and X-ray Crystallography Identify Non-Substrate Analog Inhibitors of Flavin-Dependent Thymidylate Synthase 1-gen-2016 Luciani, Rosaria; Saxena, Puneet; Surade, Sachin; Santucci, Matteo; Venturelli, Alberto; Borsari, Chiara; Marverti, Gaetano; Ponterini, Glauco; Ferrari, Stefania; Blundell, Tom L; Costi, Maria Paola
X-ray crystal structures of Enterococcus faecalis thymidylate synthase with folate binding site inhibitors 1-gen-2016 Catalano, Alessia; Luciani, Rosaria; Carocci, Alessia; Cortesi, Debora; Pozzi, Cecilia; Borsari, Chiara; Ferrari, Stefania; Mangani, Stefano
Scouting new sigma receptor ligands: Synthesis, pharmacological evaluation and molecular modeling of 1,3-dioxolane-based structures and derivatives 1-gen-2016 Franchini, Silvia; Battisti, UMBERTO MARIA; Prandi, Adolfo; Tait, Annalisa; Borsari, Chiara; Cichero, Elena; Fossa, Paola; Cilia, Antonio; Prezzavento, Orazio; Ronsisvalle, Simone; Aricò, Giuseppina; Parenti, Carmela; Brasili, Livio
Profiling of Flavonol Derivatives for the Development of Antitrypanosomatidic Drugs 1-gen-2016 Borsari, Chiara; Luciani, Rosaria; Pozzi, Cecilia; Poehner, Ina; Henrich, Stefan; Trande, Matteo; Cordeiro da Silva, Anabela; Santarem, Nuno; Baptista, Catarina; Tait, Annalisa; Di Pisa, Flavio; Dello, Iacono; Lucia, Landi; Giacomo, ; Gul, Sheraz; Wolf, Markus; Kuzikov, Maria; Ellinger, Bernhard; Reinshagen, Jeanette; Witt, Gesa; Gribbon, Philip; Kohler, Manfred; Keminer, Oliver; Behrens, Birte; Costantino, Luca; Tejera Nevado, Paloma; Bifeld, Eugenia; Eick, Julia; Clos, Joachim; Torrado Santiago, Juan; Jiménez Antón, María D.; Corral, María J.; Alunda, José Ma; Pellati, Federica; Wade, Rebecca C.; Ferrari, Stefania; Mangani, Stefano; Costi, Maria Paola
Crassiflorone derivatives that inhibit Trypanosoma brucei glyceraldehyde-3-phosphate dehydrogenase (TbGAPDH) and Trypanosoma cruzi trypanothione reductase (TcTR) and display trypanocidal activity 1-gen-2017 Uliassi, Elisa; Fiorani, Giulia; Krauth-Siegel, R. Luise; Bergamini, Christian; Fato, Romana; Bianchini, Giulia; Carlos Menéndez, J.; Molina, Maria Teresa; López-Montero, Eulogio; Falchi, Federico; Cavalli, Andrea; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Witt, Gesa; Moraes, Carolina B.; Freitas-Junior, Lucio H.; Borsari, Chiara; Costi, Maria Paola; Bolognesi, Maria Laura
Target-based approaches for the discovery of new antimycobacterial drugs 1-gen-2017 Borsari, Chiara; Ferrari, Stefania; Venturelli, Alberto; Costi, Maria Paola
Methoxylated 2'-hydroxychalcones as antiparasitic hit compounds 1-gen-2017 Borsari, Chiara; Santarem, Nuno; Torrado, Juan; Olías, Ana Isabel; Corral, María Jesús; Baptista, Catarina; Gul, Sheraz; Wolf, Markus; Kuzikov, Maria; Ellinger, Bernhard; Witt, Gesa; Gribbon, Philip; Reinshagen, Jeanette; Linciano, Pasquale; Tait, Annalisa; Costantino, Luca; Freitas-Junior, Lucio H.; Moraes, Carolina B.; Bruno dos Santos, Pascoalino; Alcântara, Laura Maria; Franco, Caio Haddad; Bertolacini, Claudia Danielli; Fontana, Vanessa; Tejera Nevado, Paloma; Clos, Joachim; Alunda, José María; Cordeiro-da-Silva, Anabela; Ferrari, Stefania; Costi, Maria Paola
Development of a Focused Library of Triazole-Linked Privileged-Structure-Based Conjugates Leading to the Discovery of Novel Phenotypic Hits against Protozoan Parasitic Infections 1-gen-2018 Uliassi, Elisa; Piazzi, Lorna; Belluti, Federica; Mazzanti, Andrea; Kaiser, Marcel; Brun, Reto; Moraes, Carolina B; Freitas-Junior, Lucio H; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Borsari, Chiara; Costi, Maria Paola; Bolognesi, Maria Laura
SAR Studies and Biological Characterization of a Chromen-4-one Derivative as an Anti-Trypanosoma brucei Agent 1-gen-2019 Borsari, Chiara; Santarem, Nuno; Macedo, Sara; Jiménez-Antón, María Dolores; Torrado, Juan J.; Olías-Molero, Ana Isabel; Corral, María J.; Tait, Annalisa; Ferrari, Stefania; Costantino, Luca; Luciani, Rosaria; Ponterini, Glauco; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Behrens, Birte; Reinshagen, Jeanette; Alunda, José María; Cordeiro-da-Silva, Anabela; Costi, Maria Paola
Excited-state intramolecular proton transfer in a bioactive flavonoid provides fluorescence observables for recognizing its engagement with target proteins 1-gen-2019 Vanossi, D.; Caselli, M.; Pavesi, G.; Borsari, C.; Linciano, P.; Costi, M. P.; Ponterini, G.
Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform 1-gen-2019 Moraes, Carolina B.; Witt, Gesa; Kuzikov, Maria; Ellinger, Bernhard; Calogeropoulou, Theodora; Prousis, Kyriakos C.; Mangani, Stefano; Di Pisa, Flavio; Landi, Giacomo; Iacono, Lucia Dello; Pozzi, Cecilia; Freitas-Junior, Lucio H.; dos Santos Pascoalino, Bruno; Bertolacini, Claudia P.; Behrens, Birte; Keminer, Oliver; Leu, Jennifer; Wolf, Markus; Reinshagen, Jeanette; Cordeiro-da-Silva, Anabela; Santarem, Nuno; Venturelli, Alberto; Wrigley, Stephen; Karunakaran, Deepa; Kebede, Bethlehem; Pöhner, Ina; Müller, Wolfgang; Panecka-Hofman, Joanna; Wade, Rebecca C.; Fenske, Martina; Clos, Joachim; Alunda, José María; Corral, María Jesús; Uliassi, Elisa; Bolognesi, Maria Laura; Linciano, Pasquale; Quotadamo, Antonio; Ferrari, Stefania; Santucci, Matteo; Borsari, Chiara; Costi, Maria Paola; Gul, Sheraz
Novel Dithiolane-Based Ligands Combining Sigma and NMDA Receptor Interactions as Potential Neuroprotective Agents 1-gen-2020 Franchini, S.; Linciano, P.; Puja, G.; Tait, A.; Borsari, C.; Denora, N.; Iacobazzi, R. M.; Brasili, L.; Sorbi, C.
Mostrati risultati da 1 a 13 di 13
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